JP2022522942A5 - - Google Patents

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Publication number
JP2022522942A5
JP2022522942A5 JP2021539428A JP2021539428A JP2022522942A5 JP 2022522942 A5 JP2022522942 A5 JP 2022522942A5 JP 2021539428 A JP2021539428 A JP 2021539428A JP 2021539428 A JP2021539428 A JP 2021539428A JP 2022522942 A5 JP2022522942 A5 JP 2022522942A5
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JP
Japan
Prior art keywords
alkyl
tumor
formula
inflammation
related disorder
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2021539428A
Other languages
English (en)
Japanese (ja)
Other versions
JP7543278B2 (ja
JP2022522942A (ja
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Priority claimed from PCT/US2020/012578 external-priority patent/WO2020146384A1/en
Publication of JP2022522942A publication Critical patent/JP2022522942A/ja
Publication of JP2022522942A5 publication Critical patent/JP2022522942A5/ja
Priority to JP2024139639A priority Critical patent/JP7856707B2/ja
Application granted granted Critical
Publication of JP7543278B2 publication Critical patent/JP7543278B2/ja
Active legal-status Critical Current
Anticipated expiration legal-status Critical

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JP2021539428A 2019-01-07 2020-01-07 有機化合物 Active JP7543278B2 (ja)

Priority Applications (1)

Application Number Priority Date Filing Date Title
JP2024139639A JP7856707B2 (ja) 2019-01-07 2024-08-21 有機化合物

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201962789499P 2019-01-07 2019-01-07
US62/789,499 2019-01-07
PCT/US2020/012578 WO2020146384A1 (en) 2019-01-07 2020-01-07 Organic compounds

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2024139639A Division JP7856707B2 (ja) 2019-01-07 2024-08-21 有機化合物

Publications (3)

Publication Number Publication Date
JP2022522942A JP2022522942A (ja) 2022-04-21
JP2022522942A5 true JP2022522942A5 (cg-RX-API-DMAC10.html) 2022-12-19
JP7543278B2 JP7543278B2 (ja) 2024-09-02

Family

ID=71520889

Family Applications (2)

Application Number Title Priority Date Filing Date
JP2021539428A Active JP7543278B2 (ja) 2019-01-07 2020-01-07 有機化合物
JP2024139639A Active JP7856707B2 (ja) 2019-01-07 2024-08-21 有機化合物

Family Applications After (1)

Application Number Title Priority Date Filing Date
JP2024139639A Active JP7856707B2 (ja) 2019-01-07 2024-08-21 有機化合物

Country Status (4)

Country Link
US (2) US12396992B2 (cg-RX-API-DMAC10.html)
EP (1) EP3908285A4 (cg-RX-API-DMAC10.html)
JP (2) JP7543278B2 (cg-RX-API-DMAC10.html)
WO (1) WO2020146384A1 (cg-RX-API-DMAC10.html)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US11291666B2 (en) 2016-09-12 2022-04-05 Intra-Cellular Therapies, Inc. Uses
JP7493460B2 (ja) 2018-05-25 2024-05-31 イントラ-セルラー・セラピーズ・インコーポレイテッド 有機化合物
WO2020146384A1 (en) * 2019-01-07 2020-07-16 Intra-Cellular Therapies, Inc. Organic compounds
US12599603B2 (en) 2019-09-03 2026-04-14 Intra-Cellular Therapies, Inc. Methods of treatment
US12364695B2 (en) 2020-06-02 2025-07-22 Intra-Cellular Therapies, Inc. Methods of treating inflammatory disease
MX2024010993A (es) * 2022-03-11 2024-09-17 Intra Cellular Therapies Inc Compuestos organicos.

