JP2024512070A5 - - Google Patents

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Publication number
JP2024512070A5
JP2024512070A5 JP2023558777A JP2023558777A JP2024512070A5 JP 2024512070 A5 JP2024512070 A5 JP 2024512070A5 JP 2023558777 A JP2023558777 A JP 2023558777A JP 2023558777 A JP2023558777 A JP 2023558777A JP 2024512070 A5 JP2024512070 A5 JP 2024512070A5
Authority
JP
Japan
Prior art keywords
methyl
indoline
carboxamide
trifluoromethyl
phenyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2023558777A
Other languages
English (en)
Japanese (ja)
Other versions
JP2024512070A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/EP2022/057939 external-priority patent/WO2022200577A1/en
Publication of JP2024512070A publication Critical patent/JP2024512070A/ja
Publication of JP2024512070A5 publication Critical patent/JP2024512070A5/ja
Pending legal-status Critical Current

Links

JP2023558777A 2021-03-26 2022-03-25 Ddr阻害物質としてのインドリン Pending JP2024512070A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP21165281 2021-03-26
EP21165281.3 2021-03-26
PCT/EP2022/057939 WO2022200577A1 (en) 2021-03-26 2022-03-25 Indoline derivatives as ddrs inhibitors

Publications (2)

Publication Number Publication Date
JP2024512070A JP2024512070A (ja) 2024-03-18
JP2024512070A5 true JP2024512070A5 (https=) 2025-03-31

Family

ID=75252444

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2023558777A Pending JP2024512070A (ja) 2021-03-26 2022-03-25 Ddr阻害物質としてのインドリン

Country Status (12)

Country Link
US (1) US20240217967A1 (https=)
EP (1) EP4313972B1 (https=)
JP (1) JP2024512070A (https=)
KR (1) KR20230164105A (https=)
CN (1) CN117062812A (https=)
AU (1) AU2022245281A1 (https=)
BR (1) BR112023019288A2 (https=)
CA (1) CA3212872A1 (https=)
ES (1) ES3022533T3 (https=)
MX (1) MX2023011081A (https=)
PL (1) PL4313972T3 (https=)
WO (1) WO2022200577A1 (https=)

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EA001539B1 (ru) * 1996-11-27 2001-04-23 Пфайзер Инк. Амиды, ингибирующие секрецию аполипопротеина в (аро в) и/или микросомного протеина переноса триглицеридов (мтр)
CN104447701B (zh) * 2013-09-17 2019-03-22 广东东阳光药业有限公司 吡唑类衍生物及其用途
AU2015335980A1 (en) 2014-10-22 2017-05-18 Guangzhou Institutes Of Biomedicine And Health, Chinese Academy Of Sciences Small-molecule inhibitors targeting discoidin domain receptor 1 and uses thereof

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