JP2023022224A5 - - Google Patents

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Publication number
JP2023022224A5
JP2023022224A5 JP2022191728A JP2022191728A JP2023022224A5 JP 2023022224 A5 JP2023022224 A5 JP 2023022224A5 JP 2022191728 A JP2022191728 A JP 2022191728A JP 2022191728 A JP2022191728 A JP 2022191728A JP 2023022224 A5 JP2023022224 A5 JP 2023022224A5
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JP
Japan
Prior art keywords
invention described
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Application number
JP2022191728A
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English (en)
Japanese (ja)
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JP7561814B2 (ja
JP2023022224A (ja
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Priority claimed from US15/859,279 external-priority patent/US20180338922A1/en
Application filed filed Critical
Publication of JP2023022224A publication Critical patent/JP2023022224A/ja
Publication of JP2023022224A5 publication Critical patent/JP2023022224A5/ja
Priority to JP2024164776A priority Critical patent/JP2024178341A/ja
Application granted granted Critical
Publication of JP7561814B2 publication Critical patent/JP7561814B2/ja
Active legal-status Critical Current
Anticipated expiration legal-status Critical

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JP2022191728A 2017-05-26 2022-11-30 固定用量製剤 Active JP7561814B2 (ja)

Priority Applications (1)

Application Number Priority Date Filing Date Title
JP2024164776A JP2024178341A (ja) 2017-05-26 2024-09-24 固定用量製剤

Applications Claiming Priority (6)

Application Number Priority Date Filing Date Title
US201762511889P 2017-05-26 2017-05-26
US62/511,889 2017-05-26
US15/859,279 2017-12-29
US15/859,279 US20180338922A1 (en) 2017-05-26 2017-12-29 Fixed dose formulations
JP2019565302A JP7187488B2 (ja) 2017-05-26 2018-05-25 固定用量製剤
PCT/US2018/034646 WO2018218147A1 (en) 2017-05-26 2018-05-25 Fixed dose formulations

Related Parent Applications (1)

Application Number Title Priority Date Filing Date
JP2019565302A Division JP7187488B2 (ja) 2017-05-26 2018-05-25 固定用量製剤

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2024164776A Division JP2024178341A (ja) 2017-05-26 2024-09-24 固定用量製剤

Publications (3)

Publication Number Publication Date
JP2023022224A JP2023022224A (ja) 2023-02-14
JP2023022224A5 true JP2023022224A5 (enExample) 2023-04-10
JP7561814B2 JP7561814B2 (ja) 2024-10-04

Family

ID=62621055

Family Applications (3)

Application Number Title Priority Date Filing Date
JP2019565302A Active JP7187488B2 (ja) 2017-05-26 2018-05-25 固定用量製剤
JP2022191728A Active JP7561814B2 (ja) 2017-05-26 2022-11-30 固定用量製剤
JP2024164776A Pending JP2024178341A (ja) 2017-05-26 2024-09-24 固定用量製剤

Family Applications Before (1)

Application Number Title Priority Date Filing Date
JP2019565302A Active JP7187488B2 (ja) 2017-05-26 2018-05-25 固定用量製剤

Family Applications After (1)

Application Number Title Priority Date Filing Date
JP2024164776A Pending JP2024178341A (ja) 2017-05-26 2024-09-24 固定用量製剤

Country Status (15)

Country Link
US (2) US20180338922A1 (enExample)
EP (1) EP3630070A1 (enExample)
JP (3) JP7187488B2 (enExample)
KR (3) KR20250109242A (enExample)
CN (1) CN110996914A (enExample)
AU (2) AU2018272040A1 (enExample)
BR (1) BR112019024747A2 (enExample)
CA (1) CA3064895A1 (enExample)
CL (1) CL2019003437A1 (enExample)
IL (2) IL318957A (enExample)
MX (2) MX2019014122A (enExample)
PH (1) PH12019502782A1 (enExample)
TW (2) TW202400126A (enExample)
UA (1) UA126451C2 (enExample)
WO (1) WO2018218147A1 (enExample)

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MA42616A (fr) 2015-03-13 2021-05-19 Esperion Therapeutics Inc Combinaisons et formulations de doses fixes comprenant etc1002 et ézétimibe, et procédés de traitement ou de réduction du risque de maladie cardio-vasculaire
WO2019161307A1 (en) * 2018-02-16 2019-08-22 Esperion Therapeutics, Inc. Sustained release formulations of bempedoic acid
WO2020046836A1 (en) * 2018-08-27 2020-03-05 Esperion Therapeutics, Inc. Combination drug formulations for treating patients with cardiovascular disease and associated conditions
EP3666750A1 (en) * 2018-12-10 2020-06-17 Sandoz AG Crystalline form of bempedoic acid
WO2020213010A1 (en) * 2019-04-16 2020-10-22 Celagenex Research (India) Pvt. Ltd. Synergistic lipid controlling compositions
CA3144372A1 (en) 2019-06-21 2020-12-24 Esperion Therapeutics, Inc. Salt forms of bempedoic acid and methods for using the same
EP4038045A1 (en) 2019-10-03 2022-08-10 Synthon B.V. Crystalline forms of bempedoic acid
WO2021110929A1 (en) 2019-12-06 2021-06-10 Synthon B.V. Crystalline forms of sodium salt of bempedoic acid
WO2021205887A1 (ja) * 2020-04-10 2021-10-14 日本酢ビ・ポバール株式会社 徐放性基剤
WO2021220236A1 (en) * 2020-05-01 2021-11-04 Cadila Healthcare Limited Pharmaceutical compositions for combination therapy
CN111559961A (zh) * 2020-05-26 2020-08-21 杭州科巢生物科技有限公司 一种贝派地酸晶型及其制备方法
WO2021255180A1 (en) 2020-06-19 2021-12-23 Synthon B.V. Salts of bempedoic acid
US20250134841A1 (en) * 2021-09-13 2025-05-01 Synthon B.V. Pharmaceutical composition of bempedoic acid
CA3256768A1 (en) 2022-05-09 2023-11-16 Renata Pharmaceutical (Ireland) Ltd PHARMACEUTICAL COMPOSITION OF BEMPEDOIC ACID

