JP2022132411A5 - - Google Patents
Download PDFInfo
- Publication number
- JP2022132411A5 JP2022132411A5 JP2022112389A JP2022112389A JP2022132411A5 JP 2022132411 A5 JP2022132411 A5 JP 2022132411A5 JP 2022112389 A JP2022112389 A JP 2022112389A JP 2022112389 A JP2022112389 A JP 2022112389A JP 2022132411 A5 JP2022132411 A5 JP 2022132411A5
- Authority
- JP
- Japan
- Prior art keywords
- salt
- quinolin
- thiophen
- piperazin
- benzo
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
- 150000003839 salts Chemical class 0.000 claims 2
- 239000004480 active ingredient Substances 0.000 claims 1
- ZKIAIYBUSXZPLP-UHFFFAOYSA-N brexpiprazole Chemical compound C1=C2NC(=O)C=CC2=CC=C1OCCCCN(CC1)CCN1C1=CC=CC2=C1C=CS2 ZKIAIYBUSXZPLP-UHFFFAOYSA-N 0.000 claims 1
- 238000013270 controlled release Methods 0.000 claims 1
- 239000008194 pharmaceutical composition Substances 0.000 claims 1
- 239000000546 pharmaceutical excipient Substances 0.000 claims 1
- 239000007787 solid Substances 0.000 claims 1
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2025027501A JP2025074104A (ja) | 2019-08-13 | 2025-02-25 | 経口医薬組成物 |
Applications Claiming Priority (4)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| PCT/JP2019/031895 WO2021029020A1 (ja) | 2019-08-13 | 2019-08-13 | 経口医薬組成物 |
| JPPCT/JP2019/031895 | 2019-08-13 | ||
| PCT/JP2020/030776 WO2021029429A1 (ja) | 2019-08-13 | 2020-08-13 | 経口医薬組成物 |
| JP2021539311A JP7110495B2 (ja) | 2019-08-13 | 2020-08-13 | 経口医薬組成物 |
Related Parent Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2021539311A Division JP7110495B2 (ja) | 2019-08-13 | 2020-08-13 | 経口医薬組成物 |
Related Child Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2025027501A Division JP2025074104A (ja) | 2019-08-13 | 2025-02-25 | 経口医薬組成物 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2022132411A JP2022132411A (ja) | 2022-09-08 |
| JP2022132411A5 true JP2022132411A5 (https=) | 2023-08-21 |
Family
ID=74569440
Family Applications (7)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2021539751A Withdrawn JPWO2021029020A1 (https=) | 2019-08-13 | 2019-08-13 | |
| JP2021539311A Active JP7110495B2 (ja) | 2019-08-13 | 2020-08-13 | 経口医薬組成物 |
| JP2021539312A Active JP7148733B2 (ja) | 2019-08-13 | 2020-08-13 | 複素環化合物を含有する経口医薬組成物 |
| JP2022112389A Pending JP2022132411A (ja) | 2019-08-13 | 2022-07-13 | 経口医薬組成物 |
| JP2022150733A Active JP7635187B2 (ja) | 2019-08-13 | 2022-09-21 | 複素環化合物を含有する経口医薬組成物 |
| JP2025020427A Pending JP2025072595A (ja) | 2019-08-13 | 2025-02-12 | 複素環化合物を含有する経口医薬組成物 |
| JP2025027501A Pending JP2025074104A (ja) | 2019-08-13 | 2025-02-25 | 経口医薬組成物 |
Family Applications Before (3)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2021539751A Withdrawn JPWO2021029020A1 (https=) | 2019-08-13 | 2019-08-13 | |
| JP2021539311A Active JP7110495B2 (ja) | 2019-08-13 | 2020-08-13 | 経口医薬組成物 |
| JP2021539312A Active JP7148733B2 (ja) | 2019-08-13 | 2020-08-13 | 複素環化合物を含有する経口医薬組成物 |
Family Applications After (3)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2022150733A Active JP7635187B2 (ja) | 2019-08-13 | 2022-09-21 | 複素環化合物を含有する経口医薬組成物 |
| JP2025020427A Pending JP2025072595A (ja) | 2019-08-13 | 2025-02-12 | 複素環化合物を含有する経口医薬組成物 |
| JP2025027501A Pending JP2025074104A (ja) | 2019-08-13 | 2025-02-25 | 経口医薬組成物 |
Country Status (15)
| Country | Link |
|---|---|
| US (4) | US20220273647A1 (https=) |
| EP (2) | EP4015001A4 (https=) |
| JP (7) | JPWO2021029020A1 (https=) |
| KR (2) | KR20220046625A (https=) |
| CN (2) | CN114222562A (https=) |
| AU (2) | AU2020328351B2 (https=) |
| BR (2) | BR112022002433A2 (https=) |
| CA (2) | CA3150751A1 (https=) |
| IL (2) | IL290469B2 (https=) |
| MX (3) | MX2022001758A (https=) |
