JP2024520648A - ナトリウムチャネルの調節因子としての置換テトラヒドロフラン－２－カルボキサミド - Google Patents

ナトリウムチャネルの調節因子としての置換テトラヒドロフラン－２－カルボキサミド Download PDF

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JP2024520648A
JP2024520648A JP2023574380A JP2023574380A JP2024520648A JP 2024520648 A JP2024520648 A JP 2024520648A JP 2023574380 A JP2023574380 A JP 2023574380A JP 2023574380 A JP2023574380 A JP 2023574380A JP 2024520648 A JP2024520648 A JP 2024520648A
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pain
pharma
alkyl
acceptable salt
compound
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JP2024520648A5 (enExample
Inventor
エリザベス メアリー ベック，
ロバート プリン，
ジャルディ， ゴルカ エチェバリア
ディーン ステイモス，
イボンヌ シュミット，
ジョセフ ポンティロ，
スティーブン アンドリュー トムソン，
デイビッド マシュー ショー，
ナディア エム． アハマド，
メイレレス， リディオ マルクス カルバーリョ
サラ スケラット，
ルア， サラ エス． ハディダ
マーク トーマス ミラー，
ティモシー ドナルド ノイバート，
デニス ジェイムズ ハーレイ，
ジンラン ジョウ，
アレクサンダー キンツァー，
スティーブン ジョン デュラント，
クリストファー レイ，
アニサ ニザラリ ビラニ，
キリ ノース，
ジェイムズ ドッド，
リース ジャックス，
スティーブン マイケル ゲディス，
バイラビ ガラン，
ロナルド マーセラス ネグテル，
エワ イウォナ チャデク，
ジョアン ルイーズ ピンダー，
ブルーノ アルトゥール スーザ，
レベッカ イー． スティーブンズ，
ミランダ アデル ライト，
ヘザー クレア ツウィン，
ジェイムズ ジュン ボン ムイ，
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Vertex Pharmaceuticals Inc
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Vertex Pharmaceuticals Inc
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Publication of JP2024520648A publication Critical patent/JP2024520648A/ja
Publication of JP2024520648A5 publication Critical patent/JP2024520648A5/ja
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    • A61K31/341—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having five-membered rings with one oxygen as the only ring hetero atom, e.g. isosorbide not condensed with another ring, e.g. ranitidine, furosemide, bufetolol, muscarine
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JP2024522293A (ja) * 2021-06-04 2024-06-13 バーテックス ファーマシューティカルズ インコーポレイテッド ナトリウムチャネルのモジュレーターとしての置換テトラヒドロフラン類似体

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