JP2022521824A5 - - Google Patents
Info
- Publication number
- JP2022521824A5 JP2022521824A5 JP2021557651A JP2021557651A JP2022521824A5 JP 2022521824 A5 JP2022521824 A5 JP 2022521824A5 JP 2021557651 A JP2021557651 A JP 2021557651A JP 2021557651 A JP2021557651 A JP 2021557651A JP 2022521824 A5 JP2022521824 A5 JP 2022521824A5
- Authority
- JP
- Japan
- Prior art keywords
- alkyl
- optionally substituted
- inhibitor
- pharmaceutical composition
- combination according
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Ceased
Links
Applications Claiming Priority (7)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201962825450P | 2019-03-28 | 2019-03-28 | |
| US62/825,450 | 2019-03-28 | ||
| US201962842980P | 2019-05-03 | 2019-05-03 | |
| US62/842,980 | 2019-05-03 | ||
| US201962857519P | 2019-06-05 | 2019-06-05 | |
| US62/857,519 | 2019-06-05 | ||
| PCT/US2020/025539 WO2020198710A1 (en) | 2019-03-28 | 2020-03-27 | Pharmaceutical compositions and combinations comprising inhibitors of the androgen receptor and uses thereof |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2022521824A JP2022521824A (ja) | 2022-04-12 |
| JP2022521824A5 true JP2022521824A5 (enExample) | 2023-04-04 |
Family
ID=72610726
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2021557651A Ceased JP2022521824A (ja) | 2019-03-28 | 2020-03-27 | アンドロゲン受容体の阻害剤を含む薬学的組成物及びその組み合わせならびにその使用 |
Country Status (10)
| Country | Link |
|---|---|
| US (1) | US20220202780A1 (enExample) |
| EP (1) | EP3947353A4 (enExample) |
| JP (1) | JP2022521824A (enExample) |
| KR (1) | KR20210144827A (enExample) |
| CN (1) | CN114502539A (enExample) |
| AU (1) | AU2020248105A1 (enExample) |
| CA (1) | CA3134545A1 (enExample) |
| IL (1) | IL286726A (enExample) |
| MX (1) | MX2021011826A (enExample) |
| WO (1) | WO2020198710A1 (enExample) |
Families Citing this family (26)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US10471023B2 (en) | 2015-03-12 | 2019-11-12 | British Columbia Cancer Agency Branch | Bisphenol ether derivatives and methods for using the same |
| US20170298033A1 (en) | 2016-04-15 | 2017-10-19 | The University Of British Columbia | Bisphenol derivatives and their use as androgen receptor activity modulators |
| WO2019226991A1 (en) | 2018-05-25 | 2019-11-28 | Essa Pharma, Inc. | Androgen receptor modulators and methods for their use |
| EP3846793B1 (en) | 2018-09-07 | 2024-01-24 | PIC Therapeutics, Inc. | Eif4e inhibitors and uses thereof |
| US12637418B2 (en) | 2019-01-24 | 2026-05-26 | Takeda Pharmaceutical Company Limited | Heterocyclic compounds as antagonist of NMDA |
| US12109179B2 (en) | 2019-03-28 | 2024-10-08 | Essa Pharma Inc. | Pharmaceutical compositions and combinations comprising inhibitors of the androgen receptor and uses thereof |
| TWI873185B (zh) | 2019-09-16 | 2025-02-21 | 日商武田藥品工業股份有限公司 | 唑稠合之嗒-3(2h)-酮衍生物 |
| JP2021050161A (ja) | 2019-09-25 | 2021-04-01 | 武田薬品工業株式会社 | 複素環化合物及びその用途 |
| JP2021080177A (ja) | 2019-11-14 | 2021-05-27 | 武田薬品工業株式会社 | 複素環化合物及びその用途 |
| AR121506A1 (es) | 2020-03-03 | 2022-06-08 | Pic Therapeutics Inc | Inhibidores del eif4e y sus usos |
| EP4135675A4 (en) * | 2020-04-17 | 2024-04-10 | Essa Pharma, Inc. | SOLID FORMS OF AN N-TERMINAL DOMAIN ANDROGEN RECEPTOR INHIBITOR AND USES THEREOF |
| WO2022060969A1 (en) * | 2020-09-16 | 2022-03-24 | Essa Pharma, Inc. | Pharmaceutical compositions and combinations comprising inhibitors of the androgen receptor and uses thereof |
| WO2022169248A1 (ko) * | 2021-02-02 | 2022-08-11 | 주식회사 엘지화학 | 단백질 키나아제 억제제로서의 신규한 화합물 |
| CA3215182A1 (en) * | 2021-04-16 | 2022-10-20 | Han-Jie Zhou | Pharmaceutical compositions comprising inhibitors of the androgen receptor and uses thereof |