| MY (2) | MY208261A (https=) |
| PH (2) | PH12022550347A1 (https=) |
| TW (2) | TWI870441B (https=) |
| WO (3) | WO2021029020A1 (https=) |
| ZA (2) | ZA202202319B (https=) |
Families Citing this family (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2021029020A1 (ja) * | 2019-08-13 | 2021-02-18 | 大塚製薬株式会社 | 経口医薬組成物 |
| CN118742293A (zh) * | 2022-01-31 | 2024-10-01 | 住友精化株式会社 | 药物控释制剂用组合物和药物控释制剂 |
| JP2023173950A (ja) * | 2022-05-27 | 2023-12-07 | 同仁医薬化工株式会社 | 経口液剤 |
| AU2024247059A1 (en) * | 2023-03-29 | 2025-10-30 | Merck Sharp & Dohme (Uk) Limited | Controlled release pde10a formulations |
Family Cites Families (23)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US2799241A (en) | 1949-01-21 | 1957-07-16 | Wisconsin Alumni Res Found | Means for applying coatings to tablets or the like |
| US3173876A (en) | 1960-05-27 | 1965-03-16 | John C Zobrist | Cleaning methods and compositions |
| NL271831A (https=) | 1960-11-29 | |||
| US3276586A (en) | 1963-08-30 | 1966-10-04 | Rosaen Filter Co | Indicating means for fluid filters |
| US3546142A (en) | 1967-01-19 | 1970-12-08 | Amicon Corp | Polyelectrolyte structures |
| US3541006A (en) | 1968-07-03 | 1970-11-17 | Amicon Corp | Ultrafiltration process |
| US3541005A (en) | 1969-02-05 | 1970-11-17 | Amicon Corp | Continuous ultrafiltration of macromolecular solutions |
| US3865108A (en) | 1971-05-17 | 1975-02-11 | Ortho Pharma Corp | Expandable drug delivery device |
| US3916899A (en) | 1973-04-25 | 1975-11-04 | Alza Corp | Osmotic dispensing device with maximum and minimum sizes for the passageway |
| US4002173A (en) | 1974-07-23 | 1977-01-11 | International Paper Company | Diester crosslinked polyglucan hydrogels and reticulated sponges thereof |
| GB1478759A (en) | 1974-11-18 | 1977-07-06 | Alza Corp | Process for forming outlet passageways in pills using a laser |
| US4207893A (en) | 1977-08-29 | 1980-06-17 | Alza Corporation | Device using hydrophilic polymer for delivering drug to biological environment |
| TWI320783B (en) * | 2005-04-14 | 2010-02-21 | Otsuka Pharma Co Ltd | Heterocyclic compound |
| JP4315393B2 (ja) | 2005-04-14 | 2009-08-19 | 大塚製薬株式会社 | 複素環化合物 |
| JP4540700B2 (ja) * | 2006-10-13 | 2010-09-08 | 大塚製薬株式会社 | 医薬 |
| JOP20120083B1 (ar) * | 2011-04-05 | 2021-08-17 | Otsuka Pharma Co Ltd | توليفات تشتمل على بريكس ببرازول أو ملح منه وعقار ثاني للاستخدام في علاج اضطراب cns |
| JO3753B1 (ar) * | 2011-10-14 | 2021-01-31 | Otsuka Pharma Co Ltd | قرص يتألف من 7-[4-(4-بينزو[بي]ثيوفين-4-ايل-ببرازين-1-1ايل)بوتكسيل]-1اتش-كوينولين-2-وان أو ملح منه |
| TWI632921B (zh) * | 2011-10-19 | 2018-08-21 | 大塚製藥股份有限公司 | 口服溶液 |
| AR090775A1 (es) * | 2012-04-23 | 2014-12-03 | Otsuka Pharma Co Ltd | Preparado inyectable |
| EP2911670A1 (en) * | 2012-10-25 | 2015-09-02 | Otsuka Pharmaceutical Co., Ltd. | Prophylactic and/or therapeutic agent for behavioral and psychological symptoms associated with neurodegenerative disease or impulsive symptoms associated with mental disease containing brexpiprazole or salt thereof |
| CN106667969A (zh) * | 2017-02-23 | 2017-05-17 | 佛山市弘泰药物研发有限公司 | 一种依匹哌唑缓释胶囊及其制备方法 |
| JP6886654B2 (ja) | 2017-04-11 | 2021-06-16 | 学校法人帝京大学 | 抗カンジダ活性組成物 |
| WO2021029020A1 (ja) * | 2019-08-13 | 2021-02-18 | 大塚製薬株式会社 | 経口医薬組成物 |
-
2019
- 2019-08-13 WO PCT/JP2019/031895 patent/WO2021029020A1/ja not_active Ceased
- 2019-08-13 JP JP2021539751A patent/JPWO2021029020A1/ja not_active Withdrawn
-
2020
- 2020-08-13 WO PCT/JP2020/030777 patent/WO2021029430A1/ja not_active Ceased
- 2020-08-13 EP EP20853189.7A patent/EP4015001A4/en active Pending
- 2020-08-13 AU AU2020328351A patent/AU2020328351B2/en active Active
- 2020-08-13 MY MYPI2022000768A patent/MY208261A/en unknown
- 2020-08-13 PH PH1/2022/550347A patent/PH12022550347A1/en unknown
- 2020-08-13 KR KR1020227007745A patent/KR20220046625A/ko active Pending
- 2020-08-13 US US17/634,758 patent/US20220273647A1/en not_active Abandoned
- 2020-08-13 CA CA3150751A patent/CA3150751A1/en active Pending
- 2020-08-13 US US17/634,791 patent/US20220280418A1/en not_active Abandoned
- 2020-08-13 CN CN202080056803.2A patent/CN114222562A/zh active Pending
- 2020-08-13 JP JP2021539311A patent/JP7110495B2/ja active Active
- 2020-08-13 WO PCT/JP2020/030776 patent/WO2021029429A1/ja not_active Ceased
- 2020-08-13 TW TW109127608A patent/TWI870441B/zh active
- 2020-08-13 BR BR112022002433A patent/BR112022002433A2/pt unknown
- 2020-08-13 IL IL290469A patent/IL290469B2/en unknown
- 2020-08-13 CN CN202080056806.6A patent/CN114222575A/zh active Pending
- 2020-08-13 BR BR112022002436A patent/BR112022002436A2/pt unknown
- 2020-08-13 PH PH1/2022/550349A patent/PH12022550349B1/en unknown
- 2020-08-13 KR KR1020227007743A patent/KR20220046624A/ko active Pending
- 2020-08-13 JP JP2021539312A patent/JP7148733B2/ja active Active
- 2020-08-13 CA CA3150827A patent/CA3150827A1/en active Pending
- 2020-08-13 TW TW109127609A patent/TWI870442B/zh active
- 2020-08-13 MY MYPI2022000781A patent/MY208267A/en unknown
- 2020-08-13 AU AU2020327792A patent/AU2020327792B2/en active Active
- 2020-08-13 MX MX2022001758A patent/MX2022001758A/es unknown
- 2020-08-13 EP EP20853069.1A patent/EP4015002A4/en active Pending
- 2020-08-13 MX MX2022001759A patent/MX2022001759A/es unknown
-
2022
- 2022-02-09 IL IL290472A patent/IL290472A/en unknown
- 2022-02-10 MX MX2025006039A patent/MX2025006039A/es unknown
- 2022-02-23 ZA ZA2022/02319A patent/ZA202202319B/en unknown
- 2022-02-23 ZA ZA2022/02320A patent/ZA202202320B/en unknown
- 2022-07-13 JP JP2022112389A patent/JP2022132411A/ja active Pending
- 2022-09-21 JP JP2022150733A patent/JP7635187B2/ja active Active
-
2024
- 2024-08-26 US US18/815,060 patent/US20250127776A1/en active Pending
- 2024-09-18 US US18/888,277 patent/US20250057835A1/en active Pending
-
2025
- 2025-02-12 JP JP2025020427A patent/JP2025072595A/ja active Pending
- 2025-02-25 JP JP2025027501A patent/JP2025074104A/ja active Pending
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| JP2022132411A5 (https=) | ||
| JP2011201907A5 (https=) | ||
| HRP20210487T1 (hr) | Farmaceutski sastavi koji sadrže lokalni anestetik kao što je bupivakain za lokalnu primjenu u usta ili grlo | |
| JP2012255026A5 (https=) | ||
| JP2006516570A5 (https=) | ||
| JP2009535352A5 (https=) | ||
| JP2018168191A5 (https=) | ||
| JP2015078230A5 (https=) | ||
| HRP20171793T1 (hr) | Farmaceutske formulacije koje sadrže kristalne oblike (r)-7-kloro-n-(kinuklidin-3-il)benzo(b)tiofen-2-karboksamid hidroklorid monohidrata | |
| JP2015523407A5 (https=) | ||
| MY181645A (en) | Antibacterial quinoline derivatives | |
| JP2007533687A (ja) | 月経前の及び他の女性の性的障害の治療におけるフリバンセリンの使用 | |
| CN115315423A (zh) | 取代芳基类化合物 | |
| MX2021002259A (es) | Formas cristalinas de 3-(imidazo[1,2-b] piridazin-3- iletinil)-4-metil-n-(4-[(4-metilpiperazin-1-il) metil]-3-(trifluorometil)fenil) benzamida y su sal de monoclorhidrato. | |
| JP2019536812A5 (https=) | ||
| JP2026021451A5 (https=) | ||
| JP2000159790A5 (https=) | ||
| JP2008516004A5 (https=) | ||
| EA200901146A1 (ru) | Твердые лекарственные формы, содержащие алискирен и его фармацевтически приемлемые соли | |
| JP2012508256A5 (https=) | ||
| JP2006507295A5 (https=) | ||
| JP2010500284A5 (https=) | ||
| NO20070952L (no) | Formuleringer av suberoylanilidhydroksaminsyre og fremgangsmate for fremstilling av slike | |
| JPWO2024181437A5 (https=) | ||
| WO2009084041A3 (en) | Pharmaceutical compositions of dexibuprofen |