JP4426301B2 - オレフィンのアリール化法 - Google Patents

オレフィンのアリール化法 Download PDF

Info

Publication number
JP4426301B2
JP4426301B2 JP2003549300A JP2003549300A JP4426301B2 JP 4426301 B2 JP4426301 B2 JP 4426301B2 JP 2003549300 A JP2003549300 A JP 2003549300A JP 2003549300 A JP2003549300 A JP 2003549300A JP 4426301 B2 JP4426301 B2 JP 4426301B2
Authority
JP
Japan
Prior art keywords
alkyl
aryl
group
general formula
palladium
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Fee Related
Application number
JP2003549300A
Other languages
English (en)
Japanese (ja)
Other versions
JP2005511682A5 (enExample
JP2005511682A (ja
Inventor
ラムプフ フローリアン
エッケルト マルクス
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Lanxess Deutschland GmbH
Original Assignee
Lanxess Deutschland GmbH
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lanxess Deutschland GmbH filed Critical Lanxess Deutschland GmbH
Publication of JP2005511682A publication Critical patent/JP2005511682A/ja
Publication of JP2005511682A5 publication Critical patent/JP2005511682A5/ja
Application granted granted Critical
Publication of JP4426301B2 publication Critical patent/JP4426301B2/ja
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C231/00—Preparation of carboxylic acid amides
    • C07C231/12—Preparation of carboxylic acid amides by reactions not involving the formation of carboxamide groups
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B37/00—Reactions without formation or introduction of functional groups containing hetero atoms, involving either the formation of a carbon-to-carbon bond between two carbon atoms not directly linked already or the disconnection of two directly linked carbon atoms
    • C07B37/04—Substitution
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C2531/00—Catalysts comprising hydrides, coordination complexes or organic compounds
    • C07C2531/16—Catalysts comprising hydrides, coordination complexes or organic compounds containing coordination complexes
    • C07C2531/24—Phosphines

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
JP2003549300A 2001-12-03 2002-11-20 オレフィンのアリール化法 Expired - Fee Related JP4426301B2 (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE10159269A DE10159269A1 (de) 2001-12-03 2001-12-03 Arylierung von Olefinen
PCT/EP2002/012994 WO2003048107A1 (de) 2001-12-03 2002-11-20 Arylierung von olefinen

Publications (3)

Publication Number Publication Date
JP2005511682A JP2005511682A (ja) 2005-04-28
JP2005511682A5 JP2005511682A5 (enExample) 2006-01-05
JP4426301B2 true JP4426301B2 (ja) 2010-03-03

Family

ID=7707838

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2003549300A Expired - Fee Related JP4426301B2 (ja) 2001-12-03 2002-11-20 オレフィンのアリール化法

Country Status (7)

Country Link
US (1) US6858756B2 (enExample)
EP (1) EP1467963A1 (enExample)
JP (1) JP4426301B2 (enExample)
AU (1) AU2002358519A1 (enExample)
DE (1) DE10159269A1 (enExample)
IL (1) IL162238A0 (enExample)
WO (1) WO2003048107A1 (enExample)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN1890253A (zh) * 2003-12-12 2007-01-03 索尔维亚斯股份公司 制备邻位金属化和邻位取代芳族化合物的方法
WO2005123662A1 (en) * 2004-06-18 2005-12-29 Janssen Pharmaceutica N.V. Modified heck reaction
US8193182B2 (en) 2008-01-04 2012-06-05 Intellikine, Inc. Substituted isoquinolin-1(2H)-ones, and methods of use thereof
DK2240451T3 (da) 2008-01-04 2017-11-20 Intellikine Llc Isoquinolinonderivater substitueret med en purin, der er anvendelig som pi3k-inhibitorer
PE20180318A1 (es) 2011-01-10 2018-02-09 Infinity Pharmaceuticals Inc Procedimiento para preparar isoquinolinonas y formas solidas de isoquinolinonas
TW201238603A (en) 2011-03-10 2012-10-01 Lonza Ag Method for preparation of 3-(2,3-dimethylphenyl)-2-butenal
US8828998B2 (en) 2012-06-25 2014-09-09 Infinity Pharmaceuticals, Inc. Treatment of lupus, fibrotic conditions, and inflammatory myopathies and other disorders using PI3 kinase inhibitors
LT2914296T (lt) 2012-11-01 2018-09-25 Infinity Pharmaceuticals, Inc. Vėžio gydymas, panaudojant p13 kinazės izoformos moduliatorius
US20150320755A1 (en) 2014-04-16 2015-11-12 Infinity Pharmaceuticals, Inc. Combination therapies
UA125216C2 (uk) 2016-06-24 2022-02-02 Інфініті Фармасьютікалз, Інк. Комбінована терапія
CN114085300B (zh) * 2021-12-24 2023-09-15 南亚新材料科技股份有限公司 改性聚丁二烯树脂及其制备方法、应用

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3922299A (en) * 1974-03-05 1975-11-25 Univ Delaware Vinylic substitution reactions
CH654286A5 (de) * 1981-11-04 1986-02-14 Ciba Geigy Ag Verfahren zur pd-katalysierten arylierung von olefinen mit arylhalogeniden.
DE19825454A1 (de) * 1998-06-06 1999-12-16 Aventis Res & Tech Gmbh & Co Verfahren zur Herstellung von aromatischen Olefinen unter Katalyse von Palladiumkatalysatoren mit Phosphitliganden

Also Published As

Publication number Publication date
EP1467963A1 (de) 2004-10-20
AU2002358519A1 (en) 2003-06-17
JP2005511682A (ja) 2005-04-28
IL162238A0 (en) 2005-11-20
WO2003048107A1 (de) 2003-06-12
DE10159269A1 (de) 2003-06-18
US6858756B2 (en) 2005-02-22
US20030114707A1 (en) 2003-06-19

