JP2025507732A5 - - Google Patents

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Publication number
JP2025507732A5
JP2025507732A5 JP2024550702A JP2024550702A JP2025507732A5 JP 2025507732 A5 JP2025507732 A5 JP 2025507732A5 JP 2024550702 A JP2024550702 A JP 2024550702A JP 2024550702 A JP2024550702 A JP 2024550702A JP 2025507732 A5 JP2025507732 A5 JP 2025507732A5
Authority
JP
Japan
Prior art keywords
membered
heterocycloalkyl
cycloalkyl
alkylene
heteroaryl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2024550702A
Other languages
English (en)
Japanese (ja)
Other versions
JP2025507732A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/CN2023/077893 external-priority patent/WO2023160614A1/zh
Publication of JP2025507732A publication Critical patent/JP2025507732A/ja
Publication of JP2025507732A5 publication Critical patent/JP2025507732A5/ja
Pending legal-status Critical Current

Links

JP2024550702A 2022-02-28 2023-02-23 Fak阻害剤としての化合物およびその使用 Pending JP2025507732A (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
CN202210190680.2 2022-02-28
CN202210190680 2022-02-28
CN202210800802.5 2022-07-06
CN202210800802 2022-07-06
PCT/CN2023/077893 WO2023160614A1 (zh) 2022-02-28 2023-02-23 作为fak抑制剂的化合物及其用途

Publications (2)

Publication Number Publication Date
JP2025507732A JP2025507732A (ja) 2025-03-21
JP2025507732A5 true JP2025507732A5 (enExample) 2026-03-03

Family

ID=87764843

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2024550702A Pending JP2025507732A (ja) 2022-02-28 2023-02-23 Fak阻害剤としての化合物およびその使用

Country Status (9)

Country Link
US (1) US20250154134A1 (enExample)
EP (1) EP4488272A4 (enExample)
JP (1) JP2025507732A (enExample)
KR (1) KR20240156623A (enExample)
CN (1) CN118574825A (enExample)
AU (1) AU2023224815A1 (enExample)
CA (1) CA3252402A1 (enExample)
MX (1) MX2024010431A (enExample)
WO (1) WO2023160614A1 (enExample)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN118525015A (zh) * 2021-12-21 2024-08-20 微境生物医药科技(上海)有限公司 作为fak抑制剂的化合物及其用途

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7521457B2 (en) * 2004-08-20 2009-04-21 Boehringer Ingelheim International Gmbh Pyrimidines as PLK inhibitors
AR074210A1 (es) * 2008-11-24 2010-12-29 Boehringer Ingelheim Int Derivados de pirimidina como inhibidores de ptk2-quinasa
CN108948019B (zh) * 2017-05-18 2022-07-08 广东东阳光药业有限公司 黏着斑激酶抑制剂及其用途
IL295117A (en) * 2020-01-31 2022-09-01 Verastem Inc Combinations containing kras g12c inhibitors for the treatment of abnormal cell growth
AU2021263742A1 (en) * 2020-04-27 2022-09-22 Verastem, Inc. Methods of treating abnormal cell growth
JP7836097B2 (ja) * 2020-08-03 2026-03-26 ▲應▼世生物科技(南京)有限公司 化合物の固体形態

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