JP2025511819A5 - - Google Patents

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Publication number
JP2025511819A5
JP2025511819A5 JP2024559337A JP2024559337A JP2025511819A5 JP 2025511819 A5 JP2025511819 A5 JP 2025511819A5 JP 2024559337 A JP2024559337 A JP 2024559337A JP 2024559337 A JP2024559337 A JP 2024559337A JP 2025511819 A5 JP2025511819 A5 JP 2025511819A5
Authority
JP
Japan
Prior art keywords
pyrano
dihydro
methylpiperidine
fluoro
substituted
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2024559337A
Other languages
English (en)
Japanese (ja)
Other versions
JP2025511819A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/IB2023/053561 external-priority patent/WO2023194964A1/en
Publication of JP2025511819A publication Critical patent/JP2025511819A/ja
Publication of JP2025511819A5 publication Critical patent/JP2025511819A5/ja
Pending legal-status Critical Current

Links

JP2024559337A 2022-04-07 2023-04-07 Nlrp3阻害剤としての縮合ピリダジン誘導体 Pending JP2025511819A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US202263328709P 2022-04-07 2022-04-07
US63/328,709 2022-04-07
PCT/IB2023/053561 WO2023194964A1 (en) 2022-04-07 2023-04-07 Fused pyridazine derivatives as nlrp3 inhibitors

Publications (2)

Publication Number Publication Date
JP2025511819A JP2025511819A (ja) 2025-04-16
JP2025511819A5 true JP2025511819A5 (https=) 2026-04-13

Family

ID=86329425

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2024559337A Pending JP2025511819A (ja) 2022-04-07 2023-04-07 Nlrp3阻害剤としての縮合ピリダジン誘導体

Country Status (6)

Country Link
US (1) US20250340563A1 (https=)
EP (1) EP4504733A1 (https=)
JP (1) JP2025511819A (https=)
AR (1) AR129012A1 (https=)
TW (1) TW202345838A (https=)
WO (1) WO2023194964A1 (https=)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US11618751B1 (en) 2022-03-25 2023-04-04 Ventus Therapeutics U.S., Inc. Pyrido-[3,4-d]pyridazine amine derivatives useful as NLRP3 derivatives
US11319319B1 (en) 2021-04-07 2022-05-03 Ventus Therapeutics U.S., Inc. Compounds for inhibiting NLRP3 and uses thereof
TW202319055A (zh) * 2021-07-21 2023-05-16 日商安斯泰來製藥股份有限公司 縮環噠嗪(pyridazine)化合物
US12331048B2 (en) 2022-10-31 2025-06-17 Ventus Therapeutics U.S., Inc. Pyrido-[3,4-d]pyridazine amine derivatives useful as NLRP3 inhibitors
WO2025153532A1 (en) 2024-01-16 2025-07-24 NodThera Limited Nlrp3 inhibitors and glp-1 agonists combination therapies

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR0166088B1 (ko) 1990-01-23 1999-01-15 . 수용해도가 증가된 시클로덱스트린 유도체 및 이의 용도
US5376645A (en) 1990-01-23 1994-12-27 University Of Kansas Derivatives of cyclodextrins exhibiting enhanced aqueous solubility and the use thereof
GB9518953D0 (en) 1995-09-15 1995-11-15 Pfizer Ltd Pharmaceutical formulations
GB9711643D0 (en) 1997-06-05 1997-07-30 Janssen Pharmaceutica Nv Glass thermoplastic systems
AR119731A1 (es) * 2019-05-17 2022-01-05 Novartis Ag Inhibidores del inflamasoma nlrp3
WO2022135567A1 (zh) * 2020-12-25 2022-06-30 上海拓界生物医药科技有限公司 一类含哒嗪的化合物及其医药用途
TW202319055A (zh) * 2021-07-21 2023-05-16 日商安斯泰來製藥股份有限公司 縮環噠嗪(pyridazine)化合物

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