JP4191825B2 - ５−アミノイソキサゾール誘導体 - Google Patents

５−アミノイソキサゾール誘導体 Download PDF

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Publication number
JP4191825B2
JP4191825B2 JP27246798A JP27246798A JP4191825B2 JP 4191825 B2 JP4191825 B2 JP 4191825B2 JP 27246798 A JP27246798 A JP 27246798A JP 27246798 A JP27246798 A JP 27246798A JP 4191825 B2 JP4191825 B2 JP 4191825B2
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JP
Japan
Prior art keywords
group
isoxazole
pyridyl
fluorophenyl
formula
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
JP27246798A
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English (en)
Japanese (ja)
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JP2000086657A5 (https=
JP2000086657A (ja
Inventor
信義 南
通隆 佐藤
幸市 蓮見
則夫 山本
勝幸 慶野
照明 松井
有弘 金田
修治 太田
教久 斎藤
秀一郎 佐藤
章 朝烏
知 土井
基博 小林
潤 佐藤
創 浅野
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Aska Pharmaceutical Co Ltd
Original Assignee
Aska Pharmaceutical Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Aska Pharmaceutical Co Ltd filed Critical Aska Pharmaceutical Co Ltd
Priority to JP27246798A priority Critical patent/JP4191825B2/ja
Publication of JP2000086657A publication Critical patent/JP2000086657A/ja
Publication of JP2000086657A5 publication Critical patent/JP2000086657A5/ja
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Publication of JP4191825B2 publication Critical patent/JP4191825B2/ja
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

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  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
JP27246798A 1998-09-10 1998-09-10 ５−アミノイソキサゾール誘導体 Expired - Lifetime JP4191825B2 (ja)

Priority Applications (1)

Application Number Priority Date Filing Date Title
JP27246798A JP4191825B2 (ja) 1998-09-10 1998-09-10 ５−アミノイソキサゾール誘導体

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP27246798A JP4191825B2 (ja) 1998-09-10 1998-09-10 ５−アミノイソキサゾール誘導体

Publications (3)

Publication Number Publication Date
JP2000086657A JP2000086657A (ja) 2000-03-28
JP2000086657A5 JP2000086657A5 (https=) 2005-10-20
JP4191825B2 true JP4191825B2 (ja) 2008-12-03

Family

ID=17514333

Family Applications (1)

Application Number Title Priority Date Filing Date
JP27246798A Expired - Lifetime JP4191825B2 (ja) 1998-09-10 1998-09-10 ５−アミノイソキサゾール誘導体

Country Status (1)

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JP (1) JP4191825B2 (https=)

