JP2025515002A5 - - Google Patents

Info

Publication number
JP2025515002A5
JP2025515002A5 JP2024564484A JP2024564484A JP2025515002A5 JP 2025515002 A5 JP2025515002 A5 JP 2025515002A5 JP 2024564484 A JP2024564484 A JP 2024564484A JP 2024564484 A JP2024564484 A JP 2024564484A JP 2025515002 A5 JP2025515002 A5 JP 2025515002A5
Authority
JP
Japan
Prior art keywords
compound according
group
ring
alkyl
hydrogen
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2024564484A
Other languages
English (en)
Japanese (ja)
Other versions
JP2025515002A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2023/020546 external-priority patent/WO2023215220A1/en
Publication of JP2025515002A publication Critical patent/JP2025515002A/ja
Publication of JP2025515002A5 publication Critical patent/JP2025515002A5/ja
Pending legal-status Critical Current

Links

JP2024564484A 2022-05-02 2023-05-01 Atpクエン酸リアーゼのマクロ環式阻害剤 Pending JP2025515002A (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US202263337344P 2022-05-02 2022-05-02
US63/337,344 2022-05-02
US202363481045P 2023-01-23 2023-01-23
US63/481,045 2023-01-23
PCT/US2023/020546 WO2023215220A1 (en) 2022-05-02 2023-05-01 Macrocyclic inhibitors of atp citrate lyase

Publications (2)

Publication Number Publication Date
JP2025515002A JP2025515002A (ja) 2025-05-13
JP2025515002A5 true JP2025515002A5 (enExample) 2026-05-12

Family

ID=86776394

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2024564484A Pending JP2025515002A (ja) 2022-05-02 2023-05-01 Atpクエン酸リアーゼのマクロ環式阻害剤

Country Status (9)

Country Link
US (1) US20250289793A1 (enExample)
EP (1) EP4519251A1 (enExample)
JP (1) JP2025515002A (enExample)
KR (1) KR20250004873A (enExample)
CN (1) CN119137107A (enExample)
AU (1) AU2023264491A1 (enExample)
CA (1) CA3251749A1 (enExample)
IL (1) IL316386A (enExample)
WO (1) WO2023215220A1 (enExample)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IL328133A (en) * 2023-11-01 2026-06-01 Esperion Therapeutics Inc Macrocyclic inhibitors of atp citrate lyase

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3845770A (en) 1972-06-05 1974-11-05 Alza Corp Osmatic dispensing device for releasing beneficial agent
US4326525A (en) 1980-10-14 1982-04-27 Alza Corporation Osmotic device that improves delivery properties of agent in situ
US5364620A (en) 1983-12-22 1994-11-15 Elan Corporation, Plc Controlled absorption diltiazem formulation for once daily administration
US5023252A (en) 1985-12-04 1991-06-11 Conrex Pharmaceutical Corporation Transdermal and trans-membrane delivery of drugs
US5001139A (en) 1987-06-12 1991-03-19 American Cyanamid Company Enchancers for the transdermal flux of nivadipine
US4992445A (en) 1987-06-12 1991-02-12 American Cyanamid Co. Transdermal delivery of pharmaceuticals
US4902514A (en) 1988-07-21 1990-02-20 Alza Corporation Dosage form for administering nilvadipine for treating cardiovascular symptoms
WO2020097408A1 (en) * 2018-11-09 2020-05-14 Nimbus Artemis, Inc. Acly inhibitors and uses thereof
CN115677616B (zh) * 2021-11-03 2024-10-18 中国药科大学 大环磺酰胺类化合物及其制备方法和医药用途

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