JP2022546717A5 - - Google Patents

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Publication number
JP2022546717A5
JP2022546717A5 JP2022514513A JP2022514513A JP2022546717A5 JP 2022546717 A5 JP2022546717 A5 JP 2022546717A5 JP 2022514513 A JP2022514513 A JP 2022514513A JP 2022514513 A JP2022514513 A JP 2022514513A JP 2022546717 A5 JP2022546717 A5 JP 2022546717A5
Authority
JP
Japan
Application number
JP2022514513A
Other languages
Japanese (ja)
Other versions
JP2022546717A (ja
JPWO2021043870A5 (https=
Filing date
Publication date
Priority claimed from GBGB1912674.7A external-priority patent/GB201912674D0/en
Application filed filed Critical
Publication of JP2022546717A publication Critical patent/JP2022546717A/ja
Publication of JPWO2021043870A5 publication Critical patent/JPWO2021043870A5/ja
Publication of JP2022546717A5 publication Critical patent/JP2022546717A5/ja
Ceased legal-status Critical Current

Links

JP2022514513A 2019-09-04 2020-09-03 Usp30阻害剤としての活性を有する置換シアノピロリジン類 Ceased JP2022546717A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GBGB1912674.7A GB201912674D0 (en) 2019-09-04 2019-09-04 Novel compounds
GB1912674.7 2019-09-04
PCT/EP2020/074540 WO2021043870A1 (en) 2019-09-04 2020-09-03 Substituted cyanopyrrolidines with activity as usp30 inhibitors

Publications (3)

Publication Number Publication Date
JP2022546717A JP2022546717A (ja) 2022-11-07
JPWO2021043870A5 JPWO2021043870A5 (https=) 2023-09-11
JP2022546717A5 true JP2022546717A5 (https=) 2023-09-11

Family

ID=68207049

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2022514513A Ceased JP2022546717A (ja) 2019-09-04 2020-09-03 Usp30阻害剤としての活性を有する置換シアノピロリジン類

Country Status (14)

Country Link
US (1) US20220315572A1 (https=)
EP (1) EP4025573B9 (https=)
JP (1) JP2022546717A (https=)
KR (1) KR20220054867A (https=)
CN (1) CN114341133B (https=)
AU (1) AU2020340527A1 (https=)
BR (1) BR112022003527A2 (https=)
CA (1) CA3146040A1 (https=)
CO (1) CO2022003608A2 (https=)
GB (1) GB201912674D0 (https=)
IL (1) IL290929B2 (https=)
MX (1) MX2022002686A (https=)
WO (1) WO2021043870A1 (https=)
ZA (1) ZA202203775B (https=)

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JP7449242B2 (ja) 2018-05-17 2024-03-13 フォーマ セラピューティクス,インコーポレイテッド ユビキチン特異的ペプチダーゼ30(usp30)阻害剤として有用な縮合二環化合物
LT3860989T (lt) * 2018-10-05 2023-06-12 Forma Therapeutics, Inc. Sulieti pirolinai, kurie veikia kaip ubikvitinui specifinės proteazės 30 (ups30) inhibitoriai
WO2021204856A1 (en) 2020-04-08 2021-10-14 Mission Therapeutics Limited N-cyanopyrrolidines with activity as usp30 inhibitors
IL298526A (en) 2020-05-28 2023-01-01 Mission Therapeutics Ltd N-(1-cyano-pyrrolidin-3-yl)-5-(3-(trifluoromethyl)phenyl)oxazole-2-carboxamide derivatives and the corresponding oxadiazole derivatives as usp30 inhibitors for the treatment of mitochondrial dysfunction
BR112022019722A2 (pt) 2020-06-04 2022-12-20 Mission Therapeutics Ltd N-cianopirrolidinas com atividade como inibidores de usp30
DK4161929T3 (da) 2020-06-08 2025-08-18 Mission Therapeutics Ltd 1-(5-(2-cyanopyridin-4-yl)oxazol-2-carbonyl)-4-methylhexahydropyrrolo[3,4-b]pyrrol-5(1h)-carbonitril som usp30-hæmmer til anvendelse i behandling af mitokondriedysfunktion, cancer og fibrose
GB202016800D0 (en) 2020-10-22 2020-12-09 Mission Therapeutics Ltd Novel compounds
US20250034122A1 (en) 2021-12-01 2025-01-30 Mission Therapeutics Limited Substituted n-cyanopyrrolidines with activity as usp30 inhibitors
KR20240132148A (ko) * 2023-02-24 2024-09-03 연세대학교 산학협력단 인덴 유도체를 유효성분으로 포함하는 섬유화의 예방 또는 치료용 조성물
GB202408928D0 (en) 2024-06-21 2024-08-07 Mission Therapeutics Ltd Novel compounds
GB202411060D0 (en) 2024-07-29 2024-09-11 Mission Therapeutics Ltd Novel compounds

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LT3860989T (lt) 2018-10-05 2023-06-12 Forma Therapeutics, Inc. Sulieti pirolinai, kurie veikia kaip ubikvitinui specifinės proteazės 30 (ups30) inhibitoriai
IL298526A (en) * 2020-05-28 2023-01-01 Mission Therapeutics Ltd N-(1-cyano-pyrrolidin-3-yl)-5-(3-(trifluoromethyl)phenyl)oxazole-2-carboxamide derivatives and the corresponding oxadiazole derivatives as usp30 inhibitors for the treatment of mitochondrial dysfunction

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