JP4738172B2 - 抗感染薬 - Google Patents
抗感染薬 Download PDFInfo
- Publication number
- JP4738172B2 JP4738172B2 JP2005502238A JP2005502238A JP4738172B2 JP 4738172 B2 JP4738172 B2 JP 4738172B2 JP 2005502238 A JP2005502238 A JP 2005502238A JP 2005502238 A JP2005502238 A JP 2005502238A JP 4738172 B2 JP4738172 B2 JP 4738172B2
- Authority
- JP
- Japan
- Prior art keywords
- alkyl
- group
- alkenyl
- oxo
- hydroxy
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Fee Related
Links
- 0 C*c1c(C)[s]cc1* Chemical compound C*c1c(C)[s]cc1* 0.000 description 6
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/62—Oxygen or sulfur atoms
- C07D213/69—Two or more oxygen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
- C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
- C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D215/20—Oxygen atoms
- C07D215/22—Oxygen atoms attached in position 2 or 4
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
- C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D495/04—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
- C07D513/04—Ortho-condensed systems
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Saccharide Compounds (AREA)
- Pyridine Compounds (AREA)
- Quinoline Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Hydrogenated Pyridines (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
- Micro-Organisms Or Cultivation Processes Thereof (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Applications Claiming Priority (9)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US10/285,714 US20040097492A1 (en) | 2002-11-01 | 2002-11-01 | Anti-infective agents |
US10/285,714 | 2002-11-01 | ||
US10/410,853 US20040087577A1 (en) | 2002-11-01 | 2003-04-10 | Anti-infective agents |
US10/410,853 | 2003-04-10 | ||
US10/625,121 US20040162285A1 (en) | 2002-11-01 | 2003-07-23 | Anti-infective agents |
US10/625,121 | 2003-07-23 | ||
US10/679,881 | 2003-10-06 | ||
US10/679,881 US20050075331A1 (en) | 2003-10-06 | 2003-10-06 | Anti-infective agents |
PCT/US2003/034707 WO2004041818A1 (en) | 2002-11-01 | 2003-10-31 | Anti-infective agents |
Related Child Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
JP2011033491A Division JP5250649B2 (ja) | 2002-11-01 | 2011-02-18 | 抗感染薬 |
Publications (2)
Publication Number | Publication Date |
---|---|
JP2006509042A JP2006509042A (ja) | 2006-03-16 |
JP4738172B2 true JP4738172B2 (ja) | 2011-08-03 |
Family
ID=43426110
Family Applications (2)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
JP2005502238A Expired - Fee Related JP4738172B2 (ja) | 2002-11-01 | 2003-10-31 | 抗感染薬 |
JP2011033491A Expired - Fee Related JP5250649B2 (ja) | 2002-11-01 | 2011-02-18 | 抗感染薬 |
Family Applications After (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
JP2011033491A Expired - Fee Related JP5250649B2 (ja) | 2002-11-01 | 2011-02-18 | 抗感染薬 |
Country Status (6)
Country | Link |
---|---|
JP (2) | JP4738172B2 (de) |
AT (1) | ATE493408T1 (de) |
DE (1) | DE60335564D1 (de) |
DK (1) | DK1560827T3 (de) |
PT (1) | PT1560827E (de) |
SI (1) | SI1560827T1 (de) |
Families Citing this family (7)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
UA100120C2 (en) | 2007-04-03 | 2012-11-26 | Анадис Фармасьютикалз, Инк. | 5,6-dihydro-1h-pyridin-2-one compounds |
GB0800855D0 (en) * | 2008-01-17 | 2008-02-27 | Syngenta Ltd | Herbicidal compounds |
US20090257979A1 (en) * | 2008-04-15 | 2009-10-15 | Intermune, Inc. | Novel Inhibitors of Hepatitis C Virus Replication |
BRPI0919652A2 (pt) * | 2008-10-29 | 2015-08-18 | Basf Se | Compostos de piridina, agente, e, processo para combater vegetação indesejada |
TW201035083A (en) * | 2009-03-06 | 2010-10-01 | Hoffmann La Roche | Heterocyclic antiviral compounds |
JP2013525368A (ja) * | 2010-04-23 | 2013-06-20 | キネタ・インコーポレイテツド | 抗ウイルス性化合物 |
EP2718273A4 (de) * | 2011-06-07 | 2014-12-10 | Anadys Pharmaceuticals Inc | [1,2,4]-thiadiazin-1,1-dioxidverbindungen zur senkung des harnsäurespiegels im serum |
Citations (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO2001085172A1 (en) * | 2000-05-10 | 2001-11-15 | Smithkline Beecham Corporation | Novel anti-infectives |
WO2002098424A1 (en) * | 2001-06-07 | 2002-12-12 | Smithkline Beecham Corporation | Novel anti-infectives |
Family Cites Families (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
AU2002365198A1 (en) * | 2001-10-30 | 2003-07-30 | Smithkline Beecham Corporation | Novel anti-infectives |
-
2003
- 2003-10-31 DE DE60335564T patent/DE60335564D1/de not_active Expired - Lifetime
- 2003-10-31 PT PT03768559T patent/PT1560827E/pt unknown
- 2003-10-31 DK DK03768559.1T patent/DK1560827T3/da active
- 2003-10-31 AT AT03768559T patent/ATE493408T1/de active
- 2003-10-31 SI SI200331953T patent/SI1560827T1/sl unknown
- 2003-10-31 JP JP2005502238A patent/JP4738172B2/ja not_active Expired - Fee Related
-
2011
- 2011-02-18 JP JP2011033491A patent/JP5250649B2/ja not_active Expired - Fee Related
Patent Citations (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO2001085172A1 (en) * | 2000-05-10 | 2001-11-15 | Smithkline Beecham Corporation | Novel anti-infectives |
WO2002098424A1 (en) * | 2001-06-07 | 2002-12-12 | Smithkline Beecham Corporation | Novel anti-infectives |
Also Published As
Publication number | Publication date |
---|---|
DK1560827T3 (da) | 2011-04-18 |
JP5250649B2 (ja) | 2013-07-31 |
JP2011144183A (ja) | 2011-07-28 |
PT1560827E (pt) | 2011-03-17 |
SI1560827T1 (sl) | 2011-04-29 |
ATE493408T1 (de) | 2011-01-15 |
DE60335564D1 (de) | 2011-02-10 |
JP2006509042A (ja) | 2006-03-16 |
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