JP2024515062A5 - - Google Patents

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Publication number
JP2024515062A5
JP2024515062A5 JP2023561906A JP2023561906A JP2024515062A5 JP 2024515062 A5 JP2024515062 A5 JP 2024515062A5 JP 2023561906 A JP2023561906 A JP 2023561906A JP 2023561906 A JP2023561906 A JP 2023561906A JP 2024515062 A5 JP2024515062 A5 JP 2024515062A5
Authority
JP
Japan
Application number
JP2023561906A
Other languages
Japanese (ja)
Other versions
JP2024515062A (ja
JPWO2022214691A5 (https=
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/EP2022/059527 external-priority patent/WO2022214691A1/en
Publication of JP2024515062A publication Critical patent/JP2024515062A/ja
Publication of JPWO2022214691A5 publication Critical patent/JPWO2022214691A5/ja
Publication of JP2024515062A5 publication Critical patent/JP2024515062A5/ja
Pending legal-status Critical Current

Links

JP2023561906A 2021-04-09 2022-04-08 重水素化dhodh阻害剤 Pending JP2024515062A (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
EP21167690 2021-04-09
EP21167690.3 2021-04-09
EP21181134 2021-06-23
EP21181134.4 2021-06-23
PCT/EP2022/059527 WO2022214691A1 (en) 2021-04-09 2022-04-08 Deuterated dhodh inhibitors

Publications (3)

Publication Number Publication Date
JP2024515062A JP2024515062A (ja) 2024-04-04
JPWO2022214691A5 JPWO2022214691A5 (https=) 2025-04-15
JP2024515062A5 true JP2024515062A5 (https=) 2025-04-15

Family

ID=81585846

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2023561906A Pending JP2024515062A (ja) 2021-04-09 2022-04-08 重水素化dhodh阻害剤

Country Status (10)

Country Link
US (1) US20240199535A1 (https=)
EP (1) EP4320100A1 (https=)
JP (1) JP2024515062A (https=)
KR (1) KR20240007144A (https=)
AU (1) AU2022253683A1 (https=)
BR (1) BR112023020806A2 (https=)
CA (1) CA3215002A1 (https=)
IL (1) IL307559A (https=)
MX (1) MX2023011864A (https=)
WO (1) WO2022214691A1 (https=)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PL3139914T3 (pl) 2014-05-08 2023-11-27 Kiora Pharmaceuticals Gmbh Związki stosowane w leczeniu chorób i schorzeń okulistycznych
ES2972099T3 (es) 2018-03-09 2024-06-11 Kiora Pharmaceuticals Gmbh Formulación oftálmica
WO2023172818A1 (en) * 2022-03-09 2023-09-14 Kiora Pharmaceuticals Gmbh Polymorphs of a dihydroorotate dehydrogenase (dhod) inhibitor
TW202444688A (zh) 2023-03-29 2024-11-16 德商埃慕尼克股份公司 作為nurr1激動劑之維多氟地莫(vidofludimus)及相關結構
TW202506107A (zh) 2023-06-28 2025-02-16 德商埃慕尼克股份公司 雜芳族dhodh抑制劑
WO2025215126A1 (en) 2024-04-12 2025-10-16 Immunic Ag Synthesis of vidofludimus and its calcium salt
WO2026074007A1 (en) 2024-10-02 2026-04-09 Immunic Ag Nurr1 agonists with replacement of the carboxylic acid or carboxamide moiety for use in the treatment of neurodegenerative diseases

Family Cites Families (18)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
MXPA04000224A (es) * 2001-07-10 2005-07-25 4Sc Ag Novedosos compuestos como agentes antiinflamatorios, inmunomoduladores y antiproliferativos.
US7071355B2 (en) 2002-12-23 2006-07-04 4 Sc Ag Compounds as anti-inflammatory, immunomodulatory and anti-proliferatory agents
EP1581478A1 (en) 2002-12-23 2005-10-05 4Sc Ag Dhodh-inhibitors and method for their identification
MXPA05006890A (es) 2002-12-23 2006-04-07 4Sc Ag Compuestos como agentes anti-inflamatorios, inmunomoduladores y anti-proliferativos.
DK2050749T3 (en) 2006-08-08 2018-01-08 Chugai Pharmaceutical Co Ltd PYRIMIDINE DERIVATIVES AS PI3K INHIBITOR AND USE THEREOF
WO2009140279A2 (en) 2008-05-12 2009-11-19 Concert Pharmaceuticals, Inc. Sulfonyl urea compounds
CN102271674A (zh) 2008-11-07 2011-12-07 4Sc股份公司 用于治疗自身免疫病的包含dhodh抑制剂和氨甲喋呤的联合治疗
TWI530286B (zh) 2009-05-04 2016-04-21 帕納特斯製藥格斯有限公司 作為抑制病毒化合物之抗發炎劑
UA108760C2 (uk) 2010-07-01 2015-06-10 Кальцієві солі сполуки як протизапальні, імуномодулюючі та антипроліферативні засоби
KR102265277B1 (ko) * 2014-04-11 2021-06-16 판옵테스 파르마 게스.엠.베.하. 바이러스 억제 화합물로서의 항-염증제
PL3139914T3 (pl) 2014-05-08 2023-11-27 Kiora Pharmaceuticals Gmbh Związki stosowane w leczeniu chorób i schorzeń okulistycznych
WO2016045587A1 (zh) 2014-09-26 2016-03-31 常州寅盛药业有限公司 作为ns4b抑制剂的苯并呋喃类似物
CN108430998B (zh) 2016-09-28 2021-07-09 四川科伦博泰生物医药股份有限公司 氮杂双环衍生物及其制备方法和用途
WO2018177151A1 (en) * 2017-03-28 2018-10-04 Xiamen University Compounds modulating activity of farnesoid x receptor and methods for the use thereof
CN111343975A (zh) 2017-11-23 2020-06-26 埃慕尼克股份公司 用于预防或治疗慢性炎性疾病和/或自身免疫疾病的维多地莫的剂量方案
JP6804790B1 (ja) 2017-12-07 2020-12-23 エモリー ユニバーシティー N4−ヒドロキシシチジンおよび誘導体ならびにそれらに関連する抗ウイルス用途
ES2972099T3 (es) 2018-03-09 2024-06-11 Kiora Pharmaceuticals Gmbh Formulación oftálmica
WO2019175396A1 (en) 2018-03-16 2019-09-19 Immunic Ag Novel calcium salt polymorphs as anti-inflammatory, immunomodulatory and anti-proliferatory agents

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