JP2022554019A5 - - Google Patents

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Publication number
JP2022554019A5
JP2022554019A5 JP2022525889A JP2022525889A JP2022554019A5 JP 2022554019 A5 JP2022554019 A5 JP 2022554019A5 JP 2022525889 A JP2022525889 A JP 2022525889A JP 2022525889 A JP2022525889 A JP 2022525889A JP 2022554019 A5 JP2022554019 A5 JP 2022554019A5
Authority
JP
Japan
Prior art keywords
pharmaceutical composition
composition according
free base
disease
disorder
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Withdrawn
Application number
JP2022525889A
Other languages
English (en)
Japanese (ja)
Other versions
JP2022554019A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2020/059287 external-priority patent/WO2021092292A1/en
Publication of JP2022554019A publication Critical patent/JP2022554019A/ja
Publication of JP2022554019A5 publication Critical patent/JP2022554019A5/ja
Withdrawn legal-status Critical Current

Links

JP2022525889A 2019-11-08 2020-11-06 補体成分C5a受容体の遊離塩基結晶形態 Withdrawn JP2022554019A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201962932652P 2019-11-08 2019-11-08
US62/932,652 2019-11-08
PCT/US2020/059287 WO2021092292A1 (en) 2019-11-08 2020-11-06 FREE BASE CRYSTALLINE FORM OF A COMPLEMENT COMPONENT C5a RECEPTOR

Publications (2)

Publication Number Publication Date
JP2022554019A JP2022554019A (ja) 2022-12-27
JP2022554019A5 true JP2022554019A5 (https=) 2023-11-09

Family

ID=75846182

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2022525889A Withdrawn JP2022554019A (ja) 2019-11-08 2020-11-06 補体成分C5a受容体の遊離塩基結晶形態

Country Status (13)

Country Link
US (3) US11026935B2 (https=)
EP (1) EP4054577A4 (https=)
JP (1) JP2022554019A (https=)
KR (1) KR20220098179A (https=)
CN (1) CN114641289A (https=)
AU (1) AU2020378061A1 (https=)
BR (1) BR112022007488A2 (https=)
CA (1) CA3155596A1 (https=)
CL (1) CL2022001173A1 (https=)
IL (1) IL292317A (https=)
MX (1) MX2022005403A (https=)
WO (1) WO2021092292A1 (https=)
ZA (1) ZA202305622B (https=)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN114867473A (zh) 2019-11-08 2022-08-05 凯莫森特里克斯股份有限公司 补体成分c5a受体的盐形式
US11603356B2 (en) 2019-11-08 2023-03-14 Chemocentryx, Inc. Amorphous form of a complement component C5a receptor
JP2022554019A (ja) * 2019-11-08 2022-12-27 ケモセントリックス,インコーポレイティド 補体成分C5a受容体の遊離塩基結晶形態
WO2022078269A1 (zh) * 2020-10-16 2022-04-21 苏州科睿思制药有限公司 Avacopan的晶型及其制备方法和用途
JP7839157B2 (ja) * 2020-10-28 2026-04-01 ケモセントリックス, インコーポレイテッド 化膿性汗腺炎を処置する方法
EP4137133A1 (en) 2021-08-19 2023-02-22 Sandoz AG Crystalline form of avacopan
WO2022263263A1 (en) 2021-06-16 2022-12-22 Sandoz Ag Crystalline form of avacopan
US20260027049A1 (en) 2024-07-23 2026-01-29 Amgen Inc. Avacopan formulations

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP4996467B2 (ja) * 2004-09-27 2012-08-08 アカディア ファーマシューティカルズ インコーポレイテッド N−(4−フルオロベンジル)−n−(1−メチルピペリジン−4−イル)−n’−(4−(2−メチルプロピルオキシ)フェニルメチル)カルバミド、並びにその酒石酸塩及び結晶形態の合成
RS54998B1 (sr) 2008-12-22 2016-11-30 Chemocentryx Inc Antagonisti c5ar
US20110275639A1 (en) 2008-12-22 2011-11-10 Chemocentryx, Inc. C5aR ANTAGONISTS
RS56332B1 (sr) 2010-06-24 2017-12-29 Chemocentryx Inc Antagonisti c5ar
DK3200791T3 (da) 2014-09-29 2020-05-25 Chemocentryx Inc Fremgangsmåder og mellemprodukter i fremstilling af C5AR- antagonister
CN114867473A (zh) * 2019-11-08 2022-08-05 凯莫森特里克斯股份有限公司 补体成分c5a受体的盐形式
JP2022554019A (ja) * 2019-11-08 2022-12-27 ケモセントリックス,インコーポレイティド 補体成分C5a受容体の遊離塩基結晶形態
WO2022078269A1 (zh) * 2020-10-16 2022-04-21 苏州科睿思制药有限公司 Avacopan的晶型及其制备方法和用途

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