JP2024508890A5 - - Google Patents

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Publication number
JP2024508890A5
JP2024508890A5 JP2023553246A JP2023553246A JP2024508890A5 JP 2024508890 A5 JP2024508890 A5 JP 2024508890A5 JP 2023553246 A JP2023553246 A JP 2023553246A JP 2023553246 A JP2023553246 A JP 2023553246A JP 2024508890 A5 JP2024508890 A5 JP 2024508890A5
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JP
Japan
Prior art keywords
approximately
cancer
compound
effective dose
lymphoma
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Withdrawn
Application number
JP2023553246A
Other languages
English (en)
Japanese (ja)
Other versions
JP2024508890A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/IB2021/051776 external-priority patent/WO2022185097A1/en
Publication of JP2024508890A publication Critical patent/JP2024508890A/ja
Publication of JP2024508890A5 publication Critical patent/JP2024508890A5/ja
Withdrawn legal-status Critical Current

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JP2023553246A 2021-03-03 2021-03-03 治療有効用量のmalt1阻害剤jnj-67856633(1-(1-オキソ-1,2-ジヒドロイソキノリン-5-イル)-5-(トリフルオロメチル)-n-(2-(トリフルオロメチル)ピリジン-4-イル)-1h-ピラゾール-4-カルボキサミド)を使用して状態を治療する方法 Withdrawn JP2024508890A (ja)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
PCT/IB2021/051776 WO2022185097A1 (en) 2021-03-03 2021-03-03 Method of treating a condition using a therapeutically effective dose of the malt1 inhibitor jnj -67856633 (1 -(1 -oxo-1,2-dihydroisoquinolin-5-yl)-5-(trifluoromethyl)-n-(2-(trifluoromethyl)pyridin-4-yl)-1 h-py razole-4-carboxamide)

Publications (2)

Publication Number Publication Date
JP2024508890A JP2024508890A (ja) 2024-02-28
JP2024508890A5 true JP2024508890A5 (https=) 2024-03-13

Family

ID=74860360

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2023553246A Withdrawn JP2024508890A (ja) 2021-03-03 2021-03-03 治療有効用量のmalt1阻害剤jnj-67856633(1-(1-オキソ-1,2-ジヒドロイソキノリン-5-イル)-5-(トリフルオロメチル)-n-(2-(トリフルオロメチル)ピリジン-4-イル)-1h-ピラゾール-4-カルボキサミド)を使用して状態を治療する方法

Country Status (10)

Country Link
US (1) US20240299376A1 (https=)
EP (1) EP4301364A1 (https=)
JP (1) JP2024508890A (https=)
KR (1) KR20230154227A (https=)
CN (1) CN117279639A (https=)
AU (1) AU2021431485A1 (https=)
BR (1) BR112023017689A2 (https=)
CA (1) CA3212339A1 (https=)
MX (1) MX2023010322A (https=)
WO (1) WO2022185097A1 (https=)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TWI795381B (zh) 2016-12-21 2023-03-11 比利時商健生藥品公司 作為malt1抑制劑之吡唑衍生物
EP3953345B1 (en) 2019-04-11 2023-04-05 Janssen Pharmaceutica NV Pyridine rings containing derivatives as malt1 inhibitors
CN118451068A (zh) * 2021-12-30 2024-08-06 上海翰森生物医药科技有限公司 三并环类衍生物抑制剂、其制备方法和应用

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TWI795381B (zh) 2016-12-21 2023-03-11 比利時商健生藥品公司 作為malt1抑制劑之吡唑衍生物
US12269813B2 (en) 2019-02-22 2025-04-08 Janssen Pharmaceutica Nv Crystalline form of 1-(1-oxo-1,2-dihydroisoquinolin-5-yl)-5-(trifluoromethyl)-N-(2-(trifluoromethyl)pyridin-4-yl)-1H-pyrazole-4-carboxamide monohydrate
US20220175760A1 (en) * 2019-02-22 2022-06-09 Janssen Pharmaceutica Nv Pharmaceutical formulations

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