JP2025509846A5 - - Google Patents

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Publication number
JP2025509846A5
JP2025509846A5 JP2024555367A JP2024555367A JP2025509846A5 JP 2025509846 A5 JP2025509846 A5 JP 2025509846A5 JP 2024555367 A JP2024555367 A JP 2024555367A JP 2024555367 A JP2024555367 A JP 2024555367A JP 2025509846 A5 JP2025509846 A5 JP 2025509846A5
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JP
Japan
Prior art keywords
substituted
alkyl
compound
oxygen
unsubstituted
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2024555367A
Other languages
English (en)
Japanese (ja)
Other versions
JP2025509846A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2023/015024 external-priority patent/WO2023177593A1/en
Publication of JP2025509846A publication Critical patent/JP2025509846A/ja
Publication of JP2025509846A5 publication Critical patent/JP2025509846A5/ja
Pending legal-status Critical Current

Links

JP2024555367A 2022-03-14 2023-03-10 フェニルトリアゾールmll1-wdr5タンパク質-タンパク質間相互作用阻害剤 Pending JP2025509846A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US202263319582P 2022-03-14 2022-03-14
US63/319,582 2022-03-14
PCT/US2023/015024 WO2023177593A1 (en) 2022-03-14 2023-03-10 Phenyl triazole mll1-wdr5 protein-protein interaction inhibitor

Publications (2)

Publication Number Publication Date
JP2025509846A JP2025509846A (ja) 2025-04-11
JP2025509846A5 true JP2025509846A5 (https=) 2026-03-17

Family

ID=87932382

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2024555367A Pending JP2025509846A (ja) 2022-03-14 2023-03-10 フェニルトリアゾールmll1-wdr5タンパク質-タンパク質間相互作用阻害剤

Country Status (7)

Country Link
US (1) US20230286925A1 (https=)
EP (1) EP4493182A1 (https=)
JP (1) JP2025509846A (https=)
KR (1) KR20250023339A (https=)
CA (1) CA3245868A1 (https=)
MX (1) MX2024011348A (https=)
WO (1) WO2023177593A1 (https=)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN109734674B (zh) * 2019-02-26 2022-08-26 中国药科大学 苯胺类wdr5蛋白-蛋白相互作用抑制剂及其制法和用途
WO2025155755A1 (en) * 2024-01-16 2025-07-24 Rutgers, The State University Of New Jersey Sterically hindered 1h-1,2,3-triazol-5-ylidene abnormal n-heterocyclic carbene (anhc) ligands, catalyst complexes thereof, and methods using same
WO2026058961A1 (en) 2024-09-13 2026-03-19 Alivexis, Inc. Wdr5 inhibitors, compounds, pharmaceutical compositions, and methods of use thereof

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ATE501128T1 (de) * 2003-12-03 2011-03-15 Boehringer Ingelheim Pharma 1,2,3-triazolamidderivate als inhibitoren der cytokinproduktion
WO2015187827A1 (en) * 2014-06-03 2015-12-10 The Trustees Of The University Of Pennsylvania Novel effective antiviral compounds and methods using same
CN108715585A (zh) * 2018-04-23 2018-10-30 中国药科大学 苯基联三氮唑类mll1-wdr5蛋白-蛋白相互作用抑制剂
EP3810145A4 (en) * 2018-06-21 2022-06-01 Icahn School of Medicine at Mount Sinai Wd40 repeat domain protein 5 (wdr5) degradation / disruption compounds and methods of use

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