JP2022533747A5 - - Google Patents
Info
- Publication number
- JP2022533747A5 JP2022533747A5 JP2021569238A JP2021569238A JP2022533747A5 JP 2022533747 A5 JP2022533747 A5 JP 2022533747A5 JP 2021569238 A JP2021569238 A JP 2021569238A JP 2021569238 A JP2021569238 A JP 2021569238A JP 2022533747 A5 JP2022533747 A5 JP 2022533747A5
- Authority
- JP
- Japan
- Prior art keywords
- formula
- compound
- process according
- reaction
- salt
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| CN2019087823 | 2019-05-21 | ||
| CNPCT/CN2019/087823 | 2019-05-21 | ||
| PCT/EP2020/064123 WO2020234381A1 (en) | 2019-05-21 | 2020-05-20 | Processes and intermediates for preparing a btk inhibitor |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2022533747A JP2022533747A (ja) | 2022-07-25 |
| JP2022533747A5 true JP2022533747A5 (https=) | 2024-12-09 |
| JP7658916B2 JP7658916B2 (ja) | 2025-04-08 |
Family
ID=70857160
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2021569238A Active JP7658916B2 (ja) | 2019-05-21 | 2020-05-20 | Btk阻害剤を調製するためのプロセス及び中間体 |
Country Status (11)
| Country | Link |
|---|---|
| US (1) | US12215110B2 (https=) |
| EP (1) | EP3972977A1 (https=) |
| JP (1) | JP7658916B2 (https=) |
| KR (1) | KR20220011668A (https=) |
| CN (1) | CN113874378A (https=) |
| AU (1) | AU2020278162A1 (https=) |
| BR (1) | BR112021022347A2 (https=) |
| CA (1) | CA3135240A1 (https=) |
| IL (1) | IL288154A (https=) |
| MX (1) | MX2021014246A (https=) |
| WO (1) | WO2020234381A1 (https=) |
Families Citing this family (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US12450495B2 (en) | 2022-06-13 | 2025-10-21 | International Business Machines Corporation | Neural capacitance: neural network selection via edge dynamics |
Family Cites Families (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DK2526933T3 (en) * | 2006-09-22 | 2015-05-18 | Pharmacyclics Inc | Inhibitors of Bruton's tyrosine kinase |
| PT2414363E (pt) * | 2009-03-31 | 2014-02-26 | Boehringer Ingelheim Int | Derivados de 1-heterociclil-1,5-di-hidro-pirazolo[3,4- d]pirimidin-4-ona e sua utilização como moduladores de pde9a |
| CN103121999A (zh) * | 2012-08-29 | 2013-05-29 | 苏州迪飞医药科技有限公司 | 一种酪氨酸激酶抑制剂pci-32765的合成方法 |
| US9156847B2 (en) * | 2013-03-15 | 2015-10-13 | Janssen Pharmaceutica Nv | Processes and intermediates for preparing a medicament |
| CA2901510C (en) * | 2013-03-15 | 2022-11-29 | Janssen Pharmaceutica Nv | Processes for preparing ibrutinib derivatives and intermediates thereof |
| SI3057969T1 (sl) | 2013-10-17 | 2018-10-30 | Blueprint Medicines Corporation | Sestavki, uporabni za zdravljenje motenj, povezanih s KIT |
| MA41350A (fr) | 2015-01-14 | 2017-11-21 | Janssen Pharmaceutica Nv | Synthèse d'un inhibiteur de la tyrosine kinase de bruton |
| JP6681922B2 (ja) | 2015-02-12 | 2020-04-15 | 上▲海▼度▲徳▼医▲藥▼科技有限公司 | イブルチニブの製造方法 |
-
2020
- 2020-05-20 WO PCT/EP2020/064123 patent/WO2020234381A1/en not_active Ceased
- 2020-05-20 BR BR112021022347A patent/BR112021022347A2/pt unknown
- 2020-05-20 US US17/612,082 patent/US12215110B2/en active Active
- 2020-05-20 EP EP20728440.7A patent/EP3972977A1/en active Pending
- 2020-05-20 MX MX2021014246A patent/MX2021014246A/es unknown
- 2020-05-20 JP JP2021569238A patent/JP7658916B2/ja active Active
- 2020-05-20 KR KR1020217041326A patent/KR20220011668A/ko not_active Withdrawn
- 2020-05-20 AU AU2020278162A patent/AU2020278162A1/en not_active Abandoned
- 2020-05-20 CN CN202080037397.5A patent/CN113874378A/zh active Pending
- 2020-05-20 CA CA3135240A patent/CA3135240A1/en active Pending
-
2021
- 2021-11-16 IL IL288154A patent/IL288154A/en unknown
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