JP2024527427A5 - - Google Patents

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Publication number
JP2024527427A5
JP2024527427A5 JP2024503904A JP2024503904A JP2024527427A5 JP 2024527427 A5 JP2024527427 A5 JP 2024527427A5 JP 2024503904 A JP2024503904 A JP 2024503904A JP 2024503904 A JP2024503904 A JP 2024503904A JP 2024527427 A5 JP2024527427 A5 JP 2024527427A5
Authority
JP
Japan
Application number
JP2024503904A
Other languages
Japanese (ja)
Other versions
JPWO2023002011A5 (https=
JP2024527427A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/EP2022/070601 external-priority patent/WO2023002011A1/en
Publication of JP2024527427A publication Critical patent/JP2024527427A/ja
Publication of JP2024527427A5 publication Critical patent/JP2024527427A5/ja
Publication of JPWO2023002011A5 publication Critical patent/JPWO2023002011A5/ja
Pending legal-status Critical Current

Links

JP2024503904A 2021-07-23 2022-07-22 グラム陰性細菌排出ポンプ阻害剤 Pending JP2024527427A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP21306032.0 2021-07-23
EP21306032 2021-07-23
PCT/EP2022/070601 WO2023002011A1 (en) 2021-07-23 2022-07-22 Gram-negative bacteria efflux pump inhibitors

Publications (3)

Publication Number Publication Date
JP2024527427A JP2024527427A (ja) 2024-07-24
JP2024527427A5 true JP2024527427A5 (https=) 2025-07-11
JPWO2023002011A5 JPWO2023002011A5 (https=) 2025-07-11

Family

ID=77564041

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2024503904A Pending JP2024527427A (ja) 2021-07-23 2022-07-22 グラム陰性細菌排出ポンプ阻害剤

Country Status (6)

Country Link
US (1) US20240327354A1 (https=)
EP (1) EP4373808A1 (https=)
JP (1) JP2024527427A (https=)
KR (1) KR20240057402A (https=)
CN (1) CN118076585A (https=)
WO (1) WO2023002011A1 (https=)

Family Cites Families (20)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0200024B1 (de) * 1985-04-30 1992-07-01 ARZNEIMITTELWERK DRESDEN GmbH 3-Cyan-pyridine, Verfahren zu ihrer Herstellung und ihre pharmazeutische Verwendung
AU2001280091A1 (en) * 2000-08-01 2002-02-13 Wockhardt Limited Inhibitors of cellular efflux pumps of microbes
US7074794B2 (en) * 2000-08-10 2006-07-11 Mitsubishi Pharma Corporation Proline derivatives and the use thereof as drugs
JP2007507514A (ja) * 2003-09-30 2007-03-29 ジヤンセン・フアーマシユーチカ・ナームローゼ・フエンノートシヤツプ キノキサリン化合物
EP1836189A1 (en) * 2005-01-06 2007-09-26 AstraZeneca AB Novel pyridine compounds
EP1987827A1 (en) * 2006-02-20 2008-11-05 Takeda Pharmaceutical Company Limited Novel pharmaceutical
TW200815426A (en) * 2006-06-28 2008-04-01 Astrazeneca Ab New pyridine analogues II 333
MX2009000577A (es) * 2006-07-14 2009-03-09 Schering Corp Compuestos de piperazina sustituida heterociclica con actividad antagonista de cxcr3.
TW201204727A (en) * 2010-03-10 2012-02-01 Kalypsys Inc Heterocyclic inhibitors of histamine receptors for the treatment of disease
JP2011246461A (ja) * 2010-04-27 2011-12-08 Mitsubishi Tanabe Pharma Corp 新規アミド誘導体を含有する医薬組成物
EA201390476A1 (ru) * 2010-09-28 2013-08-30 Бристол-Майерс Сквибб Компани Новые пиперазиновые аналоги с замещенными гетероарильными группами в качестве противовирусных средств широкого применения против гриппа
EP3371164B1 (en) * 2015-11-06 2022-03-16 Neurocrine Biosciences, Inc. N-[2-(1-benzylpiperidin-4-yl)ethyl]-4-(pyrazin-2-yl)-piperazine-1-carboxamide derivatives and related compounds as muscarinic receptor 4 (m4) antagonists for treating neurological diseases
WO2017097927A1 (en) * 2015-12-11 2017-06-15 Syngenta Participations Ag Pesticidally active 1,2,4-triazole derivatives
US20190119236A1 (en) * 2016-02-23 2019-04-25 Portola Pharmaceuticals, Inc. Compounds for binding proprotein convertase subtilisin/kexin type 9 (pcsk9)
WO2017160069A1 (ko) * 2016-03-15 2017-09-21 재단법인 의약바이오컨버젼스연구단 신규한 벤젠설폰아미드 유도체 및 이의 용도
MX393606B (es) * 2016-12-30 2025-03-19 Mitobridge Inc Inhibidores de poli-adp ribosa polimerasa (parp)
US11518764B2 (en) * 2018-02-06 2022-12-06 Ontario Institute For Cancer Research (Oicr) Substituted heteroaryls as inhibitors of the BCL6 BTB domain protein-protein interaction
JP7637328B2 (ja) * 2019-02-07 2025-02-28 ベイジーン リミテッド Tlr7アゴニストとしてのイミダゾ[2,1-f][1,2,4]トリアジン-4-アミン誘導体
WO2021067859A1 (en) * 2019-10-03 2021-04-08 Tenaya Therapeutics, Inc. 5-fluoronicotinamide derivatives and uses thereof
WO2021127333A1 (en) * 2019-12-19 2021-06-24 Casma Therapeutics, Inc. Trpml modulators

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