JP5957452B2 - 肝臓、肺の障害、糖尿病合併症および心血管疾患の処置のためのジフェニルエーテル化合物 - Google Patents
肝臓、肺の障害、糖尿病合併症および心血管疾患の処置のためのジフェニルエーテル化合物 Download PDFInfo
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- JP5957452B2 JP5957452B2 JP2013521285A JP2013521285A JP5957452B2 JP 5957452 B2 JP5957452 B2 JP 5957452B2 JP 2013521285 A JP2013521285 A JP 2013521285A JP 2013521285 A JP2013521285 A JP 2013521285A JP 5957452 B2 JP5957452 B2 JP 5957452B2
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Classifications
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- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/425—Thiazoles
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- A—HUMAN NECESSITIES
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- A—HUMAN NECESSITIES
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- A—HUMAN NECESSITIES
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- A61P13/12—Drugs for disorders of the urinary system of the kidneys
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- A—HUMAN NECESSITIES
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- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
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- A—HUMAN NECESSITIES
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Landscapes
- Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Medicinal Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
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- Pulmonology (AREA)
- Gynecology & Obstetrics (AREA)
- Pregnancy & Childbirth (AREA)
- Oncology (AREA)
- Emergency Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
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| IN2140CH2010 | 2010-07-28 | ||
| IN2140/CHE/2010 | 2010-07-28 | ||
| IN525/CHE/2011 | 2011-02-23 | ||
| IN525CH2011 | 2011-02-23 | ||
| PCT/IN2011/000210 WO2012014218A1 (en) | 2010-07-28 | 2011-03-28 | Diphenyl ether compounds for the treatment of liver, lung disorders, diabetic complications and cardiovascular diseases |
Publications (3)
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| JP2013532682A JP2013532682A (ja) | 2013-08-19 |
| JP2013532682A5 JP2013532682A5 (enExample) | 2014-05-15 |
| JP5957452B2 true JP5957452B2 (ja) | 2016-07-27 |
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| US (1) | US20140187594A1 (enExample) |
| EP (2) | EP2987488A1 (enExample) |
| JP (1) | JP5957452B2 (enExample) |
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| PL (1) | PL2598142T3 (enExample) |
| WO (1) | WO2012014218A1 (enExample) |
| ZA (1) | ZA201300822B (enExample) |
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| EP3362053A4 (en) * | 2015-10-16 | 2019-04-17 | Hadasit Medical Research Services and Development Ltd. | TREATMENT OF NON-ALCOHOLIC FATTYLENE OR NON-ALCOHOLIC STEATOHEPATITIS WITH 6-MERCAPTOPURIN WITH DELAYED RELEASE |
| TWI762634B (zh) | 2017-05-05 | 2022-05-01 | 大陸商上海赫普化醫藥技術有限公司 | 胺基-芳基-苯甲醯胺化合物及其使用方法 |
| CN113750089B (zh) * | 2021-10-13 | 2023-09-19 | 南方医科大学南方医院 | 2-芳基-1,3二氢苯并咪唑衍生物在制备治疗慢性肝病的药物中的用途 |
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| US7781464B2 (en) * | 2003-01-17 | 2010-08-24 | Bexel Pharmaceuticals, Inc. | Heterocyclic diphenyl ethers |
| US7521465B2 (en) * | 2003-01-17 | 2009-04-21 | Bexel Pharmaceuticals, Inc. | Diphenyl ether derivatives |
| US6794401B2 (en) | 2003-01-17 | 2004-09-21 | Bexel Pharmaceuticals, Inc. | Amino acid phenoxy ethers |
| US7087576B2 (en) * | 2003-10-07 | 2006-08-08 | Bexel Pharmaceuticals, Inc. | Dipeptide phenyl ethers |
| JP2008533122A (ja) * | 2005-03-18 | 2008-08-21 | オーキッド ケミカルズ アンド ファーマシューティカルズ リミテッド | 新規なチロシン誘導体 |
| WO2006138475A2 (en) * | 2005-06-16 | 2006-12-28 | Jenrin Discovery | Mao-b inhibitors useful for treating obesity |
| WO2008106166A2 (en) * | 2007-02-28 | 2008-09-04 | Conatus Pharmaceuticals, Inc. | Methods for the treatment of liver diseases using specified matrix metalloproteinase (mmp) inhibitors |
| JP2010520306A (ja) * | 2007-03-07 | 2010-06-10 | ジヤンセン・フアーマシユーチカ・ナームローゼ・フエンノートシヤツプ | エストロゲン関連受容体−αモジュレーターとしての置換フェノキシチアゾリジンジオン |
| WO2009030968A1 (en) * | 2007-09-05 | 2009-03-12 | Orchid Research Laboratories Limited | Mao a inhibitors with a diphenyl ether-substructure. |
| WO2009070781A1 (en) * | 2007-11-30 | 2009-06-04 | The Regents Of The University Of California | Methods of treating non-alcoholic steatohepatitis (nash) using cysteamine products |
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| AU2011284256B2 (en) | 2014-05-29 |
| CN103108634A (zh) | 2013-05-15 |
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| ES2565487T3 (es) | 2016-04-05 |
| US20140187594A1 (en) | 2014-07-03 |
| AU2011284256A1 (en) | 2013-02-14 |
| AU2011284256B8 (en) | 2014-11-13 |
| WO2012014218A1 (en) | 2012-02-02 |
| CA2805245A1 (en) | 2012-02-02 |
| EP2987488A1 (en) | 2016-02-24 |
| CN103108634B (zh) | 2015-08-12 |
| HUE028725T2 (en) | 2016-12-28 |
| AU2011284256A8 (en) | 2014-11-13 |
| EP2598142B1 (en) | 2015-12-16 |
| EP2598142A1 (en) | 2013-06-05 |
| PL2598142T3 (pl) | 2016-06-30 |
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