JP2023501577A5 - - Google Patents
Info
- Publication number
- JP2023501577A5 JP2023501577A5 JP2022527717A JP2022527717A JP2023501577A5 JP 2023501577 A5 JP2023501577 A5 JP 2023501577A5 JP 2022527717 A JP2022527717 A JP 2022527717A JP 2022527717 A JP2022527717 A JP 2022527717A JP 2023501577 A5 JP2023501577 A5 JP 2023501577A5
- Authority
- JP
- Japan
- Prior art keywords
- alkyl
- group
- compound
- membered
- unsubstituted
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2025135739A JP2025161894A (ja) | 2019-11-13 | 2025-08-18 | ５－ヒドロキシトリプタミン受容体７の調節因子としての新規官能化ラクタムおよびその使用方法 |
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201962934997P | 2019-11-13 | 2019-11-13 | |
| US62/934,997 | 2019-11-13 | ||
| PCT/US2020/060270 WO2021097116A1 (en) | 2019-11-13 | 2020-11-12 | Novel functionalized lactams as modulators of the 5-hydroxytryptamine receptor 7 and their method of use |
Related Child Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2025135739A Division JP2025161894A (ja) | 2019-11-13 | 2025-08-18 | ５－ヒドロキシトリプタミン受容体７の調節因子としての新規官能化ラクタムおよびその使用方法 |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2023501577A JP2023501577A (ja) | 2023-01-18 |
| JP2023501577A5 true JP2023501577A5 (OSRAM) | 2023-11-20 |
| JP7730811B2 JP7730811B2 (ja) | 2025-08-28 |
Family
ID=74068668
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2022527717A Active JP7730811B2 (ja) | 2019-11-13 | 2020-11-12 | ５－ヒドロキシトリプタミン受容体７の調節因子としての新規官能化ラクタムおよびその使用方法 |
| JP2025135739A Pending JP2025161894A (ja) | 2019-11-13 | 2025-08-18 | ５－ヒドロキシトリプタミン受容体７の調節因子としての新規官能化ラクタムおよびその使用方法 |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2025135739A Pending JP2025161894A (ja) | 2019-11-13 | 2025-08-18 | ５－ヒドロキシトリプタミン受容体７の調節因子としての新規官能化ラクタムおよびその使用方法 |
Country Status (12)
| Country | Link |
|---|---|
| US (1) | US20230002383A1 (OSRAM) |
| EP (1) | EP4058455A1 (OSRAM) |
| JP (2) | JP7730811B2 (OSRAM) |
| KR (1) | KR20220113702A (OSRAM) |
| CN (1) | CN115003675A (OSRAM) |
| AU (1) | AU2020381460A1 (OSRAM) |
| BR (1) | BR112022009374A2 (OSRAM) |
| CA (1) | CA3160801A1 (OSRAM) |
| IL (1) | IL292811A (OSRAM) |
| MX (1) | MX2022005820A (OSRAM) |
| TW (1) | TWI905129B (OSRAM) |
| WO (1) | WO2021097116A1 (OSRAM) |
Families Citing this family (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US10961249B2 (en) | 2017-03-21 | 2021-03-30 | Temple University-Of The Commonwealth System Of Higher Education | Modulators of the sigma-2 receptor and their method of use |
| BR112020023072A2 (pt) | 2018-05-11 | 2021-02-02 | Temple University-Of The Commonwealth System Of Higher Education | novos lactâmicos funcionalizados como moduladores do receptor 7 de 5-hidroxitriptamina e seu método de uso |
Family Cites Families (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB201002563D0 (en) * | 2010-02-15 | 2010-03-31 | Cambridge Entpr Ltd | Compounds |
| WO2014164756A1 (en) * | 2013-03-11 | 2014-10-09 | Temple University Of The Commonwealth System Of Higher Education | Novel 5-hydroxytryptamine receptor 7 activity modulators and their method of use |
| EP3200589B1 (en) * | 2014-09-10 | 2026-03-11 | Temple University Of The Commonwealth System Of Higher Education | Novel 5-hydroxytryptamine receptor 7 activity modulators and their method of use |
| EP3541790B1 (en) * | 2016-11-15 | 2025-09-03 | Temple University - Of The Commonwealth System of Higher Education | 3-(2-(4-phenylpiperazin-1-yl)ethyl)-2-oxa-8-azaspiro[4.5]decan-1-one derivatives and related compounds as 5-hydroxytryptamine receptor 7 (5-ht7) modulators for treating e.g. inflammatory bowel disease, circadian rhythm disorder or depression |
| JP7365238B2 (ja) * | 2017-03-21 | 2023-10-19 | テンプル・ユニバーシティ－オブ・ザ・コモンウェルス・システム・オブ・ハイアー・エデュケイション | ５－ヒドロキシトリプタミン受容体７調節物質および治療剤としてのその使用 |
| US11365195B2 (en) * | 2017-11-13 | 2022-06-21 | The United States Of America, As Represented By The Secretary, Department Of Health And Human Services | Atypical inhibitors of monoamine transporters; method of making; and use thereof |
| BR112020023072A2 (pt) * | 2018-05-11 | 2021-02-02 | Temple University-Of The Commonwealth System Of Higher Education | novos lactâmicos funcionalizados como moduladores do receptor 7 de 5-hidroxitriptamina e seu método de uso |
-
2020
- 2020-11-12 KR KR1020227019540A patent/KR20220113702A/ko active Pending
- 2020-11-12 BR BR112022009374A patent/BR112022009374A2/pt unknown
- 2020-11-12 JP JP2022527717A patent/JP7730811B2/ja active Active
- 2020-11-12 CN CN202080093159.6A patent/CN115003675A/zh active Pending
- 2020-11-12 AU AU2020381460A patent/AU2020381460A1/en active Pending
- 2020-11-12 EP EP20829736.6A patent/EP4058455A1/en active Pending
- 2020-11-12 MX MX2022005820A patent/MX2022005820A/es unknown
- 2020-11-12 US US17/776,533 patent/US20230002383A1/en active Pending
- 2020-11-12 WO PCT/US2020/060270 patent/WO2021097116A1/en not_active Ceased
- 2020-11-12 CA CA3160801A patent/CA3160801A1/en active Pending
- 2020-11-13 TW TW109139761A patent/TWI905129B/zh active
-
2022
- 2022-05-07 IL IL292811A patent/IL292811A/en unknown
-
2025
- 2025-08-18 JP JP2025135739A patent/JP2025161894A/ja active Pending
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