JP2024525713A5 - - Google Patents

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Publication number
JP2024525713A5
JP2024525713A5 JP2024501662A JP2024501662A JP2024525713A5 JP 2024525713 A5 JP2024525713 A5 JP 2024525713A5 JP 2024501662 A JP2024501662 A JP 2024501662A JP 2024501662 A JP2024501662 A JP 2024501662A JP 2024525713 A5 JP2024525713 A5 JP 2024525713A5
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JP
Japan
Prior art keywords
group
optionally substituted
alkyl
hydroxyl
solid support
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2024501662A
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English (en)
Japanese (ja)
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JP2024525713A (ja
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Publication date
Application filed filed Critical
Priority claimed from PCT/US2022/037262 external-priority patent/WO2023288047A2/en
Publication of JP2024525713A publication Critical patent/JP2024525713A/ja
Publication of JP2024525713A5 publication Critical patent/JP2024525713A5/ja
Pending legal-status Critical Current

Links

JP2024501662A 2021-07-15 2022-07-15 糖のアノマー部位におけるクリックケミストリーを介したターゲティングリガンドの多重化 Pending JP2024525713A (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US202163222090P 2021-07-15 2021-07-15
US63/222,090 2021-07-15
US202163236029P 2021-08-23 2021-08-23
US63/236,029 2021-08-23
PCT/US2022/037262 WO2023288047A2 (en) 2021-07-15 2022-07-15 Multiplexing targeting ligands through click chemistry at the anomeric site of sugars

Publications (2)

Publication Number Publication Date
JP2024525713A JP2024525713A (ja) 2024-07-12
JP2024525713A5 true JP2024525713A5 (https=) 2025-07-11

Family

ID=84920555

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2024501662A Pending JP2024525713A (ja) 2021-07-15 2022-07-15 糖のアノマー部位におけるクリックケミストリーを介したターゲティングリガンドの多重化

Country Status (4)

Country Link
US (1) US20250188470A1 (https=)
EP (1) EP4370132A4 (https=)
JP (1) JP2024525713A (https=)
WO (1) WO2023288047A2 (https=)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN118146284B (zh) * 2024-05-08 2024-07-26 北京悦康科创医药科技股份有限公司 一种GalNAc化合物、其与寡核苷酸缀合物及制备方法
CN120208906B (zh) * 2024-11-21 2025-10-28 广州同隽医药科技有限公司 维生素e衍生物、其载体化合物及其应用

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5773607A (en) * 1991-11-14 1998-06-30 Zaidan Hojin Biseibutsu Kagaku Kenkyu Kai Processes for preparing 2'-deoxy-2'-fluorocoformycin and stereoisomers thereof
US5891862A (en) * 1996-03-15 1999-04-06 Geltex Pharmaceuticals, Inc. Polyvalent polymers for the treatment of rotavirus infection
ATE238328T1 (de) * 1996-10-16 2003-05-15 Ribapharm Inc Monozyklische l-nukleoside, analoga und ihre anwendungen
US7560544B2 (en) * 2004-12-17 2009-07-14 Anadys Pharmaceuticals, Inc. 3,5-Disubsitituted and 3,5,7-trisubstituted-3H-oxazolo and 3H-thiazolo[4,5-d]pyrimidin-2-one compounds and prodrugs thereof
WO2009067191A2 (en) * 2007-11-16 2009-05-28 The General Hospital Corporation Methods and compositions for the treatment of hepatitis c virus (hcv) infection
WO2009099942A2 (en) * 2008-01-31 2009-08-13 Alnylam Pharmaceuticals, Inc. Chemically modified oligonucleotides and uses thereof
AU2009298802A1 (en) * 2008-09-23 2010-04-08 Alnylam Pharmaceuticals, Inc. Chemical modifications of monomers and oligonucleotides with cycloaddition
FR2974089B1 (fr) * 2011-04-18 2014-04-25 Univ Nice Sophia Antipolis Derives de l'acadesine, produits et compositions les comprenant, leurs utilisations therapeutiques et leurs procedes de synthese.
TWI793262B (zh) * 2018-02-21 2023-02-21 法商液態空氣喬治斯克勞帝方法研究開發股份有限公司 全氫聚矽氮烷組成物和用於使用其形成氮化物膜之方法

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