JP4603528B2 - 選択的アンドロゲン受容体の大規模合成 - Google Patents
選択的アンドロゲン受容体の大規模合成 Download PDFInfo
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- JP4603528B2 JP4603528B2 JP2006500896A JP2006500896A JP4603528B2 JP 4603528 B2 JP4603528 B2 JP 4603528B2 JP 2006500896 A JP2006500896 A JP 2006500896A JP 2006500896 A JP2006500896 A JP 2006500896A JP 4603528 B2 JP4603528 B2 JP 4603528B2
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Classifications
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- C07C231/00—Preparation of carboxylic acid amides
- C07C231/12—Preparation of carboxylic acid amides by reactions not involving the formation of carboxamide groups
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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- A61P15/10—Drugs for genital or sexual disorders; Contraceptives for impotence
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- A61P17/14—Drugs for dermatological disorders for baldness or alopecia
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/08—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
- A61P19/10—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease for osteoporosis
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- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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Landscapes
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- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Animal Behavior & Ethology (AREA)
- Veterinary Medicine (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
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- Engineering & Computer Science (AREA)
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- Biomedical Technology (AREA)
- Psychiatry (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Steroid Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US43941603P | 2003-01-13 | 2003-01-13 | |
| PCT/US2004/000618 WO2004062612A2 (fr) | 2003-01-13 | 2004-01-12 | Synthese a grande echelle de modulateurs selectifs de recepteur d'androgene |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2006516033A JP2006516033A (ja) | 2006-06-15 |
| JP4603528B2 true JP4603528B2 (ja) | 2010-12-22 |
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| Application Number | Title | Priority Date | Filing Date |
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| JP2006500896A Expired - Fee Related JP4603528B2 (ja) | 2003-01-13 | 2004-01-12 | 選択的アンドロゲン受容体の大規模合成 |
Country Status (15)
| Country | Link |
|---|---|
| US (1) | US7968721B2 (fr) |
| EP (2) | EP1592658B1 (fr) |
| JP (1) | JP4603528B2 (fr) |
| CN (1) | CN1826313B (fr) |
| AU (1) | AU2004204800B8 (fr) |
| CA (1) | CA2513242C (fr) |
| CY (1) | CY1114156T1 (fr) |
| DK (1) | DK1592658T3 (fr) |
| ES (1) | ES2420129T3 (fr) |
| HK (1) | HK1082724A1 (fr) |
| IL (1) | IL169581A0 (fr) |
| MX (1) | MXPA05007536A (fr) |
| PT (1) | PT1592658E (fr) |
| TW (2) | TW201139345A (fr) |
| WO (1) | WO2004062612A2 (fr) |
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| US7759520B2 (en) * | 1996-11-27 | 2010-07-20 | University Of Tennessee Research Foundation | Synthesis of selective androgen receptor modulators |
| US7855229B2 (en) * | 2000-08-24 | 2010-12-21 | University Of Tennessee Research Foundation | Treating wasting disorders with selective androgen receptor modulators |
| US8445534B2 (en) | 2000-08-24 | 2013-05-21 | University Of Tennessee Research Foundation | Treating androgen decline in aging male (ADAM)-associated conditions with SARMs |
| US7645898B2 (en) * | 2000-08-24 | 2010-01-12 | University Of Tennessee Research Foundation | Selective androgen receptor modulators and method of use thereof |
| US20060019931A1 (en) * | 2003-10-14 | 2006-01-26 | Dalton James T | Treating bone-related disorders with selective androgen receptor modulators |
| US7622503B2 (en) | 2000-08-24 | 2009-11-24 | University Of Tennessee Research Foundation | Selective androgen receptor modulators and methods of use thereof |
