JP2022533182A5 - - Google Patents

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Publication number
JP2022533182A5
JP2022533182A5 JP2021568650A JP2021568650A JP2022533182A5 JP 2022533182 A5 JP2022533182 A5 JP 2022533182A5 JP 2021568650 A JP2021568650 A JP 2021568650A JP 2021568650 A JP2021568650 A JP 2021568650A JP 2022533182 A5 JP2022533182 A5 JP 2022533182A5
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JP
Japan
Application number
JP2021568650A
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Japanese (ja)
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JP2022533182A (ja
JP7546603B2 (ja
JPWO2020232190A5 (https=
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Priority claimed from PCT/US2020/032784 external-priority patent/WO2020232190A1/en
Publication of JP2022533182A publication Critical patent/JP2022533182A/ja
Publication of JP2022533182A5 publication Critical patent/JP2022533182A5/ja
Publication of JPWO2020232190A5 publication Critical patent/JPWO2020232190A5/ja
Priority to JP2024145040A priority Critical patent/JP2024170457A/ja
Application granted granted Critical
Publication of JP7546603B2 publication Critical patent/JP7546603B2/ja
Active legal-status Critical Current
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JP2021568650A 2019-05-16 2020-05-14 タンパク質キナーゼ阻害剤ならびに疾患および状態の治療のためのその使用 Active JP7546603B2 (ja)

Priority Applications (1)

Application Number Priority Date Filing Date Title
JP2024145040A JP2024170457A (ja) 2019-05-16 2024-08-27 タンパク質キナーゼ阻害剤ならびに疾患および状態の治療のためのその使用

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US201962848648P 2019-05-16 2019-05-16
US201962848719P 2019-05-16 2019-05-16
US62/848,648 2019-05-16
US62/848,719 2019-05-16
PCT/US2020/032784 WO2020232190A1 (en) 2019-05-16 2020-05-14 Protein kinase inhibitors and uses thereof for the treatment of diseases and conditions

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2024145040A Division JP2024170457A (ja) 2019-05-16 2024-08-27 タンパク質キナーゼ阻害剤ならびに疾患および状態の治療のためのその使用

Publications (4)

Publication Number Publication Date
JP2022533182A JP2022533182A (ja) 2022-07-21
JP2022533182A5 true JP2022533182A5 (https=) 2023-05-02
JPWO2020232190A5 JPWO2020232190A5 (https=) 2023-05-02
JP7546603B2 JP7546603B2 (ja) 2024-09-06

Family

ID=70919255

Family Applications (2)

Application Number Title Priority Date Filing Date
JP2021568650A Active JP7546603B2 (ja) 2019-05-16 2020-05-14 タンパク質キナーゼ阻害剤ならびに疾患および状態の治療のためのその使用
JP2024145040A Pending JP2024170457A (ja) 2019-05-16 2024-08-27 タンパク質キナーゼ阻害剤ならびに疾患および状態の治療のためのその使用

Family Applications After (1)

Application Number Title Priority Date Filing Date
JP2024145040A Pending JP2024170457A (ja) 2019-05-16 2024-08-27 タンパク質キナーゼ阻害剤ならびに疾患および状態の治療のためのその使用

Country Status (6)

Country Link
US (1) US12516055B2 (https=)
EP (2) EP4480485A3 (https=)
JP (2) JP7546603B2 (https=)
AU (1) AU2020275304B2 (https=)
CA (1) CA3137869A1 (https=)
WO (1) WO2020232190A1 (https=)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US11174255B2 (en) * 2017-05-15 2021-11-16 University Of Houston System Pyrido[2,3-d]pyrimidin-7-ones and related compounds as inhibitors of protein kinases
EP4480485A3 (en) * 2019-05-16 2025-02-26 University of Houston System Protein kinase inhibitors and uses thereof for the treatment of diseases and conditions
CN113072471B (zh) * 2021-03-02 2022-09-16 四川美大康华康药业有限公司 一种利非司特中间体及其制备方法
WO2024097805A1 (en) * 2022-11-01 2024-05-10 Trustees Of Tufts College Mixed lineage kinase domain like pseudokinase (mlkl) activators
WO2024199388A1 (zh) * 2023-03-29 2024-10-03 微境生物医药科技(上海)有限公司 作为myt1抑制剂的化合物

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IL117923A (en) 1995-05-03 2000-06-01 Warner Lambert Co Anti-cancer pharmaceutical compositions containing polysubstituted pyrido¬2,3-d¾pyrimidine derivatives and certain such novel compounds
US6150359A (en) * 1997-08-20 2000-11-21 Warner-Lambert Company Naphthyridinones for inhibiting protein tyrosine kinase and cell cycle kinase mediated cellular proliferation
KR20020070520A (ko) 2000-01-27 2002-09-09 워너-램버트 캄파니 신경퇴행성 질병의 치료를 위한 피리도피리미디논 유도체
WO2014031571A1 (en) * 2012-08-21 2014-02-27 Icahn School Of Medicine At Mount Sinai Treatment of viral infections
WO2015179436A1 (en) 2014-05-19 2015-11-26 Sanford-Burnham Medical Research Institute Inflammation therapy using mekk3 inhibitors or blocking peptides
US11174255B2 (en) 2017-05-15 2021-11-16 University Of Houston System Pyrido[2,3-d]pyrimidin-7-ones and related compounds as inhibitors of protein kinases
EP4480485A3 (en) * 2019-05-16 2025-02-26 University of Houston System Protein kinase inhibitors and uses thereof for the treatment of diseases and conditions

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