JP2024510312A - キナゾリン系化合物、キナゾリン系化合物の組成物及び応用 - Google Patents
キナゾリン系化合物、キナゾリン系化合物の組成物及び応用 Download PDFInfo
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- JP2024510312A JP2024510312A JP2023557350A JP2023557350A JP2024510312A JP 2024510312 A JP2024510312 A JP 2024510312A JP 2023557350 A JP2023557350 A JP 2023557350A JP 2023557350 A JP2023557350 A JP 2023557350A JP 2024510312 A JP2024510312 A JP 2024510312A
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- pyrrolidin
- alkyl
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- hydroxy
- cancer
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- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/70—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
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- C07D239/86—Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in position 4
- C07D239/94—Nitrogen atoms
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- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
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- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
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- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
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Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| CN202110296394 | 2021-03-19 | ||
| CN202110296394.X | 2021-03-19 | ||
| PCT/CN2022/081599 WO2022194265A1 (zh) | 2021-03-19 | 2022-03-18 | 一种喹唑啉类化合物、组合物及其应用 |
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| CN104736155B (zh) * | 2012-05-14 | 2018-01-02 | 杭州德润玉成生物科技有限公司 | 双环化合物作为激酶的抑制剂 |
| TWI609012B (zh) * | 2013-04-28 | 2017-12-21 | 廣東東陽光藥業有限公司 | 氨基喹唑啉類衍生物及其鹽和使用方法 |
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| CA3212079A1 (en) | 2022-09-22 |
| AU2022235956A1 (en) | 2023-10-05 |
| CN115109036A (zh) | 2022-09-27 |
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| EP4293016A1 (en) | 2023-12-20 |
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