JP2025131625A5 - - Google Patents

Info

Publication number
JP2025131625A5
JP2025131625A5 JP2025083936A JP2025083936A JP2025131625A5 JP 2025131625 A5 JP2025131625 A5 JP 2025131625A5 JP 2025083936 A JP2025083936 A JP 2025083936A JP 2025083936 A JP2025083936 A JP 2025083936A JP 2025131625 A5 JP2025131625 A5 JP 2025131625A5
Authority
JP
Japan
Prior art keywords
compound
polymer
solid dispersion
amorphous solid
pharmaceutical composition
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2025083936A
Other languages
English (en)
Japanese (ja)
Other versions
JP2025131625A (ja
Filing date
Publication date
Priority claimed from PCT/US2020/027677 external-priority patent/WO2020210629A1/en
Application filed filed Critical
Publication of JP2025131625A publication Critical patent/JP2025131625A/ja
Publication of JP2025131625A5 publication Critical patent/JP2025131625A5/ja
Pending legal-status Critical Current

Links

JP2025083936A 2019-04-11 2025-05-20 治療血漿濃度に達するために増強された非晶質固体および溶解製剤の性能 Pending JP2025131625A (ja)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US201962832606P 2019-04-11 2019-04-11
US62/832,606 2019-04-11
PCT/US2020/027677 WO2020210629A1 (en) 2019-04-11 2020-04-10 Enhanced performance of amorphous solid and solubilized formulations for achieving therapeutic plasma concentrations
JP2021559853A JP2022526656A (ja) 2019-04-11 2020-04-10 治療血漿濃度に達するために増強された非晶質固体および溶解製剤の性能

Related Parent Applications (1)

Application Number Title Priority Date Filing Date
JP2021559853A Division JP2022526656A (ja) 2019-04-11 2020-04-10 治療血漿濃度に達するために増強された非晶質固体および溶解製剤の性能

Publications (2)

Publication Number Publication Date
JP2025131625A JP2025131625A (ja) 2025-09-09
JP2025131625A5 true JP2025131625A5 (enExample) 2025-11-07

Family

ID=70465560

Family Applications (2)

Application Number Title Priority Date Filing Date
JP2021559853A Withdrawn JP2022526656A (ja) 2019-04-11 2020-04-10 治療血漿濃度に達するために増強された非晶質固体および溶解製剤の性能
JP2025083936A Pending JP2025131625A (ja) 2019-04-11 2025-05-20 治療血漿濃度に達するために増強された非晶質固体および溶解製剤の性能

Family Applications Before (1)

Application Number Title Priority Date Filing Date
JP2021559853A Withdrawn JP2022526656A (ja) 2019-04-11 2020-04-10 治療血漿濃度に達するために増強された非晶質固体および溶解製剤の性能

Country Status (17)

Country Link
EP (1) EP3953355A1 (enExample)
JP (2) JP2022526656A (enExample)
KR (1) KR20210151183A (enExample)
CN (1) CN113924300A (enExample)
AR (1) AR118650A1 (enExample)
AU (1) AU2020271103A1 (enExample)
BR (1) BR112021020257A2 (enExample)
CA (1) CA3132530A1 (enExample)
CL (1) CL2021002627A1 (enExample)
CO (1) CO2021015054A2 (enExample)
EA (1) EA202192753A1 (enExample)
IL (1) IL287103A (enExample)
MX (2) MX2021012288A (enExample)
PE (1) PE20212367A1 (enExample)
SG (1) SG11202111131VA (enExample)
TW (1) TW202104228A (enExample)
WO (1) WO2020210629A1 (enExample)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA3212644A1 (en) * 2021-03-09 2022-09-15 Bayer Aktiengesellschaft Pharmaceutical dosage forms comprising (4s)-24-chloro-4-ethyl-73-fluoro-35-methoxy-32,5- dioxo-14-(trifluoromethyl)-32h-6-aza-3(4,1)-pyridina-1(1)-[1,2,3]triazola-2(1,2),7(1)- dibenzenaheptaphane-74-carboxamide
JP2024534427A (ja) 2021-09-17 2024-09-20 ブリストル-マイヤーズ スクイブ カンパニー 血栓塞栓性障害を予防かつ治療するためのミルベキシアン
UY40381A (es) 2022-08-01 2024-01-31 Janssen Pharmaceutica Nv Uso de milvexian para el tratamiento o la prevención del accidente cerebrovascular isquémico
WO2024167899A1 (en) 2023-02-06 2024-08-15 Bristol-Myers Squibb Company Milvexian pharmaceutical compositions
WO2025099743A1 (en) * 2023-11-07 2025-05-15 Dr. Reddy’S Laboratories Limited Process for preparation of milvexian and solid-state forms thereof
WO2025126240A1 (en) * 2023-12-12 2025-06-19 Dr. Reddy's Laboratories Limited Pharmaceutical compositions and use thereof
WO2025220042A1 (en) * 2024-04-18 2025-10-23 Dr. Reddy's Laboratories Limited Pharmaceutical compositions comprising asundexian and use thereof
WO2025224678A1 (en) 2024-04-25 2025-10-30 Assia Chemical Industries Ltd. Solid state forms of milvexian and process for preparation thereof

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PT83812B (en) 1985-11-27 1988-03-15 Syntex Inc Process for preparing amorphous benzimidazole derivatives
PT901786E (pt) * 1997-08-11 2007-08-07 Pfizer Prod Inc Disperções farmacêuticas sólidas com biodisponibilidade melhorada
WO2010102245A1 (en) 2009-03-05 2010-09-10 Upsher-Smith Laboratories, Inc. Solid dispersion comprising resveratrol
UY40230A (es) * 2014-01-31 2023-08-15 Bristol Myers Squibb Company Una Corporacion Del Estado De Delaware Macrociclos con grupos P2’ heterocíclicos como inhibidores del factor XIa y composiciones farmacéuticas que los comprenden
US9453018B2 (en) 2014-10-01 2016-09-27 Bristol-Myers Squibb Company Pyrimidinones as factor XIa inhibitors
NO2721243T3 (enExample) * 2014-10-01 2018-10-20

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