JP2023521036A5 - - Google Patents

Info

Publication number
JP2023521036A5
JP2023521036A5 JP2022560245A JP2022560245A JP2023521036A5 JP 2023521036 A5 JP2023521036 A5 JP 2023521036A5 JP 2022560245 A JP2022560245 A JP 2022560245A JP 2022560245 A JP2022560245 A JP 2022560245A JP 2023521036 A5 JP2023521036 A5 JP 2023521036A5
Authority
JP
Japan
Prior art keywords
compound
pharmaceutically acceptable
acceptable salt
salt form
administered
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2022560245A
Other languages
English (en)
Japanese (ja)
Other versions
JP2023521036A (ja
JP7748386B2 (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2021/025551 external-priority patent/WO2021202981A1/en
Publication of JP2023521036A publication Critical patent/JP2023521036A/ja
Publication of JP2023521036A5 publication Critical patent/JP2023521036A5/ja
Priority to JP2025102055A priority Critical patent/JP2025120501A/ja
Application granted granted Critical
Publication of JP7748386B2 publication Critical patent/JP7748386B2/ja
Active legal-status Critical Current
Anticipated expiration legal-status Critical

Links

JP2022560245A 2020-04-03 2021-04-02 がんの治療で使用するためのミルダメチニブ及びリフィラフェニブの同時投与 Active JP7748386B2 (ja)

Priority Applications (1)

Application Number Priority Date Filing Date Title
JP2025102055A JP2025120501A (ja) 2020-04-03 2025-06-18 がんの治療で使用するためのミルダメチニブ及びリフィラフェニブの同時投与

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US202063005153P 2020-04-03 2020-04-03
US63/005,153 2020-04-03
PCT/US2021/025551 WO2021202981A1 (en) 2020-04-03 2021-04-02 Co-administration of mirdametinib and lifirafenib for use in treating cancers

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2025102055A Division JP2025120501A (ja) 2020-04-03 2025-06-18 がんの治療で使用するためのミルダメチニブ及びリフィラフェニブの同時投与

Publications (3)

Publication Number Publication Date
JP2023521036A JP2023521036A (ja) 2023-05-23
JP2023521036A5 true JP2023521036A5 (https=) 2024-04-11
JP7748386B2 JP7748386B2 (ja) 2025-10-02

Family

ID=75674969

Family Applications (2)

Application Number Title Priority Date Filing Date
JP2022560245A Active JP7748386B2 (ja) 2020-04-03 2021-04-02 がんの治療で使用するためのミルダメチニブ及びリフィラフェニブの同時投与
JP2025102055A Pending JP2025120501A (ja) 2020-04-03 2025-06-18 がんの治療で使用するためのミルダメチニブ及びリフィラフェニブの同時投与

Family Applications After (1)

Application Number Title Priority Date Filing Date
JP2025102055A Pending JP2025120501A (ja) 2020-04-03 2025-06-18 がんの治療で使用するためのミルダメチニブ及びリフィラフェニブの同時投与

Country Status (21)

Country Link
US (1) US20230128315A1 (https=)
EP (1) EP4125842B1 (https=)
JP (2) JP7748386B2 (https=)
KR (1) KR20230048476A (https=)
CN (1) CN116194095B (https=)
AU (1) AU2021246141A1 (https=)
BR (1) BR112022019914A2 (https=)
CA (1) CA3174223A1 (https=)
CL (1) CL2022002682A1 (https=)
CO (1) CO2022015891A2 (https=)
DK (1) DK4125842T3 (https=)
ES (1) ES2985012T3 (https=)
FI (1) FI4125842T3 (https=)
HU (1) HUE067894T2 (https=)
IL (1) IL296878A (https=)
MX (1) MX2022012351A (https=)
PE (1) PE20231211A1 (https=)
PL (1) PL4125842T3 (https=)
PT (1) PT4125842T (https=)
TW (1) TWI893097B (https=)
WO (1) WO2021202981A1 (https=)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA3254428A1 (en) * 2022-03-17 2023-09-21 SpringWorks Therapeutics Inc. TREATMENT OF PLEXIFORM NEUROFIBROMAS (NP) ASSOCIATED WITH TYPE 1 NEUROFIBROMATOSIS (NF1) IN PEDIATRIC PATIENTS WITH MIRDAMETINIB
WO2023178276A1 (en) * 2022-03-17 2023-09-21 SpringWorks Therapeutics Inc. Treatment of pancreatic ductal adenocarcinoma with mirdametinib
WO2023209611A1 (en) * 2022-04-26 2023-11-02 Beigene Switzerland Gmbh Methods of treating cancer with a b-raf inhibitor, in particular lifirafenib
JP2025534589A (ja) * 2022-10-14 2025-10-17 スプリングワークス、セラピューティクス、インコーポレイテッド がんの治療に使用するための併用