| US7919647B2 (en) | 2000-08-24 | 2011-04-05 | University Of Tennessee Research Foundation | Selective androgen receptor modulators and methods of use thereof |
| US20070161608A1 (en) * | 2001-12-06 | 2007-07-12 | Dalton James T | Selective androgen receptor modulators for treating muscle wasting |
| US8853266B2 (en) * | 2001-12-06 | 2014-10-07 | University Of Tennessee Research Foundation | Selective androgen receptor modulators for treating diabetes |
| AU2003287077B2 (en) * | 2002-10-15 | 2007-09-20 | University Of Tennessee Research Foundation | Methylene-bridged selective androgen receptor modulators and methods of use thereof |
| FI20030958A0 (fi) * | 2003-06-27 | 2003-06-27 | Orion Corp | Uusia yhdisteitä |
| CN1805921A (zh) * | 2003-12-16 | 2006-07-19 | Gtx公司 | 选择性雄激素受体调节剂的前药及其使用方法 |
| US9884038B2 (en) | 2004-06-07 | 2018-02-06 | University Of Tennessee Research Foundation | Selective androgen receptor modulator and methods of use thereof |
| US9889110B2 (en) | 2004-06-07 | 2018-02-13 | University Of Tennessee Research Foundation | Selective androgen receptor modulator for treating hormone-related conditions |
| WO2007001448A2 (fr) | 2004-11-04 | 2007-01-04 | Massachusetts Institute Of Technology | Particules polymeres revetues a diffusion regulee comme vecteurs efficaces d'administration par voie orale de produits biopharmaceutiques |
| WO2007070682A2 (fr) | 2005-12-15 | 2007-06-21 | Massachusetts Institute Of Technology | Systeme de criblage de particules |
| WO2008105773A2 (fr) | 2006-03-31 | 2008-09-04 | Massachusetts Institute Of Technology | Système pour l'administration ciblée d'agents thérapeutiques |
| CA2652280C (fr) | 2006-05-15 | 2014-01-28 | Massachusetts Institute Of Technology | Polymeres pour particules fonctionnelles |
| US8288366B2 (en) | 2006-06-20 | 2012-10-16 | Chochinov Ronald H | Formulation for hair growth |
| WO2007150030A2 (fr) | 2006-06-23 | 2007-12-27 | Massachusetts Institute Of Technology | Synthèse microfluidique de nanoparticules organiques |
| US9217129B2 (en) | 2007-02-09 | 2015-12-22 | Massachusetts Institute Of Technology | Oscillating cell culture bioreactor |
| WO2008124634A1 (fr) | 2007-04-04 | 2008-10-16 | Massachusetts Institute Of Technology | Micelles inverses encapsulées par un polymère |
| US20090074828A1 (en) | 2007-04-04 | 2009-03-19 | Massachusetts Institute Of Technology | Poly(amino acid) targeting moieties |
| US7968603B2 (en) | 2007-09-11 | 2011-06-28 | University Of Tennessee Research Foundation | Solid forms of selective androgen receptor modulators |
| EA018611B1 (ru) * | 2007-09-11 | 2013-09-30 | ДЖиТиЭкс, ИНК. | Твердые формы селективных модуляторов рецепторов андрогена |
| EP2644192B1 (fr) | 2007-09-28 | 2017-05-10 | Pfizer Inc | Ciblage de cellules de cancer utilisant des nanoparticules |
| MX350501B (es) | 2007-10-12 | 2017-09-07 | Massachusetts Inst Technology | Nanotecnologia de vacuna. |
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|---|---|
| US7968721B2 (en) | 2011-06-28 |
| CY1114156T1 (el) | 2016-08-31 |
| WO2004062612A2 (fr) | 2004-07-29 |
| IL169581A0 (en) | 2007-07-04 |
| CN1826313A (zh) | 2006-08-30 |
| CN1826313B (zh) | 2010-12-08 |
| EP2457892A1 (fr) | 2012-05-30 |
| AU2004204800B2 (en) | 2011-05-12 |
| US20040260092A1 (en) | 2004-12-23 |
| MXPA05007536A (es) | 2005-10-20 |
| EP1592658A4 (fr) | 2006-11-29 |
| DK1592658T3 (da) | 2013-07-29 |
| AU2004204800A2 (en) | 2004-07-29 |
| AU2004204800A1 (en) | 2004-07-29 |
| TW200512180A (en) | 2005-04-01 |
| TW201139345A (en) | 2011-11-16 |
| WO2004062612A3 (fr) | 2004-11-04 |
| EP1592658A2 (fr) | 2005-11-09 |
| TWI351395B (en) | 2011-11-01 |
| ES2420129T3 (es) | 2013-08-22 |
| CA2513242C (fr) | 2013-07-09 |
| EP1592658B1 (fr) | 2013-04-24 |
| JP2006516033A (ja) | 2006-06-15 |
| HK1082724A1 (en) | 2006-06-16 |
| CA2513242A1 (fr) | 2004-07-29 |
| AU2004204800B8 (en) | 2011-05-26 |
| PT1592658E (pt) | 2013-06-25 |
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