JP5657394B2 - 疼痛の治療又は予防方法 - Google Patents
疼痛の治療又は予防方法 Download PDFInfo
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- JP5657394B2 JP5657394B2 JP2010549209A JP2010549209A JP5657394B2 JP 5657394 B2 JP5657394 B2 JP 5657394B2 JP 2010549209 A JP2010549209 A JP 2010549209A JP 2010549209 A JP2010549209 A JP 2010549209A JP 5657394 B2 JP5657394 B2 JP 5657394B2
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- pain
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- C07C233/90—Carboxylic acid amides having nitrogen atoms of carboxamide groups further acylated
- C07C233/91—Carboxylic acid amides having nitrogen atoms of carboxamide groups further acylated with carbon atoms of the carboxamide groups bound to acyclic carbon atoms
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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- A61K31/00—Medicinal preparations containing organic active ingredients
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- A61K31/165—Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F3/00—Compounds containing elements of Groups 2 or 12 of the Periodic Table
- C07F3/003—Compounds containing elements of Groups 2 or 12 of the Periodic Table without C-Metal linkages
Landscapes
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- Chemical Kinetics & Catalysis (AREA)
- Rheumatology (AREA)
- Pain & Pain Management (AREA)
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- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
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| Publication number | Priority date | Publication date | Assignee | Title |
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| JP2013504555A (ja) * | 2009-09-09 | 2013-02-07 | ノヴァレメッド リミテッド | 疼痛の治療又は予防方法 |
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| JP4939396B2 (ja) | 2004-03-26 | 2012-05-23 | ノヴァレメッド リミテッド | Aids及び他のウイルス性疾患及びhiv関連感染症の改善又はその治療用化合物及びそのような化合物を含む組成物、そのような疾患及び感染症の治療方法及びそのような化合物及び組成物の製造方法 |
| GB0804213D0 (en) | 2008-03-06 | 2008-04-16 | New Era Biotech Ltd | A method of printing or preventing pain |
| US8802734B2 (en) | 2009-09-09 | 2014-08-12 | Novaremed Limited | Method of treating or preventing pain |
| GB201116335D0 (en) * | 2011-09-21 | 2011-11-02 | Novaremed Ltd | A method of treating or preventing affective disorders |
| AU2012348529B2 (en) * | 2011-12-08 | 2017-03-30 | Novaremed Ltd. | Isolated stereoisomeric forms of (S) 2-N (3-O-(propan 2-ol) -1-propyl-4-hydroxybenzene) -3-phenylpropylamide |
| SG11202111773QA (en) | 2019-01-23 | 2021-11-29 | Novaremed Ltd | Compounds for use in the treatment or prophylaxis of pain, inflammation and/or autoimmunity |
| EP3939578A1 (en) | 2020-07-13 | 2022-01-19 | Novaremed Ltd. | Compounds for treatment or prevention of an infection resulting from a coronavirus and/or a coronavirus-induced disease |
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| US2908691A (en) * | 1958-07-14 | 1959-10-13 | Searle & Co | Hydroxyphenalkylaminoalkylindoles and ethers corresponding thereto |
| GB1037655A (en) * | 1964-05-20 | 1966-08-03 | Koninklijke Pharma Fab Nv | Di(aralkyl)amines |
| ZA732136B (en) | 1972-04-12 | 1974-03-27 | Lilly Co Eli | Dopamine derivatives |
| JPS5236606A (en) | 1975-09-12 | 1977-03-22 | Tanabe Seiyaku Co Ltd | Process for preparation of amino compounds |
| US4766106A (en) * | 1985-06-26 | 1988-08-23 | Cetus Corporation | Solubilization of proteins for pharmaceutical compositions using polymer conjugation |
| US4908322A (en) * | 1985-09-06 | 1990-03-13 | The United States Of America As Represented By The Department Of Health And Human Services | Derivatization of amines for electrochemical detection |
