JP2025511819A5 - - Google Patents
Info
- Publication number
- JP2025511819A5 JP2025511819A5 JP2024559337A JP2024559337A JP2025511819A5 JP 2025511819 A5 JP2025511819 A5 JP 2025511819A5 JP 2024559337 A JP2024559337 A JP 2024559337A JP 2024559337 A JP2024559337 A JP 2024559337A JP 2025511819 A5 JP2025511819 A5 JP 2025511819A5
- Authority
- JP
- Japan
- Prior art keywords
- pyrano
- dihydro
- methylpiperidine
- fluoro
- substituted
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US202263328709P | 2022-04-07 | 2022-04-07 | |
| US63/328,709 | 2022-04-07 | ||
| PCT/IB2023/053561 WO2023194964A1 (en) | 2022-04-07 | 2023-04-07 | Fused pyridazine derivatives as nlrp3 inhibitors |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2025511819A JP2025511819A (ja) | 2025-04-16 |
| JP2025511819A5 true JP2025511819A5 (https=) | 2026-04-13 |
Family
ID=86329425
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2024559337A Pending JP2025511819A (ja) | 2022-04-07 | 2023-04-07 | Nlrp3阻害剤としての縮合ピリダジン誘導体 |
Country Status (6)
| Country | Link |
|---|---|
| US (1) | US20250340563A1 (https=) |
| EP (1) | EP4504733A1 (https=) |
| JP (1) | JP2025511819A (https=) |
| AR (1) | AR129012A1 (https=) |
| TW (1) | TW202345838A (https=) |
| WO (1) | WO2023194964A1 (https=) |
Families Citing this family (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US11618751B1 (en) | 2022-03-25 | 2023-04-04 | Ventus Therapeutics U.S., Inc. | Pyrido-[3,4-d]pyridazine amine derivatives useful as NLRP3 derivatives |
| US11319319B1 (en) | 2021-04-07 | 2022-05-03 | Ventus Therapeutics U.S., Inc. | Compounds for inhibiting NLRP3 and uses thereof |
| TW202319055A (zh) * | 2021-07-21 | 2023-05-16 | 日商安斯泰來製藥股份有限公司 | 縮環噠嗪(pyridazine)化合物 |
| US12331048B2 (en) | 2022-10-31 | 2025-06-17 | Ventus Therapeutics U.S., Inc. | Pyrido-[3,4-d]pyridazine amine derivatives useful as NLRP3 inhibitors |
| WO2025153532A1 (en) | 2024-01-16 | 2025-07-24 | NodThera Limited | Nlrp3 inhibitors and glp-1 agonists combination therapies |
Family Cites Families (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| KR0166088B1 (ko) | 1990-01-23 | 1999-01-15 | . | 수용해도가 증가된 시클로덱스트린 유도체 및 이의 용도 |
| US5376645A (en) | 1990-01-23 | 1994-12-27 | University Of Kansas | Derivatives of cyclodextrins exhibiting enhanced aqueous solubility and the use thereof |
| GB9518953D0 (en) | 1995-09-15 | 1995-11-15 | Pfizer Ltd | Pharmaceutical formulations |
| GB9711643D0 (en) | 1997-06-05 | 1997-07-30 | Janssen Pharmaceutica Nv | Glass thermoplastic systems |
| AR119731A1 (es) * | 2019-05-17 | 2022-01-05 | Novartis Ag | Inhibidores del inflamasoma nlrp3 |
| WO2022135567A1 (zh) * | 2020-12-25 | 2022-06-30 | 上海拓界生物医药科技有限公司 | 一类含哒嗪的化合物及其医药用途 |
| TW202319055A (zh) * | 2021-07-21 | 2023-05-16 | 日商安斯泰來製藥股份有限公司 | 縮環噠嗪(pyridazine)化合物 |
-
2023
- 2023-04-05 AR ARP230100862A patent/AR129012A1/es unknown
- 2023-04-07 TW TW112113100A patent/TW202345838A/zh unknown
- 2023-04-07 WO PCT/IB2023/053561 patent/WO2023194964A1/en not_active Ceased
- 2023-04-07 EP EP23722044.7A patent/EP4504733A1/en active Pending
- 2023-04-07 US US18/854,298 patent/US20250340563A1/en active Pending
- 2023-04-07 JP JP2024559337A patent/JP2025511819A/ja active Pending
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