JP2022517399A5 - - Google Patents
Info
- Publication number
- JP2022517399A5 JP2022517399A5 JP2021541187A JP2021541187A JP2022517399A5 JP 2022517399 A5 JP2022517399 A5 JP 2022517399A5 JP 2021541187 A JP2021541187 A JP 2021541187A JP 2021541187 A JP2021541187 A JP 2021541187A JP 2022517399 A5 JP2022517399 A5 JP 2022517399A5
- Authority
- JP
- Japan
- Prior art keywords
- referred
- sequence
- sar
- peptide ligand
- amino acid
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB1900530.5 | 2019-01-15 | ||
| GBGB1900530.5A GB201900530D0 (en) | 2019-01-15 | 2019-01-15 | Bicyclic peptide ligands specific for CD38 |
| PCT/GB2020/050074 WO2020148530A1 (en) | 2019-01-15 | 2020-01-15 | Bicyclic peptide ligands specific for cd38 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2022517399A JP2022517399A (ja) | 2022-03-08 |
| JP2022517399A5 true JP2022517399A5 (OSRAM) | 2023-01-25 |
Family
ID=65528178
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2021541187A Pending JP2022517399A (ja) | 2019-01-15 | 2020-01-15 | Cd38に特異的な二環式ペプチドリガンド |
Country Status (6)
| Country | Link |
|---|---|
| US (1) | US20220133733A1 (OSRAM) |
| EP (1) | EP3911366A1 (OSRAM) |
| JP (1) | JP2022517399A (OSRAM) |
| CN (1) | CN113597317A (OSRAM) |
| GB (1) | GB201900530D0 (OSRAM) |
| WO (1) | WO2020148530A1 (OSRAM) |
Families Citing this family (15)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| KR102754019B1 (ko) | 2014-10-29 | 2025-01-14 | 바이시클러드 리미티드 | Mt1-mmp에 특이적인 바이사이클릭 펩타이드 리간드 |
| CN111032678A (zh) | 2017-06-26 | 2020-04-17 | 拜西克尔德有限公司 | 具有可检测部分的双环肽配体和其用途 |
| ES2926195T3 (es) | 2017-08-04 | 2022-10-24 | Bicycletx Ltd | Ligandos peptídicos bicíclicos específicos de CD137 |
| AU2019224659A1 (en) | 2018-02-23 | 2020-10-15 | Bicycletx Limited | Multimeric bicyclic peptide ligands |
| US11180531B2 (en) | 2018-06-22 | 2021-11-23 | Bicycletx Limited | Bicyclic peptide ligands specific for Nectin-4 |
| GB201820295D0 (en) | 2018-12-13 | 2019-01-30 | Bicyclerd Ltd | Bicyclic peptide ligands specific for MT1-MMP |
| GB201820288D0 (en) | 2018-12-13 | 2019-01-30 | Bicycle Tx Ltd | Bicycle peptide ligaands specific for MT1-MMP |
| GB201820325D0 (en) | 2018-12-13 | 2019-01-30 | Bicyclerd Ltd | Bicyclic peptide ligands specific for psma |
| CN113474045A (zh) | 2018-12-21 | 2021-10-01 | 拜斯科技术开发有限公司 | Pd-l1特异性的双环肽配体 |
| US12551567B2 (en) | 2018-12-21 | 2026-02-17 | Bicyclerd Limited | Bicyclic peptide ligands specific for PD-L1 |
| GB201900529D0 (en) | 2019-01-15 | 2019-03-06 | Bicycletx Ltd | Bicyclic peptide ligands specific for CD38 |
| TWI860386B (zh) | 2019-07-30 | 2024-11-01 | 英商拜西可泰克斯有限公司 | 異質雙環肽複合物 |
| CA3189761A1 (en) | 2020-08-03 | 2022-02-10 | Gemma Mudd | Peptide-based linkers |
| GB202016331D0 (en) * | 2020-10-15 | 2020-12-02 | Bicyclerd Ltd | Bicyclic peptide ligand drug conjugates |
| CN118388598A (zh) * | 2024-04-22 | 2024-07-26 | 苏州大学附属第一医院 | 标记前体、探针及其制备方法和应用 |
Family Cites Families (11)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP1569956B1 (en) * | 2002-12-12 | 2014-02-26 | Tel Aviv University Future Technology Development L.P. | Glycogen synthase kinase-3 inhibitors |
| EP1452868A2 (en) | 2003-02-27 | 2004-09-01 | Pepscan Systems B.V. | Method for selecting a candidate drug compound |
| ES2541436T3 (es) | 2004-02-06 | 2015-07-20 | Morphosys Ag | Anticuerpos humanos anti-CD38 y usos para ellos |
| PT1844337E (pt) | 2005-01-24 | 2014-04-03 | Pepscan Systems Bv | Compostos ligantes, compostos imunogénicos e peptidomiméticos |
| EP3312196B1 (en) * | 2005-03-23 | 2019-07-17 | Genmab A/S | Antibodies against cd38 for treatment of multiple myeloma |
| WO2009098450A2 (en) | 2008-02-05 | 2009-08-13 | Medical Research Council | Methods and compositions |
| HUE045872T2 (hu) * | 2014-05-21 | 2020-01-28 | Entrada Therapeutics Inc | Sejteket penetráló peptidek és ezek elõállítására és alkalmazására szolgáló eljárások |
| KR102754019B1 (ko) | 2014-10-29 | 2025-01-14 | 바이시클러드 리미티드 | Mt1-mmp에 특이적인 바이사이클릭 펩타이드 리간드 |
| CN107810190A (zh) * | 2015-04-28 | 2018-03-16 | 洛桑联邦政府综合工科学校(Epfl) | 酶活化因子XII (FXIIa)的新型抑制剂 |
| CN111032678A (zh) * | 2017-06-26 | 2020-04-17 | 拜西克尔德有限公司 | 具有可检测部分的双环肽配体和其用途 |
| GB201810320D0 (en) * | 2018-06-22 | 2018-08-08 | Bicycletx Ltd | Peptide ligands for binding to CD38 |
-
2019
- 2019-01-15 GB GBGB1900530.5A patent/GB201900530D0/en not_active Ceased
-
2020
- 2020-01-15 US US17/422,943 patent/US20220133733A1/en not_active Abandoned
- 2020-01-15 JP JP2021541187A patent/JP2022517399A/ja active Pending
- 2020-01-15 CN CN202080021078.5A patent/CN113597317A/zh active Pending
- 2020-01-15 WO PCT/GB2020/050074 patent/WO2020148530A1/en not_active Ceased
- 2020-01-15 EP EP20701838.3A patent/EP3911366A1/en not_active Withdrawn
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