JP2023533874A - Ｐｎ６０４７の塩酸塩の多形体 - Google Patents

Ｐｎ６０４７の塩酸塩の多形体 Download PDF

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Publication number
JP2023533874A
JP2023533874A JP2023503146A JP2023503146A JP2023533874A JP 2023533874 A JP2023533874 A JP 2023533874A JP 2023503146 A JP2023503146 A JP 2023503146A JP 2023503146 A JP2023503146 A JP 2023503146A JP 2023533874 A JP2023533874 A JP 2023533874A
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JP
Japan
Prior art keywords
crystalline
hcl2
salt
hcl salt
hcl3
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Pending
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JP2023503146A
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English (en)
Japanese (ja)
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JP2023533874A5 (https=
Inventor
メンツァー，ベンクト フォン
ストレッケ，インゲマール
ジー ニルッソン，ハンス
Original Assignee
ファームノヴォ エービー
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Application filed by ファームノヴォ エービー filed Critical ファームノヴォ エービー
Publication of JP2023533874A publication Critical patent/JP2023533874A/ja
Publication of JP2023533874A5 publication Critical patent/JP2023533874A5/ja
Priority to JP2025168607A priority Critical patent/JP2026016435A/ja
Pending legal-status Critical Current

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00—Indexing scheme relating to specific properties of organic compounds
    • C07B2200/13—Crystalline forms, e.g. polymorphs

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Plural Heterocyclic Compounds (AREA)
JP2023503146A 2020-07-17 2021-07-12 Ｐｎ６０４７の塩酸塩の多形体 Pending JP2023533874A (ja)

Priority Applications (1)

Application Number Priority Date Filing Date Title
JP2025168607A JP2026016435A (ja) 2020-07-17 2025-10-06 Ｐｎ６０４７の塩酸塩の多形体

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
SE2050910 2020-07-17
SE2050910-5 2020-07-17
PCT/EP2021/069340 WO2022013153A1 (en) 2020-07-17 2021-07-12 Polymorphs of a hydrochloride salt of pn6047

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2025168607A Division JP2026016435A (ja) 2020-07-17 2025-10-06 Ｐｎ６０４７の塩酸塩の多形体

Publications (2)

Publication Number Publication Date
JP2023533874A true JP2023533874A (ja) 2023-08-04
JP2023533874A5 JP2023533874A5 (https=) 2024-05-15

Family

ID=77168220

Family Applications (2)

Application Number Title Priority Date Filing Date
JP2023503146A Pending JP2023533874A (ja) 2020-07-17 2021-07-12 Ｐｎ６０４７の塩酸塩の多形体
JP2025168607A Pending JP2026016435A (ja) 2020-07-17 2025-10-06 Ｐｎ６０４７の塩酸塩の多形体

Family Applications After (1)

Application Number Title Priority Date Filing Date
JP2025168607A Pending JP2026016435A (ja) 2020-07-17 2025-10-06 Ｐｎ６０４７の塩酸塩の多形体

Country Status (7)

Country Link
US (1) US20230174525A1 (https=)
EP (1) EP4182312A1 (https=)
JP (2) JP2023533874A (https=)
CN (1) CN116171277B (https=)
AU (1) AU2021309364A1 (https=)
CA (1) CA3185973A1 (https=)
WO (1) WO2022013153A1 (https=)

Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2018501314A (ja) * 2014-12-19 2018-01-18 ファームノヴォ エービー ジアリールメチリデンピペリジン誘導体およびデルタオピオイド受容体アゴニストとしてそれらの使用

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SE0103313D0 (sv) * 2001-10-03 2001-10-03 Astrazeneca Ab Novel compounds
US20110207745A1 (en) * 2009-11-25 2011-08-25 Astrazeneca Ab Solid forms of 4--n,n-diethylbenzamide, compositions thereof, and uses therewith

Patent Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2018501314A (ja) * 2014-12-19 2018-01-18 ファームノヴォ エービー ジアリールメチリデンピペリジン誘導体およびデルタオピオイド受容体アゴニストとしてそれらの使用

Non-Patent Citations (2)

* Cited by examiner, † Cited by third party
Title
Ｃ．Ｇ．ＷＥＲＭＵＴＨ編, 最新 創薬化学 下巻, JPN6014029314, 1999, ISSN: 0005747387 *
芦澤一英, 医薬品の多形現象と晶析の科学, JPN6018028449, 2002, pages 56 - 102, ISSN: 0005747386 *

Also Published As

Publication number Publication date
CA3185973A1 (en) 2022-01-20
CN116171277B (zh) 2026-03-06
CN116171277A (zh) 2023-05-26
JP2026016435A (ja) 2026-02-03
EP4182312A1 (en) 2023-05-24
US20230174525A1 (en) 2023-06-08
AU2021309364A8 (en) 2023-03-16
AU2021309364A1 (en) 2023-02-16
WO2022013153A1 (en) 2022-01-20

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