JP5256189B2 - Ｍ１受容体で活性を有するベンズイミダゾールおよび医薬におけるその使用 - Google Patents
Ｍ１受容体で活性を有するベンズイミダゾールおよび医薬におけるその使用 Download PDFInfo
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- JP5256189B2 JP5256189B2 JP2009500854A JP2009500854A JP5256189B2 JP 5256189 B2 JP5256189 B2 JP 5256189B2 JP 2009500854 A JP2009500854 A JP 2009500854A JP 2009500854 A JP2009500854 A JP 2009500854A JP 5256189 B2 JP5256189 B2 JP 5256189B2
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- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
- A61P25/34—Tobacco-abuse
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
- A61P25/36—Opioid-abuse
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
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- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Biomedical Technology (AREA)
- Addiction (AREA)
- Psychiatry (AREA)
- Endocrinology (AREA)
- Psychology (AREA)
- Diabetes (AREA)
- Hospice & Palliative Care (AREA)
- Pain & Pain Management (AREA)
- Reproductive Health (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB0605785.5 | 2006-03-22 | ||
| GBGB0605785.5A GB0605785D0 (en) | 2006-03-22 | 2006-03-22 | Compounds |
| PCT/EP2007/052640 WO2007107567A1 (en) | 2006-03-22 | 2007-03-20 | Benzimidazoles which have activity at m1 receptor and their uses in medicine |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2009530348A JP2009530348A (ja) | 2009-08-27 |
| JP2009530348A5 JP2009530348A5 (enExample) | 2010-05-06 |
| JP5256189B2 true JP5256189B2 (ja) | 2013-08-07 |
Family
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Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2009500854A Expired - Fee Related JP5256189B2 (ja) | 2006-03-22 | 2007-03-20 | Ｍ１受容体で活性を有するベンズイミダゾールおよび医薬におけるその使用 |
Country Status (6)
| Country | Link |
|---|---|
| US (1) | US20110207777A1 (enExample) |
| EP (1) | EP1996189B1 (enExample) |
| JP (1) | JP5256189B2 (enExample) |
| ES (1) | ES2395532T3 (enExample) |
| GB (1) | GB0605785D0 (enExample) |
| WO (1) | WO2007107567A1 (enExample) |
Families Citing this family (9)
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| GB0706167D0 (en) * | 2007-03-29 | 2007-05-09 | Glaxo Group Ltd | Compounds |
| GB0706187D0 (en) * | 2007-03-29 | 2007-05-09 | Glaxo Group Ltd | Compounds |
| GB0706168D0 (en) * | 2007-03-29 | 2007-05-09 | Glaxo Group Ltd | Compounds |
| GB0706164D0 (en) * | 2007-03-29 | 2007-05-09 | Glaxo Group Ltd | Compounds |
| GB0706174D0 (en) * | 2007-03-29 | 2007-05-09 | Glaxo Group Ltd | Compounds |
| GB0817982D0 (en) * | 2008-10-01 | 2008-11-05 | Glaxo Group Ltd | Compounds |
| WO2010109468A1 (en) * | 2009-03-26 | 2010-09-30 | Mapi Pharma Hk Limited | Process for the preparation of alogliptin |
| CN110368375B (zh) * | 2019-07-02 | 2021-10-01 | 青岛大学附属医院 | 用于抑郁症及相关病症的缓释组合物及其制备方法 |
| EP4447953A1 (en) | 2021-12-13 | 2024-10-23 | Sage Therapeutics, Inc. | Combination of muscarinic receptor positive modulators and nmda positive allosteric modulators |
Family Cites Families (13)
| Publication number | Priority date | Publication date | Assignee | Title |
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| US5691323A (en) * | 1995-05-12 | 1997-11-25 | Merck & Co., Inc. | Muscarine antagonists |
| EP0786997A4 (en) * | 1994-10-27 | 1998-03-11 | Merck & Co Inc | MUSCARINE ANTAGONISTS |
| US5574044A (en) * | 1994-10-27 | 1996-11-12 | Merck & Co., Inc. | Muscarine antagonists |
| AU7478396A (en) * | 1995-10-31 | 1997-05-22 | Merck & Co., Inc. | Muscarine agonists |
| DE60013464T2 (de) * | 1999-10-13 | 2005-09-15 | Banyu Pharmaceutical Co., Ltd. | Substituierte imidazolin-derivate |
| WO2004089942A2 (en) * | 2001-10-02 | 2004-10-21 | Acadia Pharmaceuticals Inc. | Benzimidazolidinone derivatives as muscarinic agents |
| JP2005532361A (ja) * | 2002-06-17 | 2005-10-27 | メルク エンド カムパニー インコーポレーテッド | 高眼圧症の治療用の眼科用組成物 |
| GB0505304D0 (en) * | 2005-03-15 | 2005-04-20 | Ds Smith Plastics Ltd | Tap for liquid containers |
| WO2007036715A2 (en) * | 2005-09-30 | 2007-04-05 | Glaxo Group Limited | Compounds which have activity at m1 receptor and their uses in medicine |
| US8288413B2 (en) * | 2005-09-30 | 2012-10-16 | Glaxo Group Limited | Benzimidazolones which have activity at M1 receptor |
| GB0605786D0 (en) * | 2006-03-22 | 2006-05-03 | Glaxo Group Ltd | Compounds |
| GB0605784D0 (en) * | 2006-03-22 | 2006-05-03 | Glaxo Group Ltd | Compounds |
| GB0706189D0 (en) * | 2007-03-29 | 2007-05-09 | Glaxo Group Ltd | Compounds |
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2006
- 2006-03-22 GB GBGB0605785.5A patent/GB0605785D0/en not_active Ceased
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2007
- 2007-03-20 ES ES07727117T patent/ES2395532T3/es active Active
- 2007-03-20 JP JP2009500854A patent/JP5256189B2/ja not_active Expired - Fee Related
- 2007-03-20 EP EP07727117A patent/EP1996189B1/en active Active
- 2007-03-20 WO PCT/EP2007/052640 patent/WO2007107567A1/en not_active Ceased
- 2007-03-20 US US12/293,588 patent/US20110207777A1/en not_active Abandoned
Also Published As
| Publication number | Publication date |
|---|---|
| EP1996189A1 (en) | 2008-12-03 |
| JP2009530348A (ja) | 2009-08-27 |
| US20110207777A1 (en) | 2011-08-25 |
| GB0605785D0 (en) | 2006-05-03 |
| ES2395532T3 (es) | 2013-02-13 |
| WO2007107567A1 (en) | 2007-09-27 |
| EP1996189B1 (en) | 2012-09-26 |
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