JP2022500351A5 - - Google Patents

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Publication number
JP2022500351A5
JP2022500351A5 JP2020567621A JP2020567621A JP2022500351A5 JP 2022500351 A5 JP2022500351 A5 JP 2022500351A5 JP 2020567621 A JP2020567621 A JP 2020567621A JP 2020567621 A JP2020567621 A JP 2020567621A JP 2022500351 A5 JP2022500351 A5 JP 2022500351A5
Authority
JP
Japan
Prior art keywords
pharmaceutically acceptable
hydroxypiperidine
bipyridine
methanone
benzyl
Prior art date
Application number
JP2020567621A
Other languages
English (en)
Japanese (ja)
Other versions
JP7443255B2 (ja
JPWO2020059894A5 (https=
JP2022500351A (ja
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Publication date
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Priority claimed from PCT/JP2019/038061 external-priority patent/WO2020059894A1/en
Publication of JP2022500351A publication Critical patent/JP2022500351A/ja
Publication of JP2022500351A5 publication Critical patent/JP2022500351A5/ja
Publication of JPWO2020059894A5 publication Critical patent/JPWO2020059894A5/ja
Application granted granted Critical
Publication of JP7443255B2 publication Critical patent/JP7443255B2/ja
Active legal-status Critical Current
Anticipated expiration legal-status Critical

Links

JP2020567621A 2018-09-20 2019-09-19 疼痛使用のためのch24h阻害剤 Active JP7443255B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201862733927P 2018-09-20 2018-09-20
US62/733,927 2018-09-20
PCT/JP2019/038061 WO2020059894A1 (en) 2018-09-20 2019-09-19 CH24H Inhibitors For Pain Use

Publications (4)

Publication Number Publication Date
JP2022500351A JP2022500351A (ja) 2022-01-04
JP2022500351A5 true JP2022500351A5 (https=) 2022-09-20
JPWO2020059894A5 JPWO2020059894A5 (https=) 2022-09-20
JP7443255B2 JP7443255B2 (ja) 2024-03-05

Family

ID=68343384

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2020567621A Active JP7443255B2 (ja) 2018-09-20 2019-09-19 疼痛使用のためのch24h阻害剤

Country Status (4)

Country Link
US (1) US20210346366A1 (https=)
EP (1) EP3852757A1 (https=)
JP (1) JP7443255B2 (https=)
WO (1) WO2020059894A1 (https=)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2025126159A1 (en) * 2023-12-15 2025-06-19 Takeda Pharmaceutical Company Limited A method for treating a neurological disease in a recreational drug user

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PL2763979T3 (pl) * 2011-10-07 2019-06-28 Takeda Pharmaceutical Company Limited Związki 1-arylokarbonyl-4-oksy-piperydynowe użyteczne do leczenia chorób neurodegeneracyjnych
EP3904332B1 (en) 2011-10-14 2024-12-04 The United States of America, as represented by The Secretary, Department of Health and Human Services The use of (2r, 6r)-hydroxynorketamine, (s)-dehydronorketamine and other stereoisomeric dehydro and hydroxylated metabolites of (r,s)- ketamine in the treatment of depression and neuropathic pain
PE20151162A1 (es) 2012-12-11 2015-08-28 Takeda Pharmaceutical Compuestos heterociclicos inhibidores del colesterol 24-hidroxilasa (ch24h)
CN105164161A (zh) * 2013-03-13 2015-12-16 萨奇治疗股份有限公司 神经活性类固醇、组合物、及其用途
JP6272832B2 (ja) * 2013-04-04 2018-01-31 武田薬品工業株式会社 複素環化合物
EP3152198B1 (en) 2014-06-09 2019-02-27 Takeda Pharmaceutical Company Limited Radiolabeled compounds

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