JP2022516631A5 - - Google Patents

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Publication number
JP2022516631A5
JP2022516631A5 JP2021538743A JP2021538743A JP2022516631A5 JP 2022516631 A5 JP2022516631 A5 JP 2022516631A5 JP 2021538743 A JP2021538743 A JP 2021538743A JP 2021538743 A JP2021538743 A JP 2021538743A JP 2022516631 A5 JP2022516631 A5 JP 2022516631A5
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JP
Japan
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alkyl
independently
disease
substituted
optionally
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JP2021538743A
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English (en)
Japanese (ja)
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JP2022516631A (ja
JP7566753B2 (ja
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Priority claimed from PCT/US2020/012268 external-priority patent/WO2020142748A1/en
Publication of JP2022516631A publication Critical patent/JP2022516631A/ja
Publication of JP2022516631A5 publication Critical patent/JP2022516631A5/ja
Application granted granted Critical
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JP2021538743A 2019-01-03 2020-01-03 転写因子ebポリペプチドレベルを増加させるための方法および材料 Active JP7566753B2 (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US201962788049P 2019-01-03 2019-01-03
US62/788,049 2019-01-03
US201962879374P 2019-07-26 2019-07-26
US62/879,374 2019-07-26
PCT/US2020/012268 WO2020142748A1 (en) 2019-01-03 2020-01-03 Methods and materials for increasing transcription factor eb polypeptide levels

Publications (3)

Publication Number Publication Date
JP2022516631A JP2022516631A (ja) 2022-03-01
JP2022516631A5 true JP2022516631A5 (https=) 2023-01-06
JP7566753B2 JP7566753B2 (ja) 2024-10-15

Family

ID=71406977

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2021538743A Active JP7566753B2 (ja) 2019-01-03 2020-01-03 転写因子ebポリペプチドレベルを増加させるための方法および材料

Country Status (12)

Country Link
US (2) US12286442B2 (https=)
EP (1) EP3906033A4 (https=)
JP (1) JP7566753B2 (https=)
KR (1) KR102904932B1 (https=)
CN (1) CN113316453B (https=)
AU (1) AU2020204717B2 (https=)
BR (1) BR112021012950A2 (https=)
CA (1) CA3123902A1 (https=)
IL (1) IL284403A (https=)
MX (1) MX2021008152A (https=)
SG (1) SG11202105685TA (https=)
WO (1) WO2020142748A1 (https=)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2023533016A (ja) 2020-07-11 2023-08-01 ファイザー・インク 抗ウイルス性ヘテロアリールケトン誘導体
US11351149B2 (en) 2020-09-03 2022-06-07 Pfizer Inc. Nitrile-containing antiviral compounds
CZ309449B6 (cs) * 2020-12-24 2023-01-25 Ústav experimentální botaniky AV ČR, v. v. i. Chinazolinové deriváty jako selektivní inhibitory cyklooxygenázy-1
CN113248518B (zh) * 2021-06-21 2022-03-25 山东大学 嘧啶哌嗪类衍生物及其制备方法与应用
CN121941701A (zh) * 2023-07-28 2026-04-28 特兰埃克斯公司 用于治疗溶酶体病症的突变tfeb
CN119818678A (zh) * 2024-12-24 2025-04-15 广州医科大学附属妇女儿童医疗中心 Tfeb在制备变应性鼻炎的药物中的应用

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US5304121A (en) 1990-12-28 1994-04-19 Boston Scientific Corporation Drug delivery system making use of a hydrogel polymer coating
US5886026A (en) 1993-07-19 1999-03-23 Angiotech Pharmaceuticals Inc. Anti-angiogenic compositions and methods of use
US6099562A (en) 1996-06-13 2000-08-08 Schneider (Usa) Inc. Drug coating with topcoat
WO2002022605A1 (en) * 2000-09-15 2002-03-21 Vertex Pharmaceuticals Incorporated Pyrazole compounds useful as protein kinase inhibitors
JP2005503425A (ja) 2001-05-24 2005-02-03 アレックザ モレキュラー デリヴァリー コーポレイション 所定の吸入ルートによる薬剤エステルの送出
US20030158195A1 (en) 2001-12-21 2003-08-21 Cywin Charles L. 1,6 naphthyridines useful as inhibitors of SYK kinase
AU2003286711A1 (en) * 2002-10-25 2004-05-13 Vertex Pharmaceuticals Incorporated Indazolinone compositions useful as kinase inhibitors
CL2004000409A1 (es) 2003-03-03 2005-01-07 Vertex Pharma Compuestos derivados de 2-(cilo sustituido)-1-(amino u oxi sustituido)-quinazolina, inhibidores de canales ionicos de sodio y calcio dependientes de voltaje; composicion farmaceutica; y uso del compuesto en el tratamiento de dolor agudo, cronico, neu
US7198926B2 (en) * 2003-05-08 2007-04-03 E. I. Du Pont De Nemours And Company Preparation of (E)- and (Z)-2-methyl-2-butenoic acids
EP1622615A4 (en) 2003-05-13 2009-02-18 Smithkline Beecham Corp INHIBITORS OF THE INTEGRASE OF NAPHTHYRIDINE
WO2008157500A1 (en) * 2007-06-17 2008-12-24 Kalypsys, Inc. Aminoquinazoline cannabinoid receptor modulators for treatment of disease
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GB201007203D0 (en) 2010-04-29 2010-06-16 Glaxo Group Ltd Novel compounds
GB201007347D0 (en) 2010-04-30 2010-06-16 Karus Therapeutics Ltd Compounds
CN104812387A (zh) 2012-11-20 2015-07-29 霍夫曼-拉罗奇有限公司 取代的1,6-萘啶
CN107205976A (zh) * 2014-11-19 2017-09-26 拉什大学医学中心 用于治疗溶酶体病症的组合物和方法
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WO2018191146A1 (en) * 2017-04-10 2018-10-18 Navitor Pharmaceuticals, Inc. Heteroaryl rheb inhibitors and uses thereof

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