JP2025503451A5 - - Google Patents
Info
- Publication number
- JP2025503451A5 JP2025503451A5 JP2024536171A JP2024536171A JP2025503451A5 JP 2025503451 A5 JP2025503451 A5 JP 2025503451A5 JP 2024536171 A JP2024536171 A JP 2024536171A JP 2024536171 A JP2024536171 A JP 2024536171A JP 2025503451 A5 JP2025503451 A5 JP 2025503451A5
- Authority
- JP
- Japan
- Prior art keywords
- group
- amino
- amino acid
- acid
- residue
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Applications Claiming Priority (15)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP2021086592 | 2021-12-17 | ||
| EPPCT/EP2021/086592 | 2021-12-17 | ||
| EPPCT/EP2022/054857 | 2022-02-25 | ||
| EP2022054857 | 2022-02-25 | ||
| EPPCT/EP2022/057170 | 2022-03-18 | ||
| EP2022057170 | 2022-03-18 | ||
| EP2022057840 | 2022-03-24 | ||
| EPPCT/EP2022/057840 | 2022-03-24 | ||
| EP2022067424 | 2022-06-24 | ||
| EPPCT/EP2022/067424 | 2022-06-24 | ||
| EPPCT/EP2022/079606 | 2022-10-24 | ||
| EP2022079606 | 2022-10-24 | ||
| EP2022081674 | 2022-11-11 | ||
| EPPCT/EP2022/081674 | 2022-11-11 | ||
| PCT/EP2022/086632 WO2023111350A2 (en) | 2021-12-17 | 2022-12-19 | Carbonic anhydrase ix ligands |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2025503451A JP2025503451A (ja) | 2025-02-04 |
| JP2025503451A5 true JP2025503451A5 (https=) | 2025-12-16 |
Family
ID=84981172
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2024536171A Pending JP2025503451A (ja) | 2021-12-17 | 2022-12-19 | 炭酸脱水酵素ｉｘリガンド |
Country Status (13)
| Country | Link |
|---|---|
| US (1) | US20250339569A1 (https=) |
| EP (1) | EP4448544A2 (https=) |
| JP (1) | JP2025503451A (https=) |
| KR (1) | KR20240133798A (https=) |
| AR (1) | AR128023A1 (https=) |
| AU (1) | AU2022410422B2 (https=) |
| CA (1) | CA3242384A1 (https=) |
| CL (1) | CL2024001830A1 (https=) |
| IL (1) | IL313536A (https=) |
| MA (1) | MA66591A1 (https=) |
| MX (1) | MX2024007454A (https=) |
| TW (1) | TW202340226A (https=) |
| WO (1) | WO2023111350A2 (https=) |
Families Citing this family (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CA3243979A1 (en) * | 2022-02-11 | 2025-04-30 | C-Biomex Co., Ltd. | Peptide ligand targeting carbonic anhydrase IX, peptide construction comprising it, and associated uses |
| AR133015A1 (es) * | 2023-06-20 | 2025-08-20 | Debiopharm Int Sa | Compuesto radiomarcado para su uso en un método de tratamiento de enfermedades con anhidrasa carbónica ix positiva |
| WO2025023747A1 (ko) * | 2023-07-25 | 2025-01-30 | (주)씨바이오멕스 | 탄산탈수소효소 ⅸ를 표적으로 하는 펩타이드 구조체 및 이들의 용도 |
| CN120943901A (zh) * | 2025-05-29 | 2025-11-14 | 北京肿瘤医院(北京大学肿瘤医院) | 经修饰的caix靶向环肽、核素标记物及其在肿瘤诊疗方面的应用 |
Family Cites Families (20)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4885363A (en) | 1987-04-24 | 1989-12-05 | E. R. Squibb & Sons, Inc. | 1-substituted-1,4,7-triscarboxymethyl-1,4,7,10-tetraazacyclododecane and analogs |
| US5021556A (en) | 1987-07-22 | 1991-06-04 | Neorx Corporation | Method of radiolabeling chelating compounds comprising sulfur atoms with metal radionuclides |
| US5075099A (en) | 1988-05-31 | 1991-12-24 | Neorx Corporation | Metal radionuclide chelating compounds for improved chelation kinetics |