| US5696270A (en) * | 1989-05-23 | 1997-12-09 | Abbott Laboratories | Intermediate for making retroviral protease inhibiting compounds |
| IS2334B (is) * | 1992-09-08 | 2008-02-15 | Vertex Pharmaceuticals Inc., (A Massachusetts Corporation) | Aspartyl próteasi hemjari af nýjum flokki súlfonamíða |
| JP2848232B2 (ja) | 1993-02-19 | 1999-01-20 | 武田薬品工業株式会社 | アルデヒド誘導体 |
| AU1463997A (en) * | 1995-12-22 | 1997-07-17 | Acea Pharmaceuticals, Inc. | Subtype-selective nmda receptor ligands and the use thereof |
| WO1997029079A1 (en) | 1996-02-06 | 1997-08-14 | Japan Tobacco Inc. | Novel compounds and pharmaceutical use thereof |
| JP2941230B2 (ja) * | 1997-05-06 | 1999-08-25 | コナミ株式会社 | 画像表示処理装置,画像表示処理方法,及びコンピュータプログラムを記録した機械読取り可能な記録媒体 |
| AU2002224139A1 (en) | 2000-12-05 | 2002-06-18 | Nippon Chemiphar Co. Ltd. | Ppar (peroxisome proliferator activated receptor) activators |
| JP4667870B2 (ja) * | 2002-10-03 | 2011-04-13 | ノヴァレメッド リミテッド | 自己免疫疾患、免疫−アレルギー疾患及び臓器又は組織移植拒絶反応の治療において使用する新規な化合物 |
| WO2004047743A2 (en) * | 2002-11-22 | 2004-06-10 | Bristol-Myers Squibb Company | 1-aryl-2-hydroxyethyl amides as potassium channel openers |
| JP4939396B2 (ja) * | 2004-03-26 | 2012-05-23 | ノヴァレメッド リミテッド | Aids及び他のウイルス性疾患及びhiv関連感染症の改善又はその治療用化合物及びそのような化合物を含む組成物、そのような疾患及び感染症の治療方法及びそのような化合物及び組成物の製造方法 |
| DE102004039373A1 (de) * | 2004-08-12 | 2006-02-23 | Grünenthal GmbH | Para-Alkyl-substituierte N-(4-Hydroxy-3-methoxy-benzyl)-zimtsäureamide und deren Verwendung zur Herstellung von Arzneimitteln |
| RU2309144C2 (ru) * | 2005-03-25 | 2007-10-27 | Общество С Ограниченной Ответственностью "Фарминтерпрайсез" | Фенилсодержащие n-ацильные производные аминов, способ их получения, фармацевтическая композиция и их применение в качестве противовоспалительных и анальгетических средств |
| PL2026775T3 (pl) | 2006-05-09 | 2015-12-31 | Novaremed Ltd | Zastosowanie inhibitorów kinazy tyrozynowej Syk w leczeniu komórkowych zaburzeń proliferacyjnych |
| WO2009039218A2 (en) | 2007-09-17 | 2009-03-26 | Chi-Huey Wong | Compositions and methods for treating inflammation and inflammation-related disorders by plectranthus amboinicus extracts |
| GB0804213D0 (en) | 2008-03-06 | 2008-04-16 | New Era Biotech Ltd | A method of printing or preventing pain |
| CN101503370B (zh) | 2009-03-02 | 2012-08-22 | 上海应用技术学院 | 一种n-环丙基-反-2-顺-6-壬二烯酸酰胺的合成方法 |
| CN101503373B (zh) | 2009-03-13 | 2013-07-24 | 山东大学 | 2-氨基-1-(4-硝基苯基)-1-乙醇类金属蛋白酶抑制剂及其制备方法和用途 |
| US8802734B2 (en) * | 2009-09-09 | 2014-08-12 | Novaremed Limited | Method of treating or preventing pain |
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Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2013504555A (ja) * | 2009-09-09 | 2013-02-07 | ノヴァレメッド リミテッド | 疼痛の治療又は予防方法 |
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| AU2009220931A1 (en) | 2009-09-11 |
| EP2323644A2 (en) | 2011-05-25 |
| PL2323644T3 (pl) | 2014-10-31 |
| IL207965A0 (en) | 2010-12-30 |
| AU2009220931B2 (en) | 2014-11-13 |
| WO2009109850A2 (en) | 2009-09-11 |
| GB0804213D0 (en) | 2008-04-16 |
| CA2717692A1 (en) | 2009-09-11 |
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| DK2323644T3 (da) | 2014-07-21 |
| US20110039936A1 (en) | 2011-02-17 |
| WO2009109850A3 (en) | 2009-12-10 |
| CA2717692C (en) | 2016-06-07 |
| US9199917B2 (en) | 2015-12-01 |
| JP2011513377A (ja) | 2011-04-28 |
| IL207965A (en) | 2015-10-29 |
| EP2323644B1 (en) | 2014-04-23 |
| ES2505325T3 (es) | 2014-10-09 |
| US20150080473A1 (en) | 2015-03-19 |
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