JP2024506387A5 - - Google Patents
Info
- Publication number
- JP2024506387A5 JP2024506387A5 JP2023548877A JP2023548877A JP2024506387A5 JP 2024506387 A5 JP2024506387 A5 JP 2024506387A5 JP 2023548877 A JP2023548877 A JP 2023548877A JP 2023548877 A JP2023548877 A JP 2023548877A JP 2024506387 A5 JP2024506387 A5 JP 2024506387A5
- Authority
- JP
- Japan
- Prior art keywords
- compound according
- hydrogen
- amino
- pharmaceutical composition
- alkyl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US202163147859P | 2021-02-10 | 2021-02-10 | |
| US63/147,859 | 2021-02-10 | ||
| PCT/US2022/015767 WO2022173795A1 (en) | 2021-02-10 | 2022-02-09 | OXADIAZOLYL DIHYDROPYRANO[2,3-b]PYRIDINE INHIBITORS OF HIPK2 FOR TREATING KIDNEY FIBROSIS |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2024506387A JP2024506387A (ja) | 2024-02-13 |
| JP2024506387A5 true JP2024506387A5 (https=) | 2025-01-27 |
Family
ID=82837244
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2023548877A Pending JP2024506387A (ja) | 2021-02-10 | 2022-02-09 | 腎線維症を治療するためのオキサジアゾリルジヒドロピラノ[2,3‐b]ピリジン系HIPK2阻害剤 |
Country Status (9)
| Country | Link |
|---|---|
| US (1) | US20250179084A1 (https=) |
| EP (1) | EP4291183B1 (https=) |
| JP (1) | JP2024506387A (https=) |
| KR (1) | KR20230154194A (https=) |
| CN (1) | CN117479934A (https=) |
| AU (1) | AU2022221336A1 (https=) |
| CA (1) | CA3210658A1 (https=) |
| MX (1) | MX2023009323A (https=) |
| WO (1) | WO2022173795A1 (https=) |
Families Citing this family (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US20240051965A1 (en) * | 2022-08-05 | 2024-02-15 | Icahn School Of Medicine At Mount Sinai | Oxygen-containing heterocyclic compound and use thereof |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| PL2069335T3 (pl) * | 2006-09-08 | 2013-05-31 | Actelion Pharmaceuticals Ltd | Pochodne pirydyn-3-ylu jako środki immunomodulujące |
| PE20091339A1 (es) * | 2007-12-21 | 2009-09-26 | Glaxo Group Ltd | Derivados de oxadiazol con actividad sobre receptores s1p1 |
| EP2210890A1 (en) * | 2009-01-19 | 2010-07-28 | Almirall, S.A. | Oxadiazole derivatives as S1P1 receptor agonists |
| ES2907624T3 (es) * | 2017-01-06 | 2022-04-25 | Icahn School Med Mount Sinai | Inhibidores de oxadiazol de HIPK2 para el tratamiento de la fibrosis renal |
| JP7252908B2 (ja) * | 2017-06-14 | 2023-04-05 | トレベナ・インコーポレイテッド | S1p1活性を調節するための化合物およびその使用法 |
-
2022
- 2022-02-09 AU AU2022221336A patent/AU2022221336A1/en active Pending
- 2022-02-09 CN CN202280014176.5A patent/CN117479934A/zh active Pending
- 2022-02-09 WO PCT/US2022/015767 patent/WO2022173795A1/en not_active Ceased
- 2022-02-09 MX MX2023009323A patent/MX2023009323A/es unknown
- 2022-02-09 JP JP2023548877A patent/JP2024506387A/ja active Pending
- 2022-02-09 KR KR1020237030728A patent/KR20230154194A/ko active Pending
- 2022-02-09 EP EP22753240.5A patent/EP4291183B1/en active Active
- 2022-02-09 US US18/264,809 patent/US20250179084A1/en active Pending
- 2022-02-09 CA CA3210658A patent/CA3210658A1/en active Pending
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