| CN115340527B (zh) * | 2021-05-13 | 2023-09-15 | 成都先导药物开发股份有限公司 | 一种bcl-xl抑制剂及其制备方法和用途 |
| CN113603695B (zh) * | 2021-08-05 | 2022-06-14 | 青岛恒宁生物科技有限公司 | 一种取代的嘧啶胺类化合物或其作为农药可接受的盐、组合物及其用途 |
| IL310924A (en) | 2021-08-25 | 2024-04-01 | Pic Therapeutics Inc | Eif4e inhibitors and uses thereof |
| US12157732B2 (en) | 2021-08-25 | 2024-12-03 | PIC Therapeutics, Inc. | eIF4E inhibitors and uses thereof |
| AU2022340817A1 (en) * | 2021-09-01 | 2024-03-14 | Essa Pharma Inc. | Pharmaceutical compositions and combinations comprising inhibitors of the androgen receptor and uses thereof |
| US20240398797A1 (en) * | 2021-09-01 | 2024-12-05 | Janssen Pharmaceutica Nv | Combination therapies for metastatic castration-resistant prostate cancer |
| WO2023151662A1 (zh) * | 2022-02-10 | 2023-08-17 | 上海奕拓医药科技有限责任公司 | 雄激素受体活性调节剂及其应用 |
| CN117065022A (zh) * | 2022-05-17 | 2023-11-17 | 海创药业股份有限公司 | 一种治疗三阴乳腺癌的药物 |
| WO2024006207A1 (en) * | 2022-06-26 | 2024-01-04 | Essa Pharma Inc. | An n-terminal domain androgen receptor inhibitor and uses thereof |
| EP4626878A1 (en) | 2022-12-02 | 2025-10-08 | Neumora Therapeutics, Inc. | Methods of treating neurological disorders |
| CN118255693A (zh) * | 2024-03-28 | 2024-06-28 | 大连理工大学 | 联苯类化合物及其在制备治疗白血病、肺癌以及乳腺癌药物中的应用 |
| CN121698845A (zh) * | 2024-09-12 | 2026-03-20 | 青岛普泰科生物医药科技有限公司 | 一种四氢喹啉类ntd抑制剂及其应用 |
Family Cites Families (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| BRPI0709771B1 (pt) * | 2006-03-27 | 2022-01-25 | The Regents Of The University Of California | Composto e composição farmacêutica |
| ES2613098T3 (es) * | 2011-08-19 | 2017-05-22 | British Columbia Cancer Agency Branch | Compuestos de éter de bisfenol fluorado y métodos para su uso |
| EP3733170A1 (en) * | 2012-07-13 | 2020-11-04 | Oncternal Therapeutics, Inc. | A method of treating androgen receptor (ar) -positive breast cancers with selective androgen receptor modulator (sarms) |
| FI3988541T3 (fi) * | 2015-01-13 | 2024-09-17 | British Columbia Cancer Agency Branch | Heterosyklisiä yhdisteitä syövän kuvantamiseksi ja hoitamiseksi ja menetelmiä niiden käyttämiseksi |
| US10980806B2 (en) * | 2016-03-24 | 2021-04-20 | University of Pittsburgh—of the Commonwealth System of Higher Education | Small molecule inhibitors of the nuclear translocation of androgen receptor for the treatment of castration-resistant prostate cancer |
| US20170298033A1 (en) * | 2016-04-15 | 2017-10-19 | The University Of British Columbia | Bisphenol derivatives and their use as androgen receptor activity modulators |
| WO2017223115A1 (en) * | 2016-06-22 | 2017-12-28 | Radius Health, Inc. | Ar+ breast cancer treatment methods |
| AU2019362061B2 (en) * | 2018-10-18 | 2024-09-26 | Essa Pharma Inc | Androgen receptor modulators and methods for their use |
-
2020
- 2020-03-27 WO PCT/US2020/025539 patent/WO2020198710A1/en not_active Ceased
- 2020-03-27 MX MX2021011826A patent/MX2021011826A/es unknown
- 2020-03-27 US US17/599,338 patent/US20220202780A1/en not_active Abandoned
- 2020-03-27 AU AU2020248105A patent/AU2020248105A1/en not_active Abandoned
- 2020-03-27 EP EP20779267.2A patent/EP3947353A4/en not_active Withdrawn
- 2020-03-27 KR KR1020217034804A patent/KR20210144827A/ko not_active Ceased
- 2020-03-27 CN CN202080039623.3A patent/CN114502539A/zh active Pending
- 2020-03-27 CA CA3134545A patent/CA3134545A1/en active Pending
- 2020-03-27 JP JP2021557651A patent/JP2022521824A/ja not_active Ceased
-
2021
- 2021-09-26 IL IL286726A patent/IL286726A/en unknown
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