JP2023503320A5 - - Google Patents
Info
- Publication number
- JP2023503320A5 JP2023503320A5 JP2022529931A JP2022529931A JP2023503320A5 JP 2023503320 A5 JP2023503320 A5 JP 2023503320A5 JP 2022529931 A JP2022529931 A JP 2022529931A JP 2022529931 A JP2022529931 A JP 2022529931A JP 2023503320 A5 JP2023503320 A5 JP 2023503320A5
- Authority
- JP
- Japan
- Prior art keywords
- methyl
- trifluoromethyl
- phenyl
- oxadiazole
- dione
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201962940061P | 2019-11-25 | 2019-11-25 | |
| US62/940,061 | 2019-11-25 | ||
| US202063106293P | 2020-10-27 | 2020-10-27 | |
| US63/106,293 | 2020-10-27 | ||
| PCT/IB2020/061053 WO2021105857A1 (en) | 2019-11-25 | 2020-11-23 | 1,2,4-oxadiazole derivatives as liver x receptor agonists |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2023503320A JP2023503320A (ja) | 2023-01-27 |
| JP2023503320A5 true JP2023503320A5 (https=) | 2023-11-29 |
Family
ID=73654860
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2022529931A Pending JP2023503320A (ja) | 2019-11-25 | 2020-11-23 | 肝臓ｘ受容体アゴニストとしての１，２，４－オキサジアゾール誘導体 |
Country Status (22)
| Country | Link |
|---|---|
| US (2) | US11427586B2 (https=) |
| EP (1) | EP4065228A1 (https=) |
| JP (1) | JP2023503320A (https=) |
| KR (1) | KR20220106778A (https=) |
| CN (1) | CN114746149A (https=) |
| AU (1) | AU2020394597B2 (https=) |
| BR (1) | BR112022009942A2 (https=) |
| CA (1) | CA3157657A1 (https=) |
| CL (1) | CL2022001323A1 (https=) |
| CO (1) | CO2022006645A2 (https=) |
| CR (1) | CR20220227A (https=) |
| DO (1) | DOP2022000107A (https=) |
| EC (1) | ECSP22040362A (https=) |
| IL (1) | IL291958A (https=) |
| JO (1) | JOP20220124A1 (https=) |
| MX (1) | MX2022006151A (https=) |
| PE (1) | PE20221785A1 (https=) |
| PH (1) | PH12022551248A1 (https=) |
| PY (1) | PY2077235A (https=) |
| TW (1) | TW202132289A (https=) |
| UY (1) | UY38964A (https=) |
| WO (1) | WO2021105857A1 (https=) |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2024518128A (ja) * | 2021-05-20 | 2024-04-24 | ノバルティス アーゲー | ３－（（３－（４－（２－（イソブチルスルホニル）フェノキシ）－３－（トリフルオロメチル）フェニル）－１，２，４－オキサジアゾール－５－イル）メチル）－５，５－ジメチル－１－（２－モルホリノエチル）イミダゾリジン－２，４－ジオンの製剤 |
| WO2022249006A1 (en) * | 2021-05-24 | 2022-12-01 | Novartis Ag | Use of 1,2,4-oxadiazole derivatives as liver x receptor agonists |
| KR102882404B1 (ko) | 2022-10-28 | 2025-11-06 | (주)케이메디켐 | 신규 옥사디아졸 유도체, 이의 제조방법 및 이를 포함하는 인지기능 개선용 조성물 |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| TW201120016A (en) | 2009-12-08 | 2011-06-16 | Abbott Lab | Novel oxadiazole compounds |
| US8729109B2 (en) * | 2011-09-08 | 2014-05-20 | Allergan, Inc. | 3-(4-(5-phenyl-1 ,2,4-oxadiazol-3-yl)phenoxy)propan-2-ol derivatives as sphingosine-1phosphate receptors modulators |
| WO2013131018A1 (en) | 2012-03-02 | 2013-09-06 | Zalicus Pharmaceuticals Ltd. | Biaryl inhibitors of the sodium channel |
| WO2015187840A2 (en) * | 2014-06-03 | 2015-12-10 | Duke University | Methods and formulations for treatment of ocular disorders |
| JP2022514257A (ja) | 2018-12-13 | 2022-02-10 | アイノス，インコーポレイテッド | ドライアイ疾患の治療のための局所点眼製剤におけるｌｘｒアゴニスト |
-
2020
- 2020-11-20 PY PY202002077235A patent/PY2077235A/es unknown
- 2020-11-20 UY UY0001038964A patent/UY38964A/es not_active Application Discontinuation
- 2020-11-23 KR KR1020227020461A patent/KR20220106778A/ko not_active Ceased
- 2020-11-23 CN CN202080081467.7A patent/CN114746149A/zh active Pending
- 2020-11-23 BR BR112022009942A patent/BR112022009942A2/pt not_active Application Discontinuation
- 2020-11-23 JP JP2022529931A patent/JP2023503320A/ja active Pending
- 2020-11-23 EP EP20817082.9A patent/EP4065228A1/en not_active Withdrawn
- 2020-11-23 CR CR20220227A patent/CR20220227A/es unknown
- 2020-11-23 IL IL291958A patent/IL291958A/en unknown
- 2020-11-23 TW TW109140930A patent/TW202132289A/zh unknown
- 2020-11-23 PH PH1/2022/551248A patent/PH12022551248A1/en unknown
- 2020-11-23 AU AU2020394597A patent/AU2020394597B2/en not_active Expired - Fee Related
- 2020-11-23 US US17/101,510 patent/US11427586B2/en active Active
- 2020-11-23 CA CA3157657A patent/CA3157657A1/en active Pending
- 2020-11-23 WO PCT/IB2020/061053 patent/WO2021105857A1/en not_active Ceased
- 2020-11-23 PE PE2022000828A patent/PE20221785A1/es unknown
- 2020-11-23 MX MX2022006151A patent/MX2022006151A/es unknown
-
2022
- 2022-05-19 EC ECSENADI202240362A patent/ECSP22040362A/es unknown
- 2022-05-19 CO CONC2022/0006645A patent/CO2022006645A2/es unknown
- 2022-05-19 CL CL2022001323A patent/CL2022001323A1/es unknown
- 2022-05-20 DO DO2022000107A patent/DOP2022000107A/es unknown
- 2022-05-23 JO JOP/2022/0124A patent/JOP20220124A1/ar unknown
- 2022-06-06 US US17/805,487 patent/US20220340573A1/en not_active Abandoned
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