JP5855098B2 - 癌の処置のための三環式ラクトン類 - Google Patents
癌の処置のための三環式ラクトン類 Download PDFInfo
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- JP5855098B2 JP5855098B2 JP2013520108A JP2013520108A JP5855098B2 JP 5855098 B2 JP5855098 B2 JP 5855098B2 JP 2013520108 A JP2013520108 A JP 2013520108A JP 2013520108 A JP2013520108 A JP 2013520108A JP 5855098 B2 JP5855098 B2 JP 5855098B2
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D303/00—Compounds containing three-membered rings having one oxygen atom as the only ring hetero atom
- C07D303/02—Compounds containing oxirane rings
- C07D303/38—Compounds containing oxirane rings with hydrocarbon radicals, substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
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- C07—ORGANIC CHEMISTRY
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- C07D303/00—Compounds containing three-membered rings having one oxygen atom as the only ring hetero atom
- C07D303/02—Compounds containing oxirane rings
- C07D303/38—Compounds containing oxirane rings with hydrocarbon radicals, substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
- C07D303/40—Compounds containing oxirane rings with hydrocarbon radicals, substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals by ester radicals
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Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| SE1050815-8 | 2010-07-19 | ||
| SE1050815 | 2010-07-19 | ||
| PCT/EP2011/062243 WO2012010555A1 (en) | 2010-07-19 | 2011-07-18 | Tricyclic lactones for treatment of cancer |
Publications (3)
| Publication Number | Publication Date |
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| JP2013531051A JP2013531051A (ja) | 2013-08-01 |
| JP2013531051A5 JP2013531051A5 (enExample) | 2014-09-04 |
| JP5855098B2 true JP5855098B2 (ja) | 2016-02-09 |
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| JP2013520108A Expired - Fee Related JP5855098B2 (ja) | 2010-07-19 | 2011-07-18 | 癌の処置のための三環式ラクトン類 |
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| US (1) | US9150531B2 (enExample) |
| EP (1) | EP2595972B1 (enExample) |
| JP (1) | JP5855098B2 (enExample) |
| CN (1) | CN103097368B (enExample) |
| ES (1) | ES2553248T3 (enExample) |
| WO (1) | WO2012010555A1 (enExample) |
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| US20150306099A1 (en) * | 2012-11-27 | 2015-10-29 | Glaxosmithkline Llc | Combination |
| US10077246B2 (en) | 2014-03-07 | 2018-09-18 | Glactone Pharma Development Ab | Tricyclic prodrugs |
| JP2016193870A (ja) * | 2015-04-01 | 2016-11-17 | 国立大学法人広島大学 | 慢性骨髄性白血病治療剤 |
| SE539204C2 (en) | 2015-06-05 | 2017-05-09 | Glactone Pharma Dev Ab | Ether analogues of galiellalactone |
| SE540295C2 (en) * | 2016-12-05 | 2018-05-29 | Glactone Pharma Dev Ab | Sulfonamide analogues of galiellalactone |
| CN111297898B (zh) * | 2020-02-18 | 2022-01-25 | 山东大学齐鲁医院 | 间充质干细胞来源的细胞外囊泡在脑缺血再灌注损伤中的应用 |
| CN114507203B (zh) * | 2020-11-17 | 2025-09-30 | 华东理工大学 | 具有抗炎和抗癌活性的倍半萜内酯衍生物及其制备方法和用途 |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CA2414660A1 (en) * | 2000-07-03 | 2002-01-10 | Ibwf Institut Fur Biotechnologie Und Wirkstoff-Forschung E. V. | Use of galiella lactone |
| WO2008135419A2 (en) | 2007-05-04 | 2008-11-13 | Charité Universitätsmedizin Berlin | Anti-il-6-agents for improving primary functioning of allogenic grafts |
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2011
- 2011-07-18 US US13/811,015 patent/US9150531B2/en not_active Expired - Fee Related
- 2011-07-18 CN CN201180035500.3A patent/CN103097368B/zh not_active Expired - Fee Related
- 2011-07-18 JP JP2013520108A patent/JP5855098B2/ja not_active Expired - Fee Related
- 2011-07-18 WO PCT/EP2011/062243 patent/WO2012010555A1/en not_active Ceased
- 2011-07-18 EP EP11739028.6A patent/EP2595972B1/en not_active Not-in-force
- 2011-07-18 ES ES11739028.6T patent/ES2553248T3/es active Active
Also Published As
| Publication number | Publication date |
|---|---|
| ES2553248T3 (es) | 2015-12-07 |
| US9150531B2 (en) | 2015-10-06 |
| JP2013531051A (ja) | 2013-08-01 |
| WO2012010555A1 (en) | 2012-01-26 |
| US20130310451A1 (en) | 2013-11-21 |
| CN103097368A (zh) | 2013-05-08 |
| EP2595972B1 (en) | 2015-08-19 |
| EP2595972A1 (en) | 2013-05-29 |
| CN103097368B (zh) | 2015-08-05 |
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