JP2025507382A5 - - Google Patents

Info

Publication number
JP2025507382A5
JP2025507382A5 JP2024547761A JP2024547761A JP2025507382A5 JP 2025507382 A5 JP2025507382 A5 JP 2025507382A5 JP 2024547761 A JP2024547761 A JP 2024547761A JP 2024547761 A JP2024547761 A JP 2024547761A JP 2025507382 A5 JP2025507382 A5 JP 2025507382A5
Authority
JP
Japan
Prior art keywords
alkyl
present
compound
compound according
aryl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2024547761A
Other languages
English (en)
Japanese (ja)
Other versions
JP2025507382A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2023/062593 external-priority patent/WO2023154962A1/en
Publication of JP2025507382A publication Critical patent/JP2025507382A/ja
Publication of JP2025507382A5 publication Critical patent/JP2025507382A5/ja
Pending legal-status Critical Current

Links

JP2024547761A 2022-02-14 2023-02-14 cGAS阻害物質およびその使用法 Pending JP2025507382A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US202263309894P 2022-02-14 2022-02-14
US63/309,894 2022-02-14
PCT/US2023/062593 WO2023154962A1 (en) 2022-02-14 2023-02-14 Cgas inhibitors and uses thereof

Publications (2)

Publication Number Publication Date
JP2025507382A JP2025507382A (ja) 2025-03-18
JP2025507382A5 true JP2025507382A5 (https=) 2026-02-25

Family

ID=85556604

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2024547761A Pending JP2025507382A (ja) 2022-02-14 2023-02-14 cGAS阻害物質およびその使用法

Country Status (5)

Country Link
US (1) US20250163052A1 (https=)
EP (1) EP4479134A1 (https=)
JP (1) JP2025507382A (https=)
CA (1) CA3252179A1 (https=)
WO (1) WO2023154962A1 (https=)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN119490508A (zh) * 2023-08-21 2025-02-21 上海交通大学 一类螺环四氢-γ-咔啉衍生物的制备方法以及应用
WO2025218659A1 (en) * 2024-04-16 2025-10-23 Insilico Medicine Ip Limited Novel compounds as cyclic gmp-amp synthase inhibitor and uses thereof

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP3507486B2 (ja) 1991-03-15 2004-03-15 アムジエン・インコーポレーテツド 顆粒球コロニー刺激因子の肺内投与
US5451569A (en) 1994-04-19 1995-09-19 Hong Kong University Of Science And Technology R & D Corporation Limited Pulmonary drug delivery system
BR112020016008A2 (pt) 2018-02-05 2020-12-15 The Rockefeller University Composto, método para inibir uma resposta inflamatória em um paciente, método para inibir inflamação em um paciente, método para inibir expressão de interferon ativada por dsdna em um mamífero, método para tratar metástase de câncer em um paciente e formulação farmacêutica
US12522603B2 (en) * 2019-03-13 2026-01-13 The Rockefeller University Inhibitors of gas for treating autoinflammatory diseases and cancer metastasis
CN115197207B (zh) * 2021-04-09 2024-03-22 上海交通大学 一类四氢-γ-咔啉类衍生物、其药物组合物及应用

Similar Documents

Publication Publication Date Title
JP2020183410A5 (https=)
JP2025507382A5 (https=)
JP2006502143A5 (https=)
JP2008513496A5 (https=)
JP2023540344A5 (https=)
JP2017533968A5 (https=)
JP2020507589A5 (https=)
JP2011515482A5 (https=)
JP2017515844A5 (https=)
JP2011529918A5 (https=)
JP2019520416A5 (https=)
JP2021500394A5 (https=)
JP2019518766A5 (https=)
JP2012503018A5 (https=)
JP2008513498A5 (https=)
JP2011525927A5 (https=)
JP2018505898A5 (https=)
JP2008509166A5 (https=)
JP2017537158A5 (https=)
JP2007535496A5 (https=)
JP2010527913A5 (https=)
JP2008513504A5 (https=)
JP2011509309A5 (https=)
JP2017526677A5 (https=)
JP2013542267A5 (https=)