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Publication number Priority date Publication date Assignee Title
US5631365A (en) 1993-09-21 1997-05-20 Schering Corporation Hydroxy-substituted azetidinone compounds useful as hypocholesterolemic agents
ES2274013T3 (es) 2001-01-26 2007-05-16 Schering Corporation Combinaciones de activador(es) del receptor activado por el proliferador de los peroxisomas (ppar) e inhibidor(es)m de la absorcion de estelores y tratamientos para trastornos vasculares.
JP4438268B2 (ja) * 2001-03-07 2010-03-24 大日本住友製薬株式会社 薬物顆粒の製造方法、および薬物顆粒、ならびにそれを用いた医薬製剤
US7053080B2 (en) * 2001-09-21 2006-05-30 Schering Corporation Methods and therapeutic combinations for the treatment of obesity using sterol absorption inhibitors
WO2004067489A2 (en) 2003-01-23 2004-08-12 Esperion Therapeutics, Inc. Hydroxyl compounds and compositions for cholesterol management and related uses
NZ592194A (en) * 2008-09-17 2013-04-26 Mylan Inc Reversed wet granulation process for preparing granulates and pharmaceutical products containing them
JO3239B1 (ar) * 2008-09-22 2018-03-08 Novartis Ag تركيبات جالينية من مركبات عضوية
EP2168573A1 (en) * 2008-09-30 2010-03-31 LEK Pharmaceuticals D.D. Formulations comprising ezetimibe
NZ595071A (en) * 2009-03-13 2013-01-25 Toyama Chemical Co Ltd Tablet and granulated powder containing 6-fluoro-3-hydroxy-2-pyrazinecarboxamide
EP2229938B9 (en) * 2009-03-13 2012-04-25 Sanovel Ilac Sanayi ve Ticaret A.S. Ezetimibe compositions
HUE038048T2 (hu) * 2009-07-28 2018-09-28 Egyt Gyogyszervegyeszeti Gyar Új granulálási eljárás és ezzel elõállított granulátum
CN101926756B (zh) * 2010-08-12 2012-01-18 北京赛科药业有限责任公司 一种氯吡格雷或其药学上可接受盐的固体制剂
AR083417A1 (es) * 2010-10-14 2013-02-21 Novartis Ag Composiciones farmaceuticas que contienen un dgat1 inhibidor
EP2468258A1 (en) * 2010-12-22 2012-06-27 LEK Pharmaceuticals d.d. Process for the preparation of a pharmaceutical composition comprising a low soluble pharmaceutically active ingredient
AR086675A1 (es) * 2011-06-14 2014-01-15 Merck Sharp & Dohme Composiciones farmaceuticas de combinaciones de inhibidores de la dipeptidil peptidasa-4 con simvastatina
WO2013023250A1 (en) * 2011-08-16 2013-02-21 Baker Idi Heart & Diabetes Institute Holdings Limited Controlled-release formulation
MX378845B (es) * 2014-01-21 2025-03-10 Bpsi Holdings Llc Revestimientos de pelicula de liberacion inmediata que contienen gliceridos de cadena media y sustratos revestidos con los mismos.
MA42616A (fr) * 2015-03-13 2021-05-19 Esperion Therapeutics Inc Combinaisons et formulations de doses fixes comprenant etc1002 et ézétimibe, et procédés de traitement ou de réduction du risque de maladie cardio-vasculaire
MA41793A (fr) * 2015-03-16 2018-01-23 Esperion Therapeutics Inc Associations de doses fixes comprenant du etc1002 et une ou plusieurs statines permettant de traiter ou de réduire un risque cardiovasculaire
WO2017023165A1 (en) * 2015-08-04 2017-02-09 Dezima Pharma B.V. Pharmaceutical composition and therapeutic combination comprising a cholesteryl ester transfer protein inhibitor and an atp citrate lyase inhibitor – ampk activator
JP2018536710A (ja) * 2015-11-06 2018-12-13 ジェンファイア・セラピューティクス・インコーポレイテッドGemphire Therapeutics Inc. 混合型脂質異常症の治療

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