Families Citing this family (33)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP1312601A4 (en) * 2000-08-22 2005-09-21 Ono Pharmaceutical Co CARBOXYLENE DERIVATIVES, METHOD FOR THE PRODUCTION THEREOF, AND MEDICAMENTS CONTAINING THEM AS AN ACTIVE SUBSTANCE
CA2419722A1 (en) * 2000-09-01 2003-02-21 Masaki Asada Benzoic acid derivatives and drugs containing the same as the active ingredient
EP1317453B1 (en) * 2000-09-15 2006-08-09 Vertex Pharmaceuticals Incorporated Isoxazoles and their use as inhibitors of erk
JP2004521892A (ja) * 2000-12-20 2004-07-22 メルク　エンド　カムパニー　インコーポレーテッド （ハロ−ベンゾカルボニル）複素環縮合フェニル系ｐ３８キナーゼ阻害剤
SE0102764D0 (sv) 2001-08-17 2001-08-17 Astrazeneca Ab Compounds
ES2278170T3 (es) 2002-07-09 2007-08-01 BOEHRINGER INGELHEIM PHARMA GMBH & CO.KG Composiciones farmaceuticas de anticolinergicos e inhibidores de la quinasa p38 en el tratamiento de enfermedades respiratorias.
GB0226930D0 (en) 2002-11-19 2002-12-24 Astrazeneca Ab Chemical compounds
GB0226931D0 (en) 2002-11-19 2002-12-24 Astrazeneca Ab Chemical compounds
TW200600086A (en) 2004-06-05 2006-01-01 Astrazeneca Ab Chemical compound
US20060035893A1 (en) 2004-08-07 2006-02-16 Boehringer Ingelheim International Gmbh Pharmaceutical compositions for treatment of respiratory and gastrointestinal disorders
KR20070085371A (ko) 2004-10-16 2007-08-27 아스트라제네카 아베 페녹시 벤즈아미드 화합물의 제조 방법
PE20060777A1 (es) 2004-12-24 2006-10-06 Boehringer Ingelheim Int Derivados de indolinona para el tratamiento o la prevencion de enfermedades fibroticas
US7939536B2 (en) 2004-12-28 2011-05-10 Aska Pharmaceutical Co., Ltd. Pyrimidinylisoxazole derivatives
MX2007009888A (es) 2005-02-17 2007-10-16 Synta Pharmaceuticals Corp Compuestos para el tratamiento de trastornos proliferativos.
TW200714597A (en) 2005-05-27 2007-04-16 Astrazeneca Ab Chemical compounds
KR101346902B1 (ko) 2005-07-09 2014-01-02 아스트라제네카 아베 당뇨병 치료에 있어 ｇｌｋ 활성화제로서 사용하기 위한헤테로아릴 벤즈아미드 유도체
CA2627497C (en) 2005-10-28 2014-10-14 Takeda Pharmaceutical Company Limited Heterocyclic amide compound and use thereof
TW200738621A (en) 2005-11-28 2007-10-16 Astrazeneca Ab Chemical process
DK1975158T3 (da) * 2005-12-27 2011-10-24 Ct Nac Investigaciones Oncologicas Cnio Hidtil ukendte pyrrolderivater med histondeacetylase-inhibitoraktivitet
WO2008001929A1 (en) 2006-06-28 2008-01-03 Aska Pharmaceutical Co., Ltd. Treatment agent for inflammatory bowel disease
EP2036905B1 (en) * 2006-06-28 2012-12-12 ASKA Pharmaceutical Co., Ltd. Pyridylisoxazole derivative
TW200825063A (en) 2006-10-23 2008-06-16 Astrazeneca Ab Chemical compounds
TW200825060A (en) 2006-10-26 2008-06-16 Astrazeneca Ab Chemical compounds
KR20090090390A (ko) 2006-12-21 2009-08-25 아스트라제네카 아베 Ｇｌｋ 활성제로서 유용한 신규 결정 화합물
AU2008215659B2 (en) 2007-02-16 2012-11-01 Aska Pharmaceutical Co., Ltd. Pharmaceutical composition comprising microparticle oily suspension
EP1992344A1 (en) 2007-05-18 2008-11-19 Institut Curie P38 alpha as a therapeutic target in pathologies linked to FGFR3 mutation
CN101784516B (zh) * 2007-06-13 2014-07-02 百时美施贵宝公司 作为凝血因子抑制剂的二肽类似物
EP2324028A2 (en) 2008-08-04 2011-05-25 AstraZeneca AB Therapeutic agents 414
GB0902406D0 (en) 2009-02-13 2009-04-01 Astrazeneca Ab Crystalline polymorphic form
GB0902434D0 (en) 2009-02-13 2009-04-01 Astrazeneca Ab Chemical process
WO2010116177A1 (en) 2009-04-09 2010-10-14 Astrazeneca Ab A pyrazolo [4,5-e] pyrimidine derivative and its use to treat diabetes and obesity
AR076221A1 (es) 2009-04-09 2011-05-26 Astrazeneca Ab Derivado de pirazol [4,5-e] pirimidina y su uso para tratar diabetes y obesidad
WO2019022152A1 (ja) 2017-07-26 2019-01-31 学校法人同志社 ＴＧＦ－βシグナルに起因する障害を治療または予防するための医薬およびその応用

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Publication number Publication date
JP2000086657A (ja) 2000-03-28

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