Family Cites Families (28)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4690935A (en) 1983-03-31 1987-09-01 Wayne State University Inhibition of tumor growth and metastasis with calcium channel blocker compounds
WO2006133261A2 (en) 2005-06-06 2006-12-14 Intra-Cellular Therapies, Inc. Organic compounds
EP2939676A1 (en) 2007-12-06 2015-11-04 Intra-Cellular Therapies, Inc. Organic compounds
EA201170769A1 (ru) 2008-12-06 2012-02-28 Интра-Селлулар Терапиз, Инк. Органические соединения
AU2009322903A1 (en) 2008-12-06 2010-06-10 Intra-Cellular Therapies, Inc. Organic compounds
US10695431B2 (en) 2010-10-29 2020-06-30 Infirst Healthcare Limited Solid solution compositions and use in cardiovascular disease
WO2012177263A1 (en) 2011-06-24 2012-12-27 Intra-Cellular Therapies, Inc. Compounds and methods of prophylaxis and treatment regarding nictonic receptor antagonists
JP6224597B2 (ja) 2011-09-27 2017-11-01 バイオメッド バレー ディスカバリーズ,インコーポレイティド グリオーマを処置するための組成物及び方法
WO2013138118A1 (en) 2012-03-14 2013-09-19 The Regents Of The University Of California Treatment of inflammatory disorders in non-human mammals
US9499562B2 (en) 2012-06-18 2016-11-22 Dart Neuroscience (Cayman) Ltd. Substituted thiophene- and furan-fused azolopyrimidine-5-(6H)-one compounds
DK2970279T3 (da) 2013-03-15 2020-11-30 Intra Cellular Therapies Inc Organiske forbindelser
ES2717688T3 (es) 2013-03-15 2019-06-24 Intra Cellular Therapies Inc Inhibidores de la PDE1 para uso en el tratamiento y/o prevención de lesiones de SNC, y enfermedades, trastornos o lesiones de SNP
JP6696904B2 (ja) * 2014-01-08 2020-05-20 イントラ−セルラー・セラピーズ・インコーポレイテッドIntra−Cellular Therapies, Inc. 製剤および医薬組成物
DK3157926T3 (da) 2014-06-20 2019-08-19 Intra Cellular Therapies Inc Organiske forbindelser
US10131671B2 (en) * 2014-08-07 2018-11-20 Intra-Cellular Therapies, Inc. Organic compounds
CA2961212C (en) 2014-09-17 2024-02-06 Intra-Cellular Therapies, Inc. Compounds and methods
US10849862B2 (en) 2014-12-26 2020-12-01 Theravalues Corporation Formulation of curcumin and anti-PD-1 antibody
EP3288980B1 (en) * 2015-04-28 2021-03-10 Bristol-Myers Squibb Company Treatment of pd-l1-positive melanoma using an anti-pd-1 antibody
CA2991628C (en) 2015-07-16 2020-04-07 Bioxcel Therapeutics, Inc. A novel approach for treatment of cancer using immunomodulation
US11291666B2 (en) 2016-09-12 2022-04-05 Intra-Cellular Therapies, Inc. Uses
MA46716A (fr) 2016-11-03 2019-09-11 Juno Therapeutics Inc Polythérapie de thérapie cellulaire et d'inhibiteur de la microglie
CA3047579A1 (en) 2016-12-22 2018-06-28 Abbvie Inc. Compositions and methods of enhancing or augmenting type i ifn production
AU2018325445A1 (en) 2017-08-31 2020-03-19 Abbvie Inc. Ectonucleotide pyrophosphatase-phosphodiesterase 1 (ENPP-1) inhibitors and uses thereof
JP7493460B2 (ja) 2018-05-25 2024-05-31 イントラ-セルラー・セラピーズ・インコーポレイテッド 有機化合物
EP3856191A4 (en) 2018-09-25 2022-06-22 Intra-Cellular Therapies, Inc. NOVEL USES
WO2020146384A1 (en) * 2019-01-07 2020-07-16 Intra-Cellular Therapies, Inc. Organic compounds
US12599603B2 (en) 2019-09-03 2026-04-14 Intra-Cellular Therapies, Inc. Methods of treatment
MX2024010993A (es) 2022-03-11 2024-09-17 Intra Cellular Therapies Inc Compuestos organicos.

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