JP2024503637A5 - - Google Patents

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Publication number
JP2024503637A5
JP2024503637A5 JP2023541264A JP2023541264A JP2024503637A5 JP 2024503637 A5 JP2024503637 A5 JP 2024503637A5 JP 2023541264 A JP2023541264 A JP 2023541264A JP 2023541264 A JP2023541264 A JP 2023541264A JP 2024503637 A5 JP2024503637 A5 JP 2024503637A5
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JP
Japan
Prior art keywords
pharmaceutically acceptable
group
hydrate
amino acid
acceptable salt
Prior art date
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Pending
Application number
JP2023541264A
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English (en)
Japanese (ja)
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JP2024503637A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/EP2022/050280 external-priority patent/WO2022148843A1/en
Publication of JP2024503637A publication Critical patent/JP2024503637A/ja
Publication of JP2024503637A5 publication Critical patent/JP2024503637A5/ja
Pending legal-status Critical Current

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JP2023541264A 2021-01-07 2022-01-07 線維芽細胞活性化タンパク質リガンドを含む化合物およびその使用 Pending JP2024503637A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US202163134704P 2021-01-07 2021-01-07
US63/134,704 2021-01-07
PCT/EP2022/050280 WO2022148843A1 (en) 2021-01-07 2022-01-07 Compounds comprising a fibroblast activation protein ligand and use thereof

Publications (2)

Publication Number Publication Date
JP2024503637A JP2024503637A (ja) 2024-01-26
JP2024503637A5 true JP2024503637A5 (enExample) 2025-11-12

Family

ID=80050672

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2023541264A Pending JP2024503637A (ja) 2021-01-07 2022-01-07 線維芽細胞活性化タンパク質リガンドを含む化合物およびその使用

Country Status (11)

Country Link
US (1) US20230212549A1 (enExample)
EP (1) EP4274835A1 (enExample)
JP (1) JP2024503637A (enExample)
KR (1) KR20230129261A (enExample)
CN (1) CN116940585A (enExample)
AU (1) AU2022205523A1 (enExample)
CA (1) CA3206863A1 (enExample)
CL (5) CL2023001991A1 (enExample)
IL (1) IL303925A (enExample)
MX (1) MX2023007869A (enExample)
WO (1) WO2022148843A1 (enExample)

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CN118930606A (zh) * 2023-05-11 2024-11-12 成都纽瑞特医疗科技股份有限公司 靶向成纤维细胞活化蛋白的多肽放射性核素配合物及其应用
AU2024304266A1 (en) * 2023-06-14 2025-12-04 Mariana Oncology Inc. Dll3 targeting peptides and constructs thereof
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TW202502800A (zh) * 2023-07-11 2025-01-16 大陸商江蘇恆瑞醫藥股份有限公司 一種成纖維細胞活化蛋白配體及其用途
WO2025082283A1 (zh) * 2023-10-16 2025-04-24 四川科伦博泰生物医药股份有限公司 环肽结构的配体化合物及其核素标记物、药物组合物及应用
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WO2025179168A1 (en) * 2024-02-22 2025-08-28 Mariana Oncology Inc. Synthesis of dll3-binding peptides
CN118725026B (zh) * 2024-06-07 2026-05-01 中国科学院上海药物研究所 一类靶向肿瘤相关成纤维细胞激活蛋白的糖肽、放射性核素标记物及其应用
WO2026046340A1 (zh) * 2024-08-30 2026-03-05 江苏恒瑞医药股份有限公司 一种f-18标记反应前体分子的方法
WO2026056964A1 (zh) * 2024-09-14 2026-03-19 四川科伦博泰生物医药股份有限公司 环肽结构的配体化合物及其核素标记物、药物组合物及应用
WO2026149506A1 (zh) * 2025-01-10 2026-07-16 天津恒瑞医药有限公司 一种药物组合物及其制备方法
WO2026149529A1 (zh) * 2025-01-10 2026-07-16 天津恒瑞医药有限公司 一种成纤维细胞活化蛋白配体及其用途
WO2026163110A1 (en) 2025-01-30 2026-08-06 Novartis Ag Combinations with fap targeting compounds and conjugates thereof
CN121494877A (zh) * 2025-10-24 2026-02-10 复旦大学附属眼耳鼻喉科医院 一种硼原子标记的靶向成纤维细胞激活蛋白的化合物及其制备方法和应用
CN121045338B (zh) * 2025-11-05 2026-05-19 原子高科股份有限公司 一种靶向caix的环肽及其制备方法与应用

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JP2021500373A (ja) * 2017-10-23 2021-01-07 ザ・ジョンズ・ホプキンス・ユニバーシティ 線維芽細胞活性化タンパク質α（ＦＡＰ−α）を標的とする撮像剤および放射線療法用薬剤
EP3763726A1 (en) * 2019-07-08 2021-01-13 3B Pharmaceuticals GmbH Compounds comprising a fibroblast activation protein ligand and use thereof

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