JP2022533747A5 - - Google Patents

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Publication number
JP2022533747A5
JP2022533747A5 JP2021569238A JP2021569238A JP2022533747A5 JP 2022533747 A5 JP2022533747 A5 JP 2022533747A5 JP 2021569238 A JP2021569238 A JP 2021569238A JP 2021569238 A JP2021569238 A JP 2021569238A JP 2022533747 A5 JP2022533747 A5 JP 2022533747A5
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JP
Japan
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formula
compound
process according
reaction
salt
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JP2021569238A
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English (en)
Japanese (ja)
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JP7658916B2 (ja
JP2022533747A (ja
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Priority claimed from PCT/EP2020/064123 external-priority patent/WO2020234381A1/en
Publication of JP2022533747A publication Critical patent/JP2022533747A/ja
Publication of JP2022533747A5 publication Critical patent/JP2022533747A5/ja
Application granted granted Critical
Publication of JP7658916B2 publication Critical patent/JP7658916B2/ja
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JP2021569238A 2019-05-21 2020-05-20 Btk阻害剤を調製するためのプロセス及び中間体 Active JP7658916B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
CN2019087823 2019-05-21
CNPCT/CN2019/087823 2019-05-21
PCT/EP2020/064123 WO2020234381A1 (en) 2019-05-21 2020-05-20 Processes and intermediates for preparing a btk inhibitor

Publications (3)

Publication Number Publication Date
JP2022533747A JP2022533747A (ja) 2022-07-25
JP2022533747A5 true JP2022533747A5 (https=) 2024-12-09
JP7658916B2 JP7658916B2 (ja) 2025-04-08

Family

ID=70857160

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2021569238A Active JP7658916B2 (ja) 2019-05-21 2020-05-20 Btk阻害剤を調製するためのプロセス及び中間体

Country Status (11)

Country Link
US (1) US12215110B2 (https=)
EP (1) EP3972977A1 (https=)
JP (1) JP7658916B2 (https=)
KR (1) KR20220011668A (https=)
CN (1) CN113874378A (https=)
AU (1) AU2020278162A1 (https=)
BR (1) BR112021022347A2 (https=)
CA (1) CA3135240A1 (https=)
IL (1) IL288154A (https=)
MX (1) MX2021014246A (https=)
WO (1) WO2020234381A1 (https=)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US12450495B2 (en) 2022-06-13 2025-10-21 International Business Machines Corporation Neural capacitance: neural network selection via edge dynamics

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DK2526933T3 (en) * 2006-09-22 2015-05-18 Pharmacyclics Inc Inhibitors of Bruton's tyrosine kinase
PT2414363E (pt) * 2009-03-31 2014-02-26 Boehringer Ingelheim Int Derivados de 1-heterociclil-1,5-di-hidro-pirazolo[3,4- d]pirimidin-4-ona e sua utilização como moduladores de pde9a
CN103121999A (zh) * 2012-08-29 2013-05-29 苏州迪飞医药科技有限公司 一种酪氨酸激酶抑制剂pci-32765的合成方法
US9156847B2 (en) * 2013-03-15 2015-10-13 Janssen Pharmaceutica Nv Processes and intermediates for preparing a medicament
CA2901510C (en) * 2013-03-15 2022-11-29 Janssen Pharmaceutica Nv Processes for preparing ibrutinib derivatives and intermediates thereof
SI3057969T1 (sl) 2013-10-17 2018-10-30 Blueprint Medicines Corporation Sestavki, uporabni za zdravljenje motenj, povezanih s KIT
MA41350A (fr) 2015-01-14 2017-11-21 Janssen Pharmaceutica Nv Synthèse d'un inhibiteur de la tyrosine kinase de bruton
JP6681922B2 (ja) 2015-02-12 2020-04-15 上▲海▼度▲徳▼医▲藥▼科技有限公司 イブルチニブの製造方法

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