JP2024544538A5 - - Google Patents

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Publication number
JP2024544538A5
JP2024544538A5 JP2024527603A JP2024527603A JP2024544538A5 JP 2024544538 A5 JP2024544538 A5 JP 2024544538A5 JP 2024527603 A JP2024527603 A JP 2024527603A JP 2024527603 A JP2024527603 A JP 2024527603A JP 2024544538 A5 JP2024544538 A5 JP 2024544538A5
Authority
JP
Japan
Prior art keywords
pharmaceutical composition
compound
composition according
approximately
pharmaceutically acceptable
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2024527603A
Other languages
English (en)
Japanese (ja)
Other versions
JP2024544538A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/CN2022/131297 external-priority patent/WO2023083288A1/en
Publication of JP2024544538A publication Critical patent/JP2024544538A/ja
Publication of JP2024544538A5 publication Critical patent/JP2024544538A5/ja
Pending legal-status Critical Current

Links

JP2024527603A 2021-11-11 2022-11-11 THR-βアゴニストによる肝障害の治療 Pending JP2024544538A (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
CNPCT/CN2021/130083 2021-11-11
CN2021130083 2021-11-11
CN2022097426 2022-06-07
CNPCT/CN2022/097426 2022-06-07
PCT/CN2022/131297 WO2023083288A1 (en) 2021-11-11 2022-11-11 TREATMENT OF LIVER DISORDERS WITH A THR-β AGONIST

Publications (2)

Publication Number Publication Date
JP2024544538A JP2024544538A (ja) 2024-12-03
JP2024544538A5 true JP2024544538A5 (https=) 2025-11-18

Family

ID=86335128

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2024527603A Pending JP2024544538A (ja) 2021-11-11 2022-11-11 THR-βアゴニストによる肝障害の治療

Country Status (14)

Country Link
US (1) US20240293416A1 (https=)
EP (1) EP4429666A4 (https=)
JP (1) JP2024544538A (https=)
KR (1) KR20240101642A (https=)
CN (1) CN118871113A (https=)
AU (1) AU2022388507A1 (https=)
CA (1) CA3238108A1 (https=)
CL (1) CL2024001399A1 (https=)
CO (1) CO2024007225A2 (https=)
IL (1) IL312637A (https=)
MX (1) MX2024005647A (https=)
PE (1) PE20241327A1 (https=)
TW (1) TW202332447A (https=)
WO (1) WO2023083288A1 (https=)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN111320609A (zh) 2018-12-13 2020-06-23 拓臻股份有限公司 一种THRβ受体激动剂化合物及其制备方法和用途
AU2020336272A1 (en) 2019-08-23 2022-04-14 Terns Pharmaceuticals, Inc. Thyroid hormone receptor beta agonist compounds
WO2021050945A1 (en) 2019-09-12 2021-03-18 Terns, Inc. Thyroid hormone receptor beta agonist compounds
EP4568664B1 (en) 2023-04-07 2026-04-01 Terns Pharmaceuticals, Inc. Combination comprising a thr-beta agonist and a glp-1r agonist for use in treating obesity
WO2025245216A1 (en) * 2024-05-22 2025-11-27 Terns Pharmaceuticals, Inc. Treatment of liver disorders with a thr-beta agonist

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2018075650A1 (en) * 2016-10-18 2018-04-26 Madrigal Pharmaceuticals, Inc. Methods of treating liver disorders or lipid disorders with a thr-beta agonist
AR115666A1 (es) * 2018-07-02 2021-02-10 Madrigal Pharmaceuticals Inc Formas sólidas de 2-(3,5-dicloro-4-((5-isopropil-6-oxo-1,6-dihidropiridazin-3-il)oxi)fenil)-3,5-dioxo-2,3,4,5-tetrahidro-1,2,4-triazin-6-carbonitrilo
CN111320609A (zh) * 2018-12-13 2020-06-23 拓臻股份有限公司 一种THRβ受体激动剂化合物及其制备方法和用途
WO2020228577A1 (zh) * 2019-05-10 2020-11-19 深圳微芯生物科技股份有限公司 一种哒嗪酮衍生物及其应用
TW202128668A (zh) * 2019-12-16 2021-08-01 大陸商江蘇恆瑞醫藥股份有限公司 并環類衍生物、其製備方法及其在醫藥上的應用
US20210379043A1 (en) * 2020-05-13 2021-12-09 Terns Pharmaceuticals, Inc. Combination treatment of liver disorders
CN114437034A (zh) * 2020-11-06 2022-05-06 深圳微芯生物科技股份有限公司 一种酞嗪类化合物的可药用盐、晶型及其制备方法

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