JP4616000B2 - 二環式オリゴペプチド及びグルカゴン受容体アンタゴニストとしてのその使用 - Google Patents
二環式オリゴペプチド及びグルカゴン受容体アンタゴニストとしてのその使用 Download PDFInfo
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- JP4616000B2 JP4616000B2 JP2004520641A JP2004520641A JP4616000B2 JP 4616000 B2 JP4616000 B2 JP 4616000B2 JP 2004520641 A JP2004520641 A JP 2004520641A JP 2004520641 A JP2004520641 A JP 2004520641A JP 4616000 B2 JP4616000 B2 JP 4616000B2
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Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K7/00—Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
- C07K7/50—Cyclic peptides containing at least one abnormal peptide link
- C07K7/54—Cyclic peptides containing at least one abnormal peptide link with at least one abnormal peptide link in the ring
- C07K7/56—Cyclic peptides containing at least one abnormal peptide link with at least one abnormal peptide link in the ring the cyclisation not occurring through 2,4-diamino-butanoic acid
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/18—Drugs for disorders of the alimentary tract or the digestive system for pancreatic disorders, e.g. pancreatic enzymes
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/12—Drugs for disorders of the urinary system of the kidneys
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/04—Anorexiants; Antiobesity agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/06—Antihyperlipidemics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/48—Drugs for disorders of the endocrine system of the pancreatic hormones
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K14/00—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
- C07K14/195—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from bacteria
- C07K14/36—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from bacteria from Actinomyces; from Streptomyces (G)
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Medicinal Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Veterinary Medicine (AREA)
- General Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Diabetes (AREA)
- Obesity (AREA)
- Heart & Thoracic Surgery (AREA)
- Cardiology (AREA)
- Hematology (AREA)
- Urology & Nephrology (AREA)
- Genetics & Genomics (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Molecular Biology (AREA)
- Endocrinology (AREA)
- Biochemistry (AREA)
- Biophysics (AREA)
- Emergency Medicine (AREA)
- Child & Adolescent Psychology (AREA)
- Vascular Medicine (AREA)
- Gastroenterology & Hepatology (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Medicines Containing Material From Animals Or Micro-Organisms (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Peptides Or Proteins (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP02015907 | 2002-07-17 | ||
| PCT/EP2003/007657 WO2004007535A1 (en) | 2002-07-17 | 2003-07-15 | Bicyclic oligopeptides and their use as glucagon receptor antagonists |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2006505507A JP2006505507A (ja) | 2006-02-16 |
| JP2006505507A5 JP2006505507A5 (cg-RX-API-DMAC10.html) | 2006-09-07 |
| JP4616000B2 true JP4616000B2 (ja) | 2011-01-19 |
Family
ID=30011078
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2004520641A Expired - Fee Related JP4616000B2 (ja) | 2002-07-17 | 2003-07-15 | 二環式オリゴペプチド及びグルカゴン受容体アンタゴニストとしてのその使用 |
Country Status (8)
| Country | Link |
|---|---|
| EP (1) | EP1525218B1 (cg-RX-API-DMAC10.html) |
| JP (1) | JP4616000B2 (cg-RX-API-DMAC10.html) |
| AT (1) | ATE415415T1 (cg-RX-API-DMAC10.html) |
| AU (2) | AU2003260306A1 (cg-RX-API-DMAC10.html) |
| CA (1) | CA2489189A1 (cg-RX-API-DMAC10.html) |
| DE (1) | DE60324936D1 (cg-RX-API-DMAC10.html) |
| ES (1) | ES2316820T3 (cg-RX-API-DMAC10.html) |
| WO (2) | WO2004007524A2 (cg-RX-API-DMAC10.html) |
Families Citing this family (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB0917072D0 (en) | 2009-09-29 | 2009-11-11 | Univ Ulster | Peptide analogues of glucagon for diabetes therapy |
| SG11201407316QA (en) * | 2012-05-08 | 2014-12-30 | Cellix Bio Private Ltd | Compositions and methods for the treatment of hyperglycemia |
Family Cites Families (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4139526A (en) * | 1977-12-01 | 1979-02-13 | Merck & Co., Inc. | Somatostatin analogs |
-
2003
- 2003-07-08 WO PCT/EP2003/007311 patent/WO2004007524A2/en not_active Ceased
- 2003-07-08 AU AU2003260306A patent/AU2003260306A1/en not_active Abandoned
- 2003-07-15 WO PCT/EP2003/007657 patent/WO2004007535A1/en not_active Ceased
- 2003-07-15 DE DE60324936T patent/DE60324936D1/de not_active Expired - Lifetime
- 2003-07-15 EP EP03763864A patent/EP1525218B1/en not_active Expired - Lifetime
- 2003-07-15 AU AU2003246702A patent/AU2003246702A1/en not_active Abandoned
- 2003-07-15 JP JP2004520641A patent/JP4616000B2/ja not_active Expired - Fee Related
- 2003-07-15 ES ES03763864T patent/ES2316820T3/es not_active Expired - Lifetime
- 2003-07-15 CA CA002489189A patent/CA2489189A1/en not_active Abandoned
- 2003-07-15 AT AT03763864T patent/ATE415415T1/de active
Also Published As
| Publication number | Publication date |
|---|---|
| JP2006505507A (ja) | 2006-02-16 |
| DE60324936D1 (de) | 2009-01-08 |
| ATE415415T1 (de) | 2008-12-15 |
| CA2489189A1 (en) | 2004-01-22 |
| ES2316820T3 (es) | 2009-04-16 |
| AU2003260306A1 (en) | 2004-02-02 |
| WO2004007524A2 (en) | 2004-01-22 |
| EP1525218A1 (en) | 2005-04-27 |
| WO2004007535A1 (en) | 2004-01-22 |
| EP1525218B1 (en) | 2008-11-26 |
| AU2003246702A1 (en) | 2004-02-02 |
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