JP2023545730A5 - - Google Patents
Info
- Publication number
- JP2023545730A5 JP2023545730A5 JP2023521335A JP2023521335A JP2023545730A5 JP 2023545730 A5 JP2023545730 A5 JP 2023545730A5 JP 2023521335 A JP2023521335 A JP 2023521335A JP 2023521335 A JP2023521335 A JP 2023521335A JP 2023545730 A5 JP2023545730 A5 JP 2023545730A5
- Authority
- JP
- Japan
- Prior art keywords
- nitrogen
- sulfur
- oxygen
- heteroatoms independently
- independently selected
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US202063088787P | 2020-10-07 | 2020-10-07 | |
| US63/088,787 | 2020-10-07 | ||
| US202063123337P | 2020-12-09 | 2020-12-09 | |
| US63/123,337 | 2020-12-09 | ||
| PCT/US2021/071762 WO2022077010A1 (en) | 2020-10-07 | 2021-10-07 | Stat degraders and uses thereof |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2023545730A JP2023545730A (ja) | 2023-10-31 |
| JP2023545730A5 true JP2023545730A5 (enExample) | 2024-10-15 |
Family
ID=81126142
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2023521335A Pending JP2023545730A (ja) | 2020-10-07 | 2021-10-07 | Ｓｔａｔ分解剤およびそれらの使用 |
Country Status (8)
| Country | Link |
|---|---|
| US (1) | US20240293423A1 (enExample) |
| EP (1) | EP4225303A4 (enExample) |
| JP (1) | JP2023545730A (enExample) |
| AU (1) | AU2021358130A1 (enExample) |
| CA (1) | CA3194492A1 (enExample) |
| IL (1) | IL301830A (enExample) |
| MX (1) | MX2023003973A (enExample) |
| WO (1) | WO2022077010A1 (enExample) |
Families Citing this family (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN120574283A (zh) | 2019-04-05 | 2025-09-02 | 凯麦拉医疗公司 | Stat降解剂和其用途 |
| CN115677831B (zh) * | 2021-07-22 | 2026-03-17 | 杭州和正医药有限公司 | 拟肽类stat降解药物、组合物及应用 |
| CA3253876A1 (en) * | 2022-03-31 | 2023-10-05 | Recludix Pharma, Inc. | STAT MODULATORS AND THEIR USES |
| WO2024064080A1 (en) * | 2022-09-19 | 2024-03-28 | Kymera Therapeutics, Inc. | Stat6 degraders and uses thereof |
| EP4709370A2 (en) * | 2023-05-09 | 2026-03-18 | Recludix Pharma, Inc. | Stat degraders and uses thereof |
| WO2024238603A2 (en) * | 2023-05-15 | 2024-11-21 | Recludix Pharma, Inc. | Stat degraders and uses thereof |
| AU2024334590A1 (en) * | 2023-08-30 | 2026-02-19 | Kymera Therapeutics, Inc. | Stat6 degraders and uses thereof |
| WO2025217647A1 (en) * | 2024-04-12 | 2025-10-16 | Kymera Therapeutics, Inc. | Stat6 degraders and uses thereof |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN102317290A (zh) * | 2008-12-08 | 2012-01-11 | 密执安大学评议会 | Stat3抑制剂及使用stat3抑制剂的治疗方法 |
| WO2019060742A1 (en) * | 2017-09-22 | 2019-03-28 | Kymera Therapeutics, Inc | AGENTS FOR DEGRADING PROTEINS AND USES THEREOF |
| WO2020198435A1 (en) * | 2019-03-26 | 2020-10-01 | The Regents Of The University Of Michigan | Small molecule degraders of stat3 |
-
2021
- 2021-10-07 IL IL301830A patent/IL301830A/en unknown
- 2021-10-07 WO PCT/US2021/071762 patent/WO2022077010A1/en not_active Ceased
- 2021-10-07 CA CA3194492A patent/CA3194492A1/en active Pending
- 2021-10-07 MX MX2023003973A patent/MX2023003973A/es unknown
- 2021-10-07 US US18/030,865 patent/US20240293423A1/en active Pending
- 2021-10-07 AU AU2021358130A patent/AU2021358130A1/en not_active Abandoned
- 2021-10-07 JP JP2023521335A patent/JP2023545730A/ja active Pending
- 2021-10-07 EP EP21878728.1A patent/EP4225303A4/en not_active Withdrawn
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