JP5675598B2 - 胃保持型製剤の製造法 - Google Patents
胃保持型製剤の製造法 Download PDFInfo
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- JP5675598B2 JP5675598B2 JP2011513066A JP2011513066A JP5675598B2 JP 5675598 B2 JP5675598 B2 JP 5675598B2 JP 2011513066 A JP2011513066 A JP 2011513066A JP 2011513066 A JP2011513066 A JP 2011513066A JP 5675598 B2 JP5675598 B2 JP 5675598B2
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- Prior art keywords
- drugs
- hydrochloride
- drug
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- powder
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Images
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
- A61K9/0065—Forms with gastric retention, e.g. floating on gastric juice, adhering to gastric mucosa, expanding to prevent passage through the pylorus
Landscapes
- Health & Medical Sciences (AREA)
- Nutrition Science (AREA)
- Physiology (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Medicinal Preparation (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP08290529A EP2133071A1 (en) | 2008-06-09 | 2008-06-09 | Process for making gastroretentive dosage forms |
| EP08290529.0 | 2008-06-09 | ||
| PCT/IB2009/005889 WO2009150514A1 (en) | 2008-06-09 | 2009-06-08 | Process for making gastroretentive dosage forms |
Related Child Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2014208291A Division JP6054931B2 (ja) | 2008-06-09 | 2014-10-09 | 胃保持型製剤の製造法 |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2011522873A JP2011522873A (ja) | 2011-08-04 |
| JP2011522873A5 JP2011522873A5 (enExample) | 2012-07-19 |
| JP5675598B2 true JP5675598B2 (ja) | 2015-02-25 |
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| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2011513066A Expired - Fee Related JP5675598B2 (ja) | 2008-06-09 | 2009-06-08 | 胃保持型製剤の製造法 |
| JP2014208291A Expired - Fee Related JP6054931B2 (ja) | 2008-06-09 | 2014-10-09 | 胃保持型製剤の製造法 |
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| Application Number | Title | Priority Date | Filing Date |
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| JP2014208291A Expired - Fee Related JP6054931B2 (ja) | 2008-06-09 | 2014-10-09 | 胃保持型製剤の製造法 |
Country Status (7)
| Country | Link |
|---|---|
| US (1) | US9060930B2 (enExample) |
| EP (2) | EP2133071A1 (enExample) |
| JP (2) | JP5675598B2 (enExample) |
| CN (1) | CN102105139B (enExample) |
| CA (1) | CA2727206A1 (enExample) |
| ES (1) | ES2561478T3 (enExample) |
| WO (1) | WO2009150514A1 (enExample) |
Families Citing this family (15)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CA2359812C (en) | 2000-11-20 | 2004-02-10 | The Procter & Gamble Company | Pharmaceutical dosage form with multiple coatings for reduced impact of coating fractures |
| EP2444064A1 (en) | 2010-10-22 | 2012-04-25 | Meliatys | Process for making multiparticulate gastroretentive dosage forms |
| US9119793B1 (en) | 2011-06-28 | 2015-09-01 | Medicis Pharmaceutical Corporation | Gastroretentive dosage forms for doxycycline |
| WO2013114390A1 (en) * | 2012-01-02 | 2013-08-08 | Medreich Limited | Gastro retentive drug delivery system of calcium supplements |
| CN113842362A (zh) | 2012-11-14 | 2021-12-28 | 格雷斯公司 | 含有生物活性材料与无序无机氧化物的组合物 |
| US10842802B2 (en) * | 2013-03-15 | 2020-11-24 | Medicis Pharmaceutical Corporation | Controlled release pharmaceutical dosage forms |
| CN103462917A (zh) * | 2013-09-12 | 2013-12-25 | 南京正宽医药科技有限公司 | 一种用于抗病毒的阿昔洛韦片剂及其制备方法 |
| CN103462926B (zh) * | 2013-09-23 | 2015-09-16 | 淄博齐鼎立专利信息咨询有限公司 | 一种泛昔洛韦片剂及其制备方法 |
| KR20170015389A (ko) | 2014-06-02 | 2017-02-08 | 테바 파마슈티컬 인더스트리즈 리미티드 | 확장 가능한 위체류 투여 형태 |
