JP2022507533A5 - - Google Patents

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Publication number
JP2022507533A5
JP2022507533A5 JP2021526561A JP2021526561A JP2022507533A5 JP 2022507533 A5 JP2022507533 A5 JP 2022507533A5 JP 2021526561 A JP2021526561 A JP 2021526561A JP 2021526561 A JP2021526561 A JP 2021526561A JP 2022507533 A5 JP2022507533 A5 JP 2022507533A5
Authority
JP
Japan
Prior art keywords
compound
pharmaceutically acceptable
acceptable salt
diazaspiro
trifluoroethoxy
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2021526561A
Other languages
English (en)
Japanese (ja)
Other versions
JP2022507533A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/IB2019/001224 external-priority patent/WO2020099926A1/en
Publication of JP2022507533A publication Critical patent/JP2022507533A/ja
Publication of JP2022507533A5 publication Critical patent/JP2022507533A5/ja
Priority to JP2023217954A priority Critical patent/JP2024019691A/ja
Pending legal-status Critical Current

Links

JP2021526561A 2018-11-16 2019-11-15 肺動脈性高血圧症および他疾患に関連する肺動脈性肺高血圧症の治療法 Pending JP2022507533A (ja)

Priority Applications (1)

Application Number Priority Date Filing Date Title
JP2023217954A JP2024019691A (ja) 2018-11-16 2023-12-25 肺動脈性高血圧症および他疾患に関連する肺動脈性肺高血圧症の治療法

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201862768575P 2018-11-16 2018-11-16
US62/768,575 2018-11-16
PCT/IB2019/001224 WO2020099926A1 (en) 2018-11-16 2019-11-15 A method for treating pulmonary arterial hypertension and associated pulmonary arterial hypertension

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2023217954A Division JP2024019691A (ja) 2018-11-16 2023-12-25 肺動脈性高血圧症および他疾患に関連する肺動脈性肺高血圧症の治療法

Publications (2)

Publication Number Publication Date
JP2022507533A JP2022507533A (ja) 2022-01-18
JP2022507533A5 true JP2022507533A5 (enExample) 2022-10-05

Family

ID=69182543

Family Applications (2)

Application Number Title Priority Date Filing Date
JP2021526561A Pending JP2022507533A (ja) 2018-11-16 2019-11-15 肺動脈性高血圧症および他疾患に関連する肺動脈性肺高血圧症の治療法
JP2023217954A Pending JP2024019691A (ja) 2018-11-16 2023-12-25 肺動脈性高血圧症および他疾患に関連する肺動脈性肺高血圧症の治療法

Family Applications After (1)

Application Number Title Priority Date Filing Date
JP2023217954A Pending JP2024019691A (ja) 2018-11-16 2023-12-25 肺動脈性高血圧症および他疾患に関連する肺動脈性肺高血圧症の治療法

Country Status (8)

Country Link
US (2) US11413287B2 (enExample)
EP (1) EP3880203A1 (enExample)
JP (2) JP2022507533A (enExample)
KR (1) KR20210105343A (enExample)
CN (1) CN113242736A (enExample)
AU (1) AU2019382168A1 (enExample)
CA (1) CA3119909A1 (enExample)
WO (1) WO2020099926A1 (enExample)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU2019382168A1 (en) 2018-11-16 2021-06-03 Altavant Sciences Gmbh A method for treating pulmonary arterial hypertension and associated pulmonary arterial hypertension
WO2020128614A1 (en) * 2018-12-17 2020-06-25 Altavant Sciences Gmbh Method for treating interstital lung disease
CN113557022A (zh) 2019-01-30 2021-10-26 阿尔塔万特科学公司 用罗达司他乙酯治疗肺动脉高压的给药方案和方法
CN113784717A (zh) * 2019-03-15 2021-12-10 阿尔塔万特科学公司 一种治疗肺动脉高压和相关性肺动脉高压的方法以及每日给药
WO2023062595A1 (en) 2021-10-14 2023-04-20 Altavant Sciences Gmbh Treatment of subjects having pulmonary arterial hypertension with rodatristat ethyl

Family Cites Families (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN101815534A (zh) 2007-07-11 2010-08-25 莱西肯医药有限公司 用于治疗肺动脉高压以及相关疾病和病症的方法和组合物
TW201245183A (en) * 2010-11-05 2012-11-16 Lexicon Pharmaceuticals Inc Solid forms of (S)-2-amino-3-(4-(2-amino-6-((R)-1-(4-chloro-2-(3-methyl-1H-pyrazol-1-yl)phenyl)-2,2,2-trifluoroethoxy)pyrimidin-4-yl)phenyl)propanoic acid
UA119247C2 (uk) * 2013-09-06 2019-05-27 РОЙВЕНТ САЙЕНСИЗ ҐмбГ Спіроциклічні сполуки як інгібітори триптофангідроксилази
US9399741B2 (en) 2013-10-09 2016-07-26 Uop Llc Methods and apparatuses for desulfurizing hydrocarbon streams
KR20210102887A (ko) * 2018-11-14 2021-08-20 알타반트 사이언시스 게엠베하 말초 세로토닌과 관련된 질병 또는 장애를 치료하기 위한 트립토판 하이드록실라제 1 (tph1)의 결정질 스피로사이클릭 화합물 억제제
AU2019382168A1 (en) 2018-11-16 2021-06-03 Altavant Sciences Gmbh A method for treating pulmonary arterial hypertension and associated pulmonary arterial hypertension
US20200188398A1 (en) * 2018-12-17 2020-06-18 Altavant Sciences Gmbh Method for treating sarcoidosis-associated pulmonary hypertension
WO2020128614A1 (en) * 2018-12-17 2020-06-25 Altavant Sciences Gmbh Method for treating interstital lung disease
CN113557022A (zh) * 2019-01-30 2021-10-26 阿尔塔万特科学公司 用罗达司他乙酯治疗肺动脉高压的给药方案和方法
CN113784717A (zh) 2019-03-15 2021-12-10 阿尔塔万特科学公司 一种治疗肺动脉高压和相关性肺动脉高压的方法以及每日给药
JP2023512025A (ja) 2020-01-31 2023-03-23 アルタバント・サイエンシズ・ゲーエムベーハー 肺動脈性肺高血圧症をロダトリスタットで処置するための投与量および方法
US11937070B2 (en) 2021-07-01 2024-03-19 Tencent America LLC Layered description of space of interest
WO2023079486A1 (en) 2021-11-03 2023-05-11 Altavant Sciences Gmbh Treatment of pulmonary arterial hypertension with rodatristat and ambrisentan

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