Similar Documents

Publication Publication Date Title
O’Keefe et al. Carbonylative cross-coupling of ortho-disubstituted aryl iodides. convenient synthesis of sterically hindered aryl ketones
Sain et al. Application of palladium-catalyzed cross-coupling reactions in organic synthesis
Tlili et al. Ruthenium-Catalyzed Carbonylative C C Coupling in Water by Directed C H Bond Activation.
Fu et al. Decarboxylative halogenation and cyanation of electron-deficient aryl carboxylic acids via Cu mediator as well as electron-rich ones through Pd catalyst under aerobic conditions
Cong et al. Role of mono-N-protected amino acid ligands in palladium (II)-catalyzed dehydrogenative Heck reactions of electron-deficient (hetero) arenes: experimental and computational studies
JP4426301B2 (ja) オレフィンのアリール化法
Serrano et al. N-heterocyclic-carbene complexes readily prepared from di-μ-hydroxopalladacycles catalyze the Suzuki arylation of 9-bromophenanthrene
Rahman et al. Pd–PEPPSI N-heterocyclic carbene complexes from caffeine: application in Suzuki, Heck, and Sonogashira reactions
RU2324678C2 (ru) Способ получения динитрилов фенилмалоновой кислоты
Ilies et al. Iron-catalyzed directed alkylation of carboxamides with olefins via a carbometalation pathway
EP1185506A1 (en) Substituted arylmalonic acid dinitriles as intermediates for the preparation of herbicides
Kumandin et al. Influence of the N→ Ru coordinate bond length on the activity of new types of hoveyda–grubbs olefin metathesis catalysts containing a six-membered chelate ring possessing a ruthenium–nitrogen bond
Chen et al. Metal-free intramolecular carbocyanation of activated alkenes: functionalized nitriles bearing β-quaternary carbon centers.
JP4386729B2 (ja) オレフィンのアリール化法
Graßl et al. Preparation of Tertiary Amines from Tris (2-cyanoethyl) amine Using Three Successive Cobalt-Catalyzed Electrophilic Aminations with Organozinc Halides
Wakuluk-Machado et al. Pd (OH) 2/C, a practical and efficient catalyst for the carboxylation of benzylic bromides with carbon monoxide
Fleckenstein et al. The role of bidentate fluorenylphosphines in palladium-catalyzed cross-coupling reactions
Uberman et al. Highly efficient palladium-catalyzed arsination. Synthesis of a biphenyl arsine ligand and its application to obtain perfluoroalkylarsines
JP2004523523A (ja) 均一に触媒されるｃ−ｃカップリング反応のための方法
CN110845364B (zh) 一种以甲酰胺为氰源的腈类化合物的制备方法
Das Sustainable Strategies in Transition Metal Catalysis for Small Molecule Synthesis
CN119978004A (zh) 一种水稳定的2-吡啶内盐硼试剂及其制备方法与在偶联反应中的应用
Anderson Expanding the substrate scope in palladium-catalyzed CN and CC bond-forming reactions
Richards-Taylor Applications of DABSO in metal catalysis
Landge Transition-metal catalyzed CH bond alkynylation

Legal Events

Date Code Title Description
A521 Request for written amendment filed

Free format text: JAPANESE INTERMEDIATE CODE: A523

Effective date: 20050815

A621 Written request for application examination

Free format text: JAPANESE INTERMEDIATE CODE: A621

Effective date: 20050815

A711 Notification of change in applicant

Free format text: JAPANESE INTERMEDIATE CODE: A711

Effective date: 20070704

A131 Notification of reasons for refusal

Free format text: JAPANESE INTERMEDIATE CODE: A131

Effective date: 20081121

A601 Written request for extension of time

Free format text: JAPANESE INTERMEDIATE CODE: A601

Effective date: 20090213

A602 Written permission of extension of time

Free format text: JAPANESE INTERMEDIATE CODE: A602

Effective date: 20090220

A521 Request for written amendment filed

Free format text: JAPANESE INTERMEDIATE CODE: A523

Effective date: 20090417

A02 Decision of refusal

Free format text: JAPANESE INTERMEDIATE CODE: A02

Effective date: 20090604

A521 Request for written amendment filed

Free format text: JAPANESE INTERMEDIATE CODE: A523

Effective date: 20091005

A911 Transfer to examiner for re-examination before appeal (zenchi)

Free format text: JAPANESE INTERMEDIATE CODE: A911

Effective date: 20091015

TRDD Decision of grant or rejection written
A01 Written decision to grant a patent or to grant a registration (utility model)

Free format text: JAPANESE INTERMEDIATE CODE: A01

Effective date: 20091120

A01 Written decision to grant a patent or to grant a registration (utility model)

Free format text: JAPANESE INTERMEDIATE CODE: A01

A61 First payment of annual fees (during grant procedure)

Free format text: JAPANESE INTERMEDIATE CODE: A61

Effective date: 20091210

R150 Certificate of patent or registration of utility model

Free format text: JAPANESE INTERMEDIATE CODE: R150

FPAY Renewal fee payment (event date is renewal date of database)

Free format text: PAYMENT UNTIL: 20121218

Year of fee payment: 3

FPAY Renewal fee payment (event date is renewal date of database)

Free format text: PAYMENT UNTIL: 20121218

Year of fee payment: 3

FPAY Renewal fee payment (event date is renewal date of database)

Free format text: PAYMENT UNTIL: 20131218

Year of fee payment: 4

R250 Receipt of annual fees

Free format text: JAPANESE INTERMEDIATE CODE: R250

LAPS Cancellation because of no payment of annual fees