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
RU2013148817A (ru) * 2011-04-01 2015-05-10 Дженентек, Инк. Комбинации соединений-ингибиторов акт и мек и способы их применения
CN113307805A (zh) * 2015-04-15 2021-08-27 百济神州有限公司 B-raf激酶抑制剂的马来酸盐、其结晶形式、制备方法和用途
WO2019113345A1 (en) * 2017-12-06 2019-06-13 Spyro Mousses Combination of cancer therapeutics for treatment of cancer and hyperproliferative diseases
EP3560516A1 (en) * 2018-04-27 2019-10-30 Bergen Teknologioverforing AS Combination therapy including beta-sitosterol in combination with at least one of a braf inhibitor, a mek inhibitor or an erk inhibitor and methods and use thereof

Similar Documents

Publication Publication Date Title
JP2023521036A5 (https=)
KR20120101456A (ko) 중추 매개의 오심 및 구토를 치료하기 위한 조성물 및 방법
JP2014515373A5 (https=)
KR102490547B1 (ko) 퀴놀린 유도체로 갑상선암을 치료하기 위한 방법과 용도 및 갑상선암을 치료하기 위한 약학적 조성물
FI4125842T3 (fi) Mirdametinibin ja lifirafenibin yhteisantaminen käytettäväksi hoidettaessa syöpiä
JP2012522837A5 (https=)
KR100894465B1 (ko) 레보도파의 지속적 효과를 위한 조성물 및 제형
CN107296811A (zh) 一种用于治疗胃癌的喹啉衍生物
WO2016091165A1 (zh) 治疗非小细胞肺癌的喹啉衍生物
CN115025090A (zh) 喹啉衍生物用于治疗食管癌的用途及其治疗方法、药物组合物和试剂盒
AU2017315357A1 (en) Combination therapies for the treatment of hepatocellular carcinoma
JP2023011549A (ja) クマリン誘導体を含有する、細胞増殖性疾患の治療又は予防用医薬
CN112533600B (zh) 用于治疗小细胞肺癌的喹啉衍生物
WO2019174590A1 (zh) 用于治疗三阴性乳腺癌的喹啉衍生物
CN115243686B (zh) 丁基苯酞及其衍生物的用途
TW202327579A (zh) Tead抑制劑的給藥方案
TW201806599A (zh) 用於快速開始抗抑鬱作用之給藥方案
CN115487188A (zh) 治疗鼻咽癌的喹啉衍生物
WO2019241495A1 (en) Pharmaceutical composition and method for acute on chronic liver failure
CN106038566A (zh) 一种用于胃癌治疗的药物组合物及其应用
CN120603593A (zh) 治疗乳腺癌的方法
EP2046321A2 (en) Pharmaceutical composition containing bicalutamide and a method for its use
WO2022047196A1 (en) Pten inhibitors for treatment and prevention of bone marrow loss
CA2473602A1 (en) Oral pediatric trimethobenzamide formulations and methods
CN121130092A (zh) 抗hiv药物在抑制非小细胞肺癌耐药中的应用