JP2022524077A5 - - Google Patents

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Publication number
JP2022524077A5
JP2022524077A5 JP2021552999A JP2021552999A JP2022524077A5 JP 2022524077 A5 JP2022524077 A5 JP 2022524077A5 JP 2021552999 A JP2021552999 A JP 2021552999A JP 2021552999 A JP2021552999 A JP 2021552999A JP 2022524077 A5 JP2022524077 A5 JP 2022524077A5
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JP
Japan
Application number
JP2021552999A
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Japanese (ja)
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JP7663503B2 (ja
JPWO2020185593A5 (https=
JP2022524077A (ja
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Priority claimed from PCT/US2020/021479 external-priority patent/WO2020185593A1/en
Publication of JP2022524077A publication Critical patent/JP2022524077A/ja
Publication of JP2022524077A5 publication Critical patent/JP2022524077A5/ja
Publication of JPWO2020185593A5 publication Critical patent/JPWO2020185593A5/ja
Application granted granted Critical
Publication of JP7663503B2 publication Critical patent/JP7663503B2/ja
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JP2021552999A 2019-03-08 2020-03-06 アゼチジニルo-糖タンパク質-2-アセトアミド-2-デオキシ-3-d-グルコピラノシダーゼ阻害剤 Active JP7663503B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201962815553P 2019-03-08 2019-03-08
US62/815,553 2019-03-08
PCT/US2020/021479 WO2020185593A1 (en) 2019-03-08 2020-03-06 Azetidinyl 0-glyc0pr0tein-2-acetamid0-2-deoxy-3-d-gluc0pyran0sidase inhibitors

Publications (4)

Publication Number Publication Date
JP2022524077A JP2022524077A (ja) 2022-04-27
JP2022524077A5 true JP2022524077A5 (https=) 2023-03-14
JPWO2020185593A5 JPWO2020185593A5 (https=) 2023-03-14
JP7663503B2 JP7663503B2 (ja) 2025-04-16

Family

ID=69960768

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2021552999A Active JP7663503B2 (ja) 2019-03-08 2020-03-06 アゼチジニルo-糖タンパク質-2-アセトアミド-2-デオキシ-3-d-グルコピラノシダーゼ阻害剤

Country Status (5)

Country Link
US (1) US12421224B2 (https=)
EP (1) EP3935055A1 (https=)
JP (1) JP7663503B2 (https=)
MA (1) MA55203A (https=)
WO (1) WO2020185593A1 (https=)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN121405694A (zh) * 2024-07-26 2026-01-27 浙江同源康医药股份有限公司 Oga抑制剂及其应用

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4938949A (en) 1988-09-12 1990-07-03 University Of New York Treatment of damaged bone marrow and dosage units therefor
EP2780013A4 (en) 2011-11-18 2015-07-01 Constellation Pharmaceuticals Inc MODULATORS OF METHYL MODIFYING ENZYMES, COMPOSITIONS AND USES THEREOF
EP2780014A4 (en) 2011-11-18 2015-07-01 Constellation Pharmaceuticals Inc MODULATORS OF METHYL MODIFYING ENZYMES, COMPOSITIONS AND USES THEREOF
WO2013078320A1 (en) 2011-11-21 2013-05-30 Constellation Pharmaceuticals Modulators of methyl modifying enzymes, compositions and uses thereof
NZ628762A (en) 2012-02-10 2016-07-29 Constellation Pharmaceuticals Inc Modulators of methyl modifying enzymes, compositions and uses thereof
SI2953941T1 (sl) 2013-02-11 2017-08-31 Constellation Pharmaceuticals, Inc. Modulatorji metil-modificirajočih encimov, sestavki in uporabe le-teh
RS58768B1 (sr) * 2013-03-14 2019-06-28 Merck Patent Gmbh Inhibitori glikozidaze
WO2014151142A1 (en) 2013-03-15 2014-09-25 Constellation Pharmaceuticals, Inc. Modulators of methyl modifying enzymes, compositions and uses thereof
EP3033334A1 (en) 2013-08-15 2016-06-22 Constellation Pharmaceuticals, Inc. Indole derivatives as modulators of methyl modifying enzymes, compositions and uses thereof
CA3045957A1 (en) 2016-12-16 2018-06-21 Janssen Pharmaceutica Nv Monocyclic oga inhibitor compounds
WO2018154133A1 (en) 2017-02-27 2018-08-30 Janssen Pharmaceutica Nv [1,2,4]-triazolo [1,5-a]-pyrimidinyl derivatives substituted with piperidine, morpholine or piperazine as oga inhibitors

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