JP2024542199A5 - - Google Patents
Info
- Publication number
- JP2024542199A5 JP2024542199A5 JP2024529504A JP2024529504A JP2024542199A5 JP 2024542199 A5 JP2024542199 A5 JP 2024542199A5 JP 2024529504 A JP2024529504 A JP 2024529504A JP 2024529504 A JP2024529504 A JP 2024529504A JP 2024542199 A5 JP2024542199 A5 JP 2024542199A5
- Authority
- JP
- Japan
- Prior art keywords
- hydrocarbyl
- membered
- halohydrocarbyl
- general formula
- optionally substituted
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Applications Claiming Priority (7)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| CN202111399876 | 2021-11-19 | ||
| CN202111399876.4 | 2021-11-19 | ||
| CN202210225663.8 | 2022-03-09 | ||
| CN202210225663 | 2022-03-09 | ||
| CN202210667619 | 2022-06-13 | ||
| CN202210667619.2 | 2022-06-13 | ||
| PCT/CN2022/132954 WO2023088441A1 (zh) | 2021-11-19 | 2022-11-18 | Kif18a抑制剂 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2024542199A JP2024542199A (ja) | 2024-11-13 |
| JP2024542199A5 true JP2024542199A5 (enExample) | 2025-11-25 |
Family
ID=86396297
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2024529504A Pending JP2024542199A (ja) | 2021-11-19 | 2022-11-18 | Kif18a阻害剤 |
Country Status (9)
| Country | Link |
|---|---|
| US (1) | US20260158017A1 (enExample) |
| EP (1) | EP4434979A4 (enExample) |
| JP (1) | JP2024542199A (enExample) |
| KR (1) | KR20240108489A (enExample) |
| CN (1) | CN118215657A (enExample) |
| AU (1) | AU2022389558A1 (enExample) |
| CA (1) | CA3237625A1 (enExample) |
| MX (1) | MX2024005996A (enExample) |
| WO (1) | WO2023088441A1 (enExample) |
Families Citing this family (14)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| IL283639B2 (en) | 2018-12-20 | 2024-06-01 | Amgen Inc | Kif18a inhibitors |
| KR20240109977A (ko) | 2021-08-26 | 2024-07-12 | 볼라스트라 쎄라퓨틱스, 인코포레이티드 | Kif18a의 스피로 인돌린 억제제 |
| WO2024022508A1 (zh) * | 2022-07-29 | 2024-02-01 | 武汉人福创新药物研发中心有限公司 | Kif18a抑制剂及用途 |
| CR20250087A (es) | 2022-08-18 | 2025-07-11 | Accent Therapeutics Inc | Inhibidores de kif18a y usos de estos |
| CN117917405A (zh) * | 2022-10-21 | 2024-04-23 | 杭州邦顺制药有限公司 | Kif18a蛋白抑制剂 |
| WO2024114730A1 (zh) * | 2022-11-30 | 2024-06-06 | 微境生物医药科技(上海)有限公司 | 一种用于癌症治疗的药物组合物 |
| JP2026508745A (ja) * | 2022-12-02 | 2026-03-12 | シェンチェン ジョングァー バイオロジカル テクノロジー カンパニー リミテッド | アミド又はウレア系化合物 |
| CN120569373A (zh) * | 2023-01-05 | 2025-08-29 | 浙江海正药业股份有限公司 | 芳香酰胺类衍生物及其制备方法和医药上的用途 |
| WO2024244972A1 (zh) * | 2023-05-30 | 2024-12-05 | 浙江海正药业股份有限公司 | 芳香酰胺类衍生物及其制备方法和用途 |
| EP4748837A1 (en) * | 2023-07-21 | 2026-05-27 | Zhejiang Hisun Pharmaceutical Co., Ltd. | Aromatic amide derivative, and preparation method therefor and use thereof |
| CN121752573A (zh) * | 2023-08-02 | 2026-03-27 | 上海湃隆生物科技有限公司 | 驱动蛋白kif18a抑制剂及其应用 |
| CN121693499A (zh) * | 2023-08-16 | 2026-03-17 | 上海湃隆生物科技有限公司 | 驱动蛋白kif18a抑制剂及其应用 |
| WO2025190888A1 (en) * | 2024-03-12 | 2025-09-18 | F. Hoffmann-La Roche Ag | Macrocyclic kif18a inhibitors and their use thereof |
| WO2025201407A1 (zh) * | 2024-03-27 | 2025-10-02 | 上海齐鲁制药研究中心有限公司 | 驱动蛋白kif18a抑制剂及其使用方法 |
Family Cites Families (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AUPO395396A0 (en) * | 1996-12-02 | 1997-01-02 | Fujisawa Pharmaceutical Co., Ltd. | Benzamide derivatives |
| MA54550A (fr) * | 2018-12-20 | 2022-03-30 | Amgen Inc | Inhibiteurs de kif18a |
| AU2019401495B2 (en) * | 2018-12-20 | 2025-06-26 | Amgen Inc. | Heteroaryl amides useful as KIF18A inhibitors |
| AU2019404576B2 (en) * | 2018-12-20 | 2025-07-17 | Amgen Inc. | Heteroaryl amides useful as KIF18A inhibitors |
| IL283639B2 (en) | 2018-12-20 | 2024-06-01 | Amgen Inc | Kif18a inhibitors |
| AU2020325115B2 (en) * | 2019-08-02 | 2026-03-12 | Amgen Inc. | Pyridine derivatives as KIF18A inhibitors |
| JP7699100B2 (ja) * | 2019-08-02 | 2025-06-26 | アムジエン・インコーポレーテツド | Kif18a阻害剤 |
| US20220289724A1 (en) * | 2019-08-02 | 2022-09-15 | Amgen Inc. | Kif18a inhibitors |
| JP2023521802A (ja) * | 2020-04-14 | 2023-05-25 | アムジエン・インコーポレーテツド | 新生物疾患の処置のためのkif18a阻害剤 |
| KR20240070604A (ko) * | 2021-09-24 | 2024-05-21 | 제논 파마슈티칼스 인크. | 소듐 채널 활성화제로서 피리디닐아세트아미드 유도체 |
-
2022
- 2022-11-18 MX MX2024005996A patent/MX2024005996A/es unknown
- 2022-11-18 EP EP22894970.7A patent/EP4434979A4/en active Pending
- 2022-11-18 AU AU2022389558A patent/AU2022389558A1/en active Pending
- 2022-11-18 CA CA3237625A patent/CA3237625A1/en active Pending
- 2022-11-18 WO PCT/CN2022/132954 patent/WO2023088441A1/zh not_active Ceased
- 2022-11-18 JP JP2024529504A patent/JP2024542199A/ja active Pending
- 2022-11-18 KR KR1020247020178A patent/KR20240108489A/ko active Pending
- 2022-11-18 CN CN202280076424.9A patent/CN118215657A/zh active Pending
- 2022-11-18 US US18/706,640 patent/US20260158017A1/en active Pending
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