| US5364613A (en) | 1989-04-07 | 1994-11-15 | Sieving Paul F | Polychelants containing macrocyclic chelant moieties |
| US5367080A (en) | 1990-11-08 | 1994-11-22 | Sterling Winthrop Inc. | Complexing agents and targeting radioactive immunoreagents useful in therapeutic and diagnostic imaging compositions and methods |
| US5965107A (en) | 1992-03-13 | 1999-10-12 | Diatide, Inc. | Technetium-99m labeled peptides for imaging |
| US6214345B1 (en) | 1993-05-14 | 2001-04-10 | Bristol-Myers Squibb Co. | Lysosomal enzyme-cleavable antitumor drug conjugates |
| US5886142A (en) | 1997-05-20 | 1999-03-23 | Thomas Jefferson University | Radiolabeled thrombus imaging agents |
| EP2478912B1 (en) | 2003-11-06 | 2016-08-31 | Seattle Genetics, Inc. | Auristatin conjugates with anti-HER2 or anti-CD22 antibodies and their use in therapy |
| EP2100900A1 (en) | 2008-03-07 | 2009-09-16 | Universitätsspital Basel | Bombesin analog peptide antagonist conjugates |
| WO2012016713A1 (en) | 2010-08-05 | 2012-02-09 | Ruprecht-Karls-Universität Heidelberg | Tumour targeting with polypeptides |
| WO2013172954A1 (en) * | 2012-05-17 | 2013-11-21 | Ra Pharmaceuticals, Inc | Peptide and peptidomimetic inhibitors |
| US10954287B2 (en) * | 2016-04-15 | 2021-03-23 | Ra Pharmaceuticals, Inc. | Ras binding peptides and methods of use |
| TW201919682A (zh) * | 2017-08-08 | 2019-06-01 | 西班牙商阿爾米雷爾有限公司 | 活化Ｎｒｆ２路徑的新穎化合物 |
| WO2019096867A1 (en) | 2017-11-14 | 2019-05-23 | Debiopharm Research & Manufacturing S.A. | Ligand-drug-conjugates as substrates for selective cleavage by the exopeptidase activity of cathepsin b |
| WO2020084305A1 (en) * | 2018-10-23 | 2020-04-30 | Bicycletx Limited | Bicyclic peptide ligands and uses thereof |
| GB201900526D0 (en) | 2019-01-15 | 2019-03-06 | Bicyclerd Ltd | Bicyclic peptide ligands specific for caix |
| GB201900525D0 (en) * | 2019-01-15 | 2019-03-06 | Bicycletx Ltd | Bicyclic peptide ligands specific for caix |
| JP7801207B2 (ja) * | 2019-07-08 | 2026-01-16 | ３ベー ファーマシューティカルズ ゲーエムベーハー | 線維芽細胞活性化タンパク質リガンドを含む化合物およびその使用 |
| TWI765195B (zh) | 2019-11-22 | 2022-05-21 | 行政院原子能委員會核能研究所 | 雙靶向碳酸酐酶第九型複合物及其造影劑 |
-
2022
- 2022-12-19 TW TW111148813A patent/TW202340226A/zh unknown
- 2022-12-19 CA CA3242384A patent/CA3242384A1/en active Pending
- 2022-12-19 AR ARP220103498A patent/AR128023A1/es unknown
- 2022-12-19 IL IL313536A patent/IL313536A/en unknown
- 2022-12-19 WO PCT/EP2022/086632 patent/WO2023111350A2/en not_active Ceased
- 2022-12-19 JP JP2024536171A patent/JP2025503451A/ja active Pending
- 2022-12-19 MA MA66591A patent/MA66591A1/fr unknown
- 2022-12-19 MX MX2024007454A patent/MX2024007454A/es unknown
- 2022-12-19 AU AU2022410422A patent/AU2022410422B2/en active Active
- 2022-12-19 US US18/720,400 patent/US20250339569A1/en active Pending
- 2022-12-19 KR KR1020247023840A patent/KR20240133798A/ko active Pending
- 2022-12-19 EP EP22843649.9A patent/EP4448544A2/en active Pending
-
2024
- 2024-06-17 CL CL2024001830A patent/CL2024001830A1/es unknown
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