JP2022510700A5 - - Google Patents

Info

Publication number
JP2022510700A5
JP2022510700A5 JP2021532119A JP2021532119A JP2022510700A5 JP 2022510700 A5 JP2022510700 A5 JP 2022510700A5 JP 2021532119 A JP2021532119 A JP 2021532119A JP 2021532119 A JP2021532119 A JP 2021532119A JP 2022510700 A5 JP2022510700 A5 JP 2022510700A5
Authority
JP
Japan
Prior art keywords
methyl
hydroxy
phenyl
oxo
dihydropyridine
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2021532119A
Other languages
English (en)
Japanese (ja)
Other versions
JP2022510700A (ja
Filing date
Publication date
Priority claimed from GBGB1819936.4A external-priority patent/GB201819936D0/en
Priority claimed from GBGB1904341.3A external-priority patent/GB201904341D0/en
Application filed filed Critical
Priority claimed from PCT/GB2019/053456 external-priority patent/WO2020115500A1/en
Publication of JP2022510700A publication Critical patent/JP2022510700A/ja
Publication of JP2022510700A5 publication Critical patent/JP2022510700A5/ja
Pending legal-status Critical Current

Links

JP2021532119A 2018-12-06 2019-12-06 治療において使用するusp19阻害剤 Pending JP2022510700A (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
GBGB1819936.4A GB201819936D0 (en) 2018-12-06 2018-12-06 Therapeutic methods
GB1819936.4 2018-12-06
GB1904341.3 2019-03-28
GBGB1904341.3A GB201904341D0 (en) 2019-03-28 2019-03-28 Therapeutic methods
PCT/GB2019/053456 WO2020115500A1 (en) 2018-12-06 2019-12-06 Usp19 inhibitors for use in therapy

Publications (2)

Publication Number Publication Date
JP2022510700A JP2022510700A (ja) 2022-01-27
JP2022510700A5 true JP2022510700A5 (enExample) 2023-01-11

Family

ID=68887434

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2021532119A Pending JP2022510700A (ja) 2018-12-06 2019-12-06 治療において使用するusp19阻害剤

Country Status (12)

Country Link
US (1) US20220016115A1 (enExample)
EP (1) EP3890737B1 (enExample)
JP (1) JP2022510700A (enExample)
KR (1) KR20210100127A (enExample)
CN (1) CN113395965A (enExample)
AU (1) AU2019393161A1 (enExample)
BR (1) BR112021010645A2 (enExample)
CA (1) CA3121422A1 (enExample)
IL (1) IL283687A (enExample)
MX (1) MX2021006542A (enExample)
SG (1) SG11202105911PA (enExample)
WO (1) WO2020115500A1 (enExample)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP3965749A4 (en) * 2019-05-06 2023-06-21 Valo Health, Inc. ESCAPEMENT OF USP19
GB202104097D0 (en) * 2021-03-24 2021-05-05 Almac Discovery Ltd Pharmaceutical compounds
GB202311227D0 (en) 2023-07-21 2023-09-06 Almac Discovery Ltd Pharmaceutical compounds

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AUPO111096A0 (en) * 1996-07-18 1996-08-08 Fujisawa Pharmaceutical Co., Ltd. New compound
AR069526A1 (es) 2007-12-03 2010-01-27 Takeda Pharmaceutical Compuesto heterociclico que contiene nitrogeno y su uso
CN104174021A (zh) * 2013-05-22 2014-12-03 复旦大学附属华山医院 蛋白酶体抑制剂在制备治疗慢性低度炎症性疾病药物中的用途
AR103297A1 (es) * 2014-12-30 2017-05-03 Forma Therapeutics Inc Pirrolo y pirazolopirimidinas como inhibidores de la proteasa 7 específica de ubiquitina
GB201612938D0 (en) * 2016-07-26 2016-09-07 Almac Discovery Ltd Pharmaceutical compounds
JP7402792B2 (ja) * 2017-09-26 2023-12-21 デイナ ファーバー キャンサー インスティチュート,インコーポレイテッド 多発性骨髄腫を治療するための新規なusp7阻害剤
GB201801562D0 (en) * 2018-01-31 2018-03-14 Almac Diagnostics Ltd Pharmaceutical compounds

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