JP5021155B2 - エピナスチンと１種以上のさらなる抗−ｈ１−ヒスタミン類との組合せを含む皮膚疾患治療用製薬組成物 - Google Patents
エピナスチンと１種以上のさらなる抗−ｈ１−ヒスタミン類との組合せを含む皮膚疾患治療用製薬組成物 Download PDFInfo
- Publication number
- JP5021155B2 JP5021155B2 JP2004223680A JP2004223680A JP5021155B2 JP 5021155 B2 JP5021155 B2 JP 5021155B2 JP 2004223680 A JP2004223680 A JP 2004223680A JP 2004223680 A JP2004223680 A JP 2004223680A JP 5021155 B2 JP5021155 B2 JP 5021155B2
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- JP
- Japan
- Prior art keywords
- epinastine
- pharmaceutical composition
- range
- pharmaceutically acceptable
- oral
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Lifetime
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- WHWZLSFABNNENI-UHFFFAOYSA-N epinastine Chemical compound C1C2=CC=CC=C2C2CN=C(N)N2C2=CC=CC=C21 WHWZLSFABNNENI-UHFFFAOYSA-N 0.000 title claims abstract description 57
- 229960003449 epinastine Drugs 0.000 title claims abstract description 40
- 208000017520 skin disease Diseases 0.000 title claims abstract description 31
- 239000008194 pharmaceutical composition Substances 0.000 title claims abstract description 28
- 150000003839 salts Chemical class 0.000 claims abstract description 28
- 239000002552 dosage form Substances 0.000 claims abstract description 22
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- 239000003826 tablet Substances 0.000 claims description 29
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- 229960002548 epinastine hydrochloride Drugs 0.000 claims description 16
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- ZZVUWRFHKOJYTH-UHFFFAOYSA-N diphenhydramine Chemical compound C=1C=CC=CC=1C(OCCN(C)C)C1=CC=CC=C1 ZZVUWRFHKOJYTH-UHFFFAOYSA-N 0.000 claims description 8
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Landscapes
- Medicinal Preparation (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
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| Application Number | Priority Date | Filing Date | Title |
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| EP03016681 | 2003-08-01 | ||
| EP03016681.3 | 2003-08-01 |
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| JP2005053907A JP2005053907A (ja) | 2005-03-03 |
| JP2005053907A5 JP2005053907A5 (https=) | 2007-09-13 |
| JP5021155B2 true JP5021155B2 (ja) | 2012-09-05 |
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|---|---|---|---|---|
| WO2008148573A2 (de) * | 2007-06-08 | 2008-12-11 | Bayer Consumer Care Ag | Arzeimittel mit einer wirkstoffkombination enthaltend pantothensäure oder deren derivate zur behandlung von allergischen symptomen |
| JP2019043853A (ja) * | 2017-08-30 | 2019-03-22 | 旭化成株式会社 | 経皮吸収促進剤、経皮吸収促進助剤、及び経皮製剤 |
| WO2022138826A1 (ja) * | 2020-12-24 | 2022-06-30 | 参天製薬株式会社 | エピナスチン又はその塩を含有する塗布投与用医薬組成物 |
| CN116744904A (zh) * | 2020-12-24 | 2023-09-12 | 参天制药株式会社 | 含有依匹斯汀或其盐和硫系抗氧化剂的经皮施予用医药组合物 |
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| JP4563522B2 (ja) * | 1999-02-19 | 2010-10-13 | 豊也 加藤 | アレルギー疾患治療剤 |
| PE20020324A1 (es) * | 2000-10-06 | 2002-06-18 | Boehringer Ingelheim Int | Nuevas composiciones farmaceuticas que contienen epinastina y pseudoefedrina |
| US6827946B2 (en) * | 2001-12-05 | 2004-12-07 | Collegium Pharmaceutical, Inc. | Compositions containing both sedative and non-sedative antihistamines |
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