JP4301757B2 - エナンチオマー濃縮されたN−アシル化されたβ−アミノ酸の製造方法並びに保護基分離によるβ−アミノ酸の製造方法及びその使用 - Google Patents
エナンチオマー濃縮されたN−アシル化されたβ−アミノ酸の製造方法並びに保護基分離によるβ−アミノ酸の製造方法及びその使用 Download PDFInfo
- Publication number
- JP4301757B2 JP4301757B2 JP2002002691A JP2002002691A JP4301757B2 JP 4301757 B2 JP4301757 B2 JP 4301757B2 JP 2002002691 A JP2002002691 A JP 2002002691A JP 2002002691 A JP2002002691 A JP 2002002691A JP 4301757 B2 JP4301757 B2 JP 4301757B2
- Authority
- JP
- Japan
- Prior art keywords
- alkyl
- acylated
- hydrogenation
- amino acid
- cycloalkyl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Fee Related
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Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C231/00—Preparation of carboxylic acid amides
- C07C231/12—Preparation of carboxylic acid amides by reactions not involving the formation of carboxamide groups
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE10100971.2 | 2001-01-11 | ||
| DE10100971A DE10100971A1 (de) | 2001-01-11 | 2001-01-11 | Verfahren zur Herstellung enantiomerenangereicherter beta-Aminosäure |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2002265425A JP2002265425A (ja) | 2002-09-18 |
| JP2002265425A5 JP2002265425A5 (https=) | 2005-07-14 |
| JP4301757B2 true JP4301757B2 (ja) | 2009-07-22 |
Family
ID=7670234
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2002002691A Expired - Fee Related JP4301757B2 (ja) | 2001-01-11 | 2002-01-09 | エナンチオマー濃縮されたN−アシル化されたβ−アミノ酸の製造方法並びに保護基分離によるβ−アミノ酸の製造方法及びその使用 |
Country Status (5)
| Country | Link |
|---|---|
| US (1) | US6492544B2 (https=) |
| EP (1) | EP1225166B1 (https=) |
| JP (1) | JP4301757B2 (https=) |
| AT (1) | ATE279388T1 (https=) |
| DE (2) | DE10100971A1 (https=) |
Families Citing this family (17)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US7007861B2 (en) | 2000-06-08 | 2006-03-07 | S.C. Johnson & Son, Inc. | Methods and personal protection devices for repelling insects |
| MXPA03004168A (es) * | 2000-12-13 | 2004-12-02 | Warner Lambert Co | Sintesis de ligandos bisfosfolanos p-quirales y de sus complejos con metales de transicion para uso como catalizadores de hidrogenacion asimetrica. |
| JP4226847B2 (ja) * | 2001-07-24 | 2009-02-18 | 高砂香料工業株式会社 | ホスフィン−ホスホラン化合物と遷移金属とを含有する遷移金属錯体の存在下、α,β−不飽和アミド誘導体から光学活性アミド類を製造する方法。 |
| GB0120167D0 (en) * | 2001-08-17 | 2001-10-10 | Chirotech Technology Ltd | Asymmetric hydrogenation |
| WO2003042135A2 (en) * | 2001-11-09 | 2003-05-22 | The Penn State Research Foundation | P-chiral phospholanes and phosphocyclic compounds and their use in asymmetric catalytic reactions |
| US7169953B2 (en) * | 2001-11-09 | 2007-01-30 | The Penn State Research Foundation | P-chiral phospholanes and phosphocyclic compounds and their use in asymmetric catalytic reactions |
| CN1318433C (zh) * | 2002-04-04 | 2007-05-30 | 德古萨股份公司 | 作为二齿配体的双膦 |
| US7084089B2 (en) * | 2002-07-31 | 2006-08-01 | Shell Oil Company | Process for the carbonylation of ethylenically unsaturated compounds, bidentate diphosphine composition used in this process and a process for preparation of this bidentate diphosphine composition |
| US6806391B2 (en) | 2002-07-31 | 2004-10-19 | Shell Oil Company | Process for the carbonylation of ethylenically unsaturated compounds and bidentate diphosphine composition used in this process |
| AR043515A1 (es) * | 2003-03-19 | 2005-08-03 | Merck & Co Inc | Procedimiento para preparar derivados quirales beta aminoacidos mediante hidrogenacion asimetrica |
| TW200602293A (en) * | 2004-04-05 | 2006-01-16 | Merck & Co Inc | Process for the preparation of enantiomerically enriched beta amino acid derivatives |
| US7013601B2 (en) * | 2004-07-22 | 2006-03-21 | Coastal Planters, Llc | Plant container with hanger |
| US7618410B2 (en) * | 2004-10-05 | 2009-11-17 | Cardia Access, Inc. | Devices and methods for access through a tissue wall |
| DE102005014055A1 (de) * | 2005-03-23 | 2006-09-28 | Degussa Ag | Unsymmetrisch substituierte Phospholankatalysatoren |
| DE102005037649A1 (de) * | 2005-08-05 | 2007-02-08 | Leibniz-Institut Für Katalyse E.V. An Der Universität Rostock | Homogene katalytische Hydrierung |
| EP2070904A1 (en) | 2007-12-12 | 2009-06-17 | Laboratorios Del. Dr. Esteve, S.A. | Rhodium-phosphorus complexes and their use in ring opening reactions |
| EP2070903A1 (en) | 2007-12-12 | 2009-06-17 | Laboratorios del Dr. Esteve S.A. | Microwave-assisted ring opening reaction |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO1999059721A1 (en) * | 1998-05-18 | 1999-11-25 | The Penn State Research Foundation | Catalytic asymmetric hydrogenation, hydroformylation, and hydrovinylation via transition metal catalysts with phosphines and phosphites |
| ATE233780T1 (de) * | 1998-11-05 | 2003-03-15 | Chirotech Technology Ltd | Chirale ligande für asymmetrische katalysis |
-
2001
- 2001-01-11 DE DE10100971A patent/DE10100971A1/de not_active Withdrawn
- 2001-12-07 DE DE2001504095 patent/DE50104095D1/de not_active Expired - Lifetime
- 2001-12-07 EP EP01129076A patent/EP1225166B1/de not_active Expired - Lifetime
- 2001-12-07 AT AT01129076T patent/ATE279388T1/de not_active IP Right Cessation
-
2002
- 2002-01-09 JP JP2002002691A patent/JP4301757B2/ja not_active Expired - Fee Related
- 2002-01-11 US US10/042,256 patent/US6492544B2/en not_active Expired - Fee Related
Also Published As
| Publication number | Publication date |
|---|---|
| EP1225166A1 (de) | 2002-07-24 |
| US6492544B2 (en) | 2002-12-10 |
| DE50104095D1 (de) | 2004-11-18 |
| ATE279388T1 (de) | 2004-10-15 |
| JP2002265425A (ja) | 2002-09-18 |
| DE10100971A1 (de) | 2002-07-18 |
| US20020128509A1 (en) | 2002-09-12 |
| EP1225166B1 (de) | 2004-10-13 |
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