| US10076494B2 (en) | 2016-06-16 | 2018-09-18 | Dexcel Pharma Technologies Ltd. | Stable orally disintegrating pharmaceutical compositions |
| US10737079B2 (en) | 2016-12-02 | 2020-08-11 | Clexio Biosciences Ltd. | Gastric residence system |
| JP7296084B2 (ja) | 2017-12-04 | 2023-06-22 | クレキシオ バイオサイエンシーズ エルティーディー． | 長時間作用型胃滞留システム |
| AU2018388577B2 (en) * | 2017-12-18 | 2024-06-06 | Tris Pharma, Inc. | Modified release drug powder composition comprising gastro-retentive raft forming systems having trigger pulse drug release |
| CN116459226B (zh) * | 2023-04-26 | 2025-04-18 | 重庆康刻尔制药股份有限公司 | 一种铝碳酸镁双层片及其制备方法 |
| CN118526484A (zh) * | 2024-07-26 | 2024-08-23 | 中国中医科学院中药研究所 | 青蒿琥酯或双氢青蒿素在制备改善罗格列酮不良反应制剂中的应用 |
Family Cites Families (13)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| PL149493B1 (en) | 1985-04-12 | 1990-02-28 | Method of obtaining a tablet capable to buoy over surface of gastric juice | |
| JPS62195323A (ja) * | 1986-02-24 | 1987-08-28 | Eisai Co Ltd | 胃内滞留型粒子 |
| US4814178A (en) | 1987-07-01 | 1989-03-21 | Sanford Bolton | Floating sustained release therapeutic compositions |
| DE3803482A1 (de) | 1988-02-05 | 1989-08-17 | Lohmann Therapie Syst Lts | Schwimmfaehiges orales therapeutisches system |
| US5169638A (en) * | 1991-10-23 | 1992-12-08 | E. R. Squibb & Sons, Inc. | Buoyant controlled release powder formulation |
| PT893992E (pt) * | 1996-04-16 | 2004-06-30 | Novartis Consumer Health Sa | Formas de dosagem oral de desintegracao rapida |
| WO2001058424A1 (en) * | 2000-02-09 | 2001-08-16 | West Pharmaceutical Services Drug Delivery & Clinical Research Centre Limited | Floating drug delivery composition |
| JP2001270827A (ja) * | 2000-03-23 | 2001-10-02 | Eisai Co Ltd | ベンズイミダゾール系化合物含有錠剤 |
| JP2002154948A (ja) * | 2000-11-22 | 2002-05-28 | Eisai Co Ltd | 崩壊性に優れた錠剤 |
| CA2471948A1 (en) * | 2002-01-03 | 2003-07-17 | Smithkline Beecham Corporation | Novel pharmaceutical dosage forms and method for producing same |
| AU2003272069A1 (en) * | 2002-06-26 | 2004-01-19 | Cadila Healthcare Limited | Novel floating dosage form |
| US20070269512A1 (en) * | 2006-05-22 | 2007-11-22 | Wang Wenhua W | Gastroretentive sustained release formulations |
| ES2368356T3 (es) * | 2007-07-06 | 2011-11-16 | Basf Corporation | Composición de retención gástrica basada en un producto de reacción hidrosoluble procedente de un precursor que contiene un grupo vinilo. |
-
2008
- 2008-06-09 EP EP08290529A patent/EP2133071A1/en not_active Withdrawn
-
2009
- 2009-06-08 ES ES09762044.7T patent/ES2561478T3/es active Active
- 2009-06-08 CN CN200980128984.9A patent/CN102105139B/zh not_active Expired - Fee Related
- 2009-06-08 US US12/997,092 patent/US9060930B2/en not_active Expired - Fee Related
- 2009-06-08 EP EP09762044.7A patent/EP2303241B1/en not_active Not-in-force
- 2009-06-08 CA CA2727206A patent/CA2727206A1/en not_active Abandoned
- 2009-06-08 WO PCT/IB2009/005889 patent/WO2009150514A1/en not_active Ceased
- 2009-06-08 JP JP2011513066A patent/JP5675598B2/ja not_active Expired - Fee Related
-
2014
- 2014-10-09 JP JP2014208291A patent/JP6054931B2/ja not_active Expired - Fee Related
Also Published As
| Publication number | Publication date |
|---|---|
| US9060930B2 (en) | 2015-06-23 |
| CN102105139A (zh) | 2011-06-22 |
| CN102105139B (zh) | 2014-12-31 |
| EP2133071A1 (en) | 2009-12-16 |
| US20120021009A1 (en) | 2012-01-26 |
| CA2727206A1 (en) | 2009-12-17 |
| JP6054931B2 (ja) | 2016-12-27 |
| ES2561478T3 (es) | 2016-02-26 |
| EP2303241A1 (en) | 2011-04-06 |
| JP2015007131A (ja) | 2015-01-15 |
| WO2009150514A1 (en) | 2009-12-17 |
| EP2303241B1 (en) | 2015-11-04 |
| JP2011522873A (ja) | 2011-08-04 |
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