JP2023547346A5 - - Google Patents

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Publication number
JP2023547346A5
JP2023547346A5 JP2023522401A JP2023522401A JP2023547346A5 JP 2023547346 A5 JP2023547346 A5 JP 2023547346A5 JP 2023522401 A JP2023522401 A JP 2023522401A JP 2023522401 A JP2023522401 A JP 2023522401A JP 2023547346 A5 JP2023547346 A5 JP 2023547346A5
Authority
JP
Japan
Prior art keywords
methyl
dimethylamino
ethoxy
oxadiazole
phenyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2023522401A
Other languages
English (en)
Japanese (ja)
Other versions
JP7687636B2 (ja
JP2023547346A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/EP2021/077660 external-priority patent/WO2022074103A1/en
Publication of JP2023547346A publication Critical patent/JP2023547346A/ja
Publication of JP2023547346A5 publication Critical patent/JP2023547346A5/ja
Application granted granted Critical
Publication of JP7687636B2 publication Critical patent/JP7687636B2/ja
Active legal-status Critical Current
Anticipated expiration legal-status Critical

Links

JP2023522401A 2020-10-08 2021-10-07 セロトニン1b受容体モジュレーターとしての強力で選択的な新規化合物 Active JP7687636B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP20382888.4 2020-10-08
EP20382888 2020-10-08
PCT/EP2021/077660 WO2022074103A1 (en) 2020-10-08 2021-10-07 Potent and selctive compounds as serotonin 1b receptor modulators

Publications (3)

Publication Number Publication Date
JP2023547346A JP2023547346A (ja) 2023-11-10
JP2023547346A5 true JP2023547346A5 (https=) 2024-07-23
JP7687636B2 JP7687636B2 (ja) 2025-06-03

Family

ID=73030029

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2023522401A Active JP7687636B2 (ja) 2020-10-08 2021-10-07 セロトニン1b受容体モジュレーターとしての強力で選択的な新規化合物

Country Status (21)

Country Link
US (1) US12540133B2 (https=)
EP (2) EP4445901A3 (https=)
JP (1) JP7687636B2 (https=)
KR (1) KR20230107566A (https=)
CN (1) CN116635390B (https=)
AU (1) AU2021356114A1 (https=)
CA (1) CA3194700A1 (https=)
CL (1) CL2023001021A1 (https=)
DK (1) DK4225753T3 (https=)
ES (1) ES2985416T3 (https=)
FI (1) FI4225753T3 (https=)
HR (1) HRP20241184T1 (https=)
HU (1) HUE068199T2 (https=)
IL (1) IL301806B1 (https=)
LT (1) LT4225753T (https=)
MX (1) MX2023004116A (https=)
PL (1) PL4225753T3 (https=)
PT (1) PT4225753T (https=)
RS (1) RS65956B1 (https=)
SI (1) SI4225753T1 (https=)
WO (1) WO2022074103A1 (https=)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AR123701A1 (es) 2020-10-08 2023-01-04 Merck Sharp & Dohme Preparación de derivados de oxindol como nuevos inhibidores de la diacilglicerol o-aciltransferasa 2
EP4382519A4 (en) * 2021-08-27 2024-12-04 Adlai Nortye Biopharma Co., Ltd. CYCLIN K DEGRADING AGENT
AU2024302643A1 (en) 2023-06-16 2026-01-22 Leukos Biotech Sl 5-htr1b modulator for use in the treatment of solid tumours

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TW240217B (https=) * 1992-12-30 1995-02-11 Glaxo Group Ltd
US5801170A (en) 1993-12-07 1998-09-01 Smithkline Beecham Plc Heterocyclic biphenylylamides useful as 5HT1D antagonists
ZA985542B (en) * 1997-07-03 1999-04-07 Smithkline Beecham Corp Substituted benzanilides as CCR5 receptor ligands antiinflammatory agents and antiviral agents
EP1098892A1 (en) 1998-07-20 2001-05-16 MERCK PATENT GmbH Biphenyl derivatives
BR0112856A (pt) 2000-07-31 2003-07-01 Smithkline Beecham Plc Método para o tratamento dos distúrbios, composto ou um sal ou solvato deste, processo para a preparação dos mesmos, composição farmacêutico, método de tratamento e/ou profilaxia de um ou mais dos distúrbios, uso de um composto, e, método para o tratamento de diabetes, grande depressão, depressão manìaca, ansiedade, esquizofrenia e distúrbios do sono, em mamìferos humanos e não humanos
US7105682B2 (en) 2001-01-12 2006-09-12 Amgen Inc. Substituted amine derivatives and methods of use
WO2007057742A2 (en) 2005-11-18 2007-05-24 Pfizer Products Inc. Novel piperazinone derivatives
WO2007077457A2 (en) * 2006-01-06 2007-07-12 The Royal Veterinary College Treatment of equine laminitis with 5-ht1b/ 1d antagonists
EP3348266A1 (en) 2017-01-16 2018-07-18 Leukos Biotech, S.L. Combination therapy